Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'C-X-C chemokine receptor type 2' and Ligand = 'BDBM50302100'
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Wuxi Pharmatech

Curated by ChEMBL
LigandPNGBDBM50302100(3-(2-(2-acetyl-2-ethylhydrazinyl)-3,4-dioxocyclobu...)
Affinity DataKi:  320nMAssay Description:Displacement of [125I]IL-8 from human CXCR2 expressed in mouse BaF3 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Wuxi Pharmatech

Curated by ChEMBL
LigandPNGBDBM50302100(3-(2-(2-acetyl-2-ethylhydrazinyl)-3,4-dioxocyclobu...)
Affinity DataIC50:  1.25E+3nMAssay Description:Antagonist activity at CXCR2 expressed in CHO cells assessed as inhibition of IL-8-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Wuxi Pharmatech

Curated by ChEMBL
LigandPNGBDBM50302100(3-(2-(2-acetyl-2-ethylhydrazinyl)-3,4-dioxocyclobu...)
Affinity DataIC50:  3.29E+3nMAssay Description:Displacement of [125I]IL-8 from human CXCR2 expressed in mouse BaF3 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed