Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50126323'
LigandPNGBDBM50126323(1-{3-[3-(4-Cyano-benzyl)-3H-imidazol-4-yl]-propion...)
Affinity DataIC50:  1.40nMAssay Description:In vitro inhibition of farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126323(1-{3-[3-(4-Cyano-benzyl)-3H-imidazol-4-yl]-propion...)
Affinity DataEC50:  28nMAssay Description:Inhibition of Ras farnesylation in Human Ha-Ras oncogene-transformed BALB/c 3T3 cells (EJ3 cells)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed