Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 1 group I member 3' and Ligand = 'BDBM50185306'
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Palacky University In Olomouc

Curated by ChEMBL
LigandPNGBDBM50185306(CHEMBL3823873)
Affinity DataEC50:  690nMAssay Description:Agonist activity at CAR LBD (108 to 348 residues) expressed in human HepG2 cells assessed as receptor binding to PGC1alpha by lanthascreenTR-FRET coa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 3(Homo sapiens (Human))
Palacky University In Olomouc

Curated by ChEMBL
LigandPNGBDBM50185306(CHEMBL3823873)
Affinity DataEC50:  6.12E+3nMAssay Description:Agonist activity at human CAR3 expressed in African green monkey COS-1 cells cotransfected with RXRalpha after 24 hrs by CYP2B6-luciferase reporter g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed