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Found 2 Enz. Inhib. hit(s) with Target = 'Oxysterols receptor LXR-beta' and Ligand = 'BDBM50298704'
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50298704(CHEMBL585552 | N-(4-(2-Phenylethyl)phenyl)phthalim...)
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity at human LXR-beta transfected in HEK293 cells after 16 hrs by luciferase reporter gene assay in presence of 0.1 uM N-(4-(1,1,1,3,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50298704(CHEMBL585552 | N-(4-(2-Phenylethyl)phenyl)phthalim...)
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity at human LXRbeta expressed in HEK293 cells assessed as inhibition of beta-galactosidase activity by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed