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Found 2 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase 1' and Ligand = 'BDBM495257'
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Agv Discovery

US Patent
LigandPNGBDBM495257(1-(3-Fluoro-4-(trifluoromethyl)benzyl)-4-(5-morpho...)
Affinity DataIC50: <10nMAssay Description:To assess compounds capacity to inhibit ERK2 enzymatic activity, Z′-Lyte biochemical assay from Life technologies was used according to manufac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Agv Discovery

US Patent
LigandPNGBDBM495257(1-(3-Fluoro-4-(trifluoromethyl)benzyl)-4-(5-morpho...)
Affinity DataIC50: <150nMAssay Description:To assess compounds capacity to inhibit ERK2 enzymatic activity, Z′-Lyte biochemical assay from Life technologies was used according to manufac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent