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Found 4 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM239078'
TargetCannabinoid receptor 1(Mus musculus (Mouse))
University of Arkansas

US Patent
LigandPNGBDBM239078(US9416103, TV-5-157)
Affinity DataKi:  1.70nMAssay Description:A functional assay screen for the inhibition of adenylate cyclase (AC) activity was chosen as the subsequent assay. This screen would allow us to gai...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Mus musculus (Mouse))
University of Arkansas

US Patent
LigandPNGBDBM239078(US9416103, TV-5-157)
Affinity DataKi:  1.70nMAssay Description:Agonist activity at CB1 receptor in mouse Neuro2a cells assessed as inhibition of forskolin-stimulated adenylyl cyclase activity after 15 mins by liq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
University of Arkansas

US Patent
LigandPNGBDBM239078(US9416103, TV-5-157)
Affinity DataIC50:  45nMAssay Description:Agonist activity at CB1 receptor in mouse Neuro2a cells assessed as inhibition of forskolin-stimulated adenylyl cyclase activity after 15 mins by liq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
University of Arkansas

US Patent
LigandPNGBDBM239078(US9416103, TV-5-157)
Affinity DataIC50:  45nMAssay Description:A functional assay screen for the inhibition of adenylate cyclase (AC) activity was chosen as the subsequent assay. This screen would allow us to gai...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent