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Found 2 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50097814'
LigandPNGBDBM50097814((S)-2-[(5-{[(1H-Imidazol-4-ylmethyl)-amino]-methyl...)
Affinity DataIC50:  20nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097814((S)-2-[(5-{[(1H-Imidazol-4-ylmethyl)-amino]-methyl...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed