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Found 11 Enz. Inhib. hit(s) with Target = 'P2X purinoceptor 4' and Ligand = 'BDBM50399183'
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of East Anglia

Curated by ChEMBL
LigandPNGBDBM50399183(CHEMBL2180160)
Affinity DataIC50:  420nMAssay Description:Antagonist activity at human P2X4R transfected in 1321N1 cells assessed as inhibition of ATP-mediated calcium influx measured after 10 mins by Fura-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of East Anglia

Curated by ChEMBL
LigandPNGBDBM50399183(CHEMBL2180160)
Affinity DataIC50:  420nMAssay Description:Antagonist activity at human P2X4R transfected in 1321N1 cells assessed as inhibition of ATP-mediated calcium influx measured after 10 mins by Fura-2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of East Anglia

Curated by ChEMBL
LigandPNGBDBM50399183(CHEMBL2180160)
Affinity DataIC50:  760nMAssay Description:Antagonist activity at human P2X4R transfected in HEK293 cells assessed as inhibition of ATP-mediated calcium influx measured after 10 mins by YOPRO-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of East Anglia

Curated by ChEMBL
LigandPNGBDBM50399183(CHEMBL2180160)
Affinity DataIC50:  760nMAssay Description:Antagonist activity at human P2X4R transfected in HEK293 cells assessed as inhibition of ATP-mediated calcium influx measured after 10 mins by YOPRO-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50399183(CHEMBL2180160)
Affinity DataIC50:  928nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of East Anglia

Curated by ChEMBL
LigandPNGBDBM50399183(CHEMBL2180160)
Affinity DataIC50:  1.38E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of East Anglia

Curated by ChEMBL
LigandPNGBDBM50399183(CHEMBL2180160)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at human P2X4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of East Anglia

Curated by ChEMBL
LigandPNGBDBM50399183(CHEMBL2180160)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at human P2X4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50399183(CHEMBL2180160)
Affinity DataIC50:  1.76E+3nMAssay Description:Antagonist activity at mouse P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of East Anglia

Curated by ChEMBL
LigandPNGBDBM50399183(CHEMBL2180160)
Affinity DataIC50:  3.30E+3nMAssay Description:Antagonist activity at human P2X4R transfected in 1321N1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of East Anglia

Curated by ChEMBL
LigandPNGBDBM50399183(CHEMBL2180160)
Affinity DataIC50:  3.30E+3nMAssay Description:Antagonist activity at human P2X4R transfected in 1321N1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed