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Found 2 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM24307'
TargetAromatase(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM24307(Letrozole derivative, 40a R-(+) | {2-bromo-4-[(R)-...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of aromatase (unknown origin) expressed in JEG-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM24307(Letrozole derivative, 40a R-(+) | {2-bromo-4-[(R)-...)
Affinity DataIC50:  3.20nMpH: 7.5 T: 2°CAssay Description:The extent of in vitro inhibition of aromatase activities was assessed using intact monolayers of JEG-3 cells. Aromatase activity was measured using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed