Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM238895'
TargetAndrogen receptor(Homo sapiens (Human))
The Regents of The University of California

US Patent
LigandPNGBDBM238895(US10053433, Casodex (CDX) | US10053433, FC 4.037 (...)
Affinity DataIC50:  15nMpH: 7.5Assay Description:Briefly, the AR LBD is expressed as a fusion with the Gal4 transcription factor, which binds to the Gal4 reporter DNA. Upon activation with agonist h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
The Regents of The University of California

US Patent
LigandPNGBDBM238895(US10053433, Casodex (CDX) | US10053433, FC 4.037 (...)
Affinity DataIC50:  190nMpH: 7.5Assay Description:An AR-response element is contained within the mmTV sequence and drives the expression of luciferase. The effect of antiandrogens (competitive antago...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
The Regents of The University of California

US Patent
LigandPNGBDBM238895(US10053433, Casodex (CDX) | US10053433, FC 4.037 (...)
Affinity DataIC50:  360nMpH: 7.5Assay Description:Briefly, the AR LBD is expressed as a fusion with the Gal4 transcription factor, which binds to the Gal4 reporter DNA. Upon activation with agonist h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
The Regents of The University of California

US Patent
LigandPNGBDBM238895(US10053433, Casodex (CDX) | US10053433, FC 4.037 (...)
Affinity DataIC50:  1.00E+3nMpH: 7.5Assay Description:An AR-response element is contained within the mmTV sequence and drives the expression of luciferase. The effect of antiandrogens (competitive antago...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent