Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50169772'
TargetKappa-type opioid receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169772((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-methoxymeth...)
Affinity DataKi:  0.400nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169772((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-methoxymeth...)
Affinity DataKi:  0.400nMAssay Description:Agonistic activity against human k-opioid receptor using [3H]diprenorphineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169772((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-methoxymeth...)
Affinity DataEC50:  0.600nMAssay Description:Activation of human k-opioid receptor as increased [35S]GTPcS binding More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50169772((3S,4aR,6S,8R,8aR,10aR)-3-Furan-3-yl-6-methoxymeth...)
Affinity DataEC50:  0.600nMAssay Description:Activation of human k-opioid receptor as increased [35S]GTPcS binding More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed