Compile Data Set for Download or QSAR
maximum 50k data
Found 6 of ic50 for monomerid = 50307932
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50307932(CHEMBL597402 | N-(4-(3-Bromoanilino)quinazolin-6-y...)
Affinity DataIC50:  23.6nMAssay Description:Inhibition of human recombinant EGFR expressed in insect cells by time-resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50307932(CHEMBL597402 | N-(4-(3-Bromoanilino)quinazolin-6-y...)
Affinity DataIC50:  24nMAssay Description:Inhibition of wild type human EGFR tyrosine kinase assessed as Ulight-CAGAGAIETDKEYYTVKD phosphorylation after 15 mins by time-resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50307932(CHEMBL597402 | N-(4-(3-Bromoanilino)quinazolin-6-y...)
Affinity DataIC50:  50nMAssay Description:Inhibition of wild type EGFR autophosphorylation in human A549 cells incubated for 1 hr followed by compound washout measured at 1 hr by Western blot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50307932(CHEMBL597402 | N-(4-(3-Bromoanilino)quinazolin-6-y...)
Affinity DataIC50:  78nMAssay Description:Inhibition of EGFR autophosphorylation in human A431 cells after 8 hrs by western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50307932(CHEMBL597402 | N-(4-(3-Bromoanilino)quinazolin-6-y...)
Affinity DataIC50:  84nMAssay Description:Inhibition of EGFR autophosphorylation in human A431 cells after 1 hr by western blotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50307932(CHEMBL597402 | N-(4-(3-Bromoanilino)quinazolin-6-y...)
Affinity DataIC50:  118nMAssay Description:Inhibition of wild type EGFR autophosphorylation in human A549 cells incubated for 1 hr followed by compound washout measured after 8 hrs by Western ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed