Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Diacylglycerol O-acyltransferase 1' and Ligand = 'BDBM20730'
TargetDiacylglycerol O-acyltransferase 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM20730((1R,2R)-2-{[4-(3-fluoro-4-{[6-(trifluoromethoxy)-1...)
Affinity DataIC50:  73nMpH: 7.5 T: 2°CAssay Description:DGAT-1 activity was characterized by catalyzing the transfer of the radiolabeled decanoyl group onto the syn-3 position of didecanoyl glycerol. The r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 1(Mus musculus (mouse))
Abbott Laboratories

LigandPNGBDBM20730((1R,2R)-2-{[4-(3-fluoro-4-{[6-(trifluoromethoxy)-1...)
Affinity DataIC50:  207nMpH: 7.5 T: 2°CAssay Description:DGAT-1 activity was characterized by catalyzing the transfer of the radiolabeled decanoyl group onto the syn-3 position of didecanoyl glycerol. The r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed