Found 1 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 8' and Ligand = 'BDBM3175'
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 9.95E+3nMAssay Description:Inhibition of human COT1 using MEK1 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair