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Found 3 Enz. Inhib. hit(s) with Target = 'Arginase-1' and Ligand = 'BDBM130381'
TargetArginase-1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM130381((R)-2-amino-6-borono-2-[1-(3,4-dichlorobenzyl)pipe...)
Affinity DataIC50:  18nMAssay Description:Inhibition of human arginase1 in presence of DNTB by thio ornithine generation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM130381((R)-2-amino-6-borono-2-[1-(3,4-dichlorobenzyl)pipe...)
Affinity DataIC50:  200nMAssay Description:Inhibition of recombinant human ARG1 expressed in Escherichia coli using L-arginine hydrochloride as substrate incubated for 1 hr by colorimetric ass...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetArginase-1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM130381((R)-2-amino-6-borono-2-[1-(3,4-dichlorobenzyl)pipe...)
Affinity DataIC50:  509nMAssay Description:Inhibition of recombinant human ARG1 expressed in Escherichia coli using L-arginine hydrochloride as substrate incubated for 1 hr by colorimetric ass...More data for this Ligand-Target Pair
In DepthDetails PubMed