Found 1 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase p300/Hypoxia-inducible factor 1-alpha' and Ligand = 'BDBM50537295'
TargetHistone acetyltransferase p300/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 3.50E+3nMAssay Description:Inhibition of HIF-1alpha (786 to 826 residues) (unknown origin)/p300 (unknown origin) protein-protein interaction by ITCMore data for this Ligand-Target Pair