Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Protein-arginine deiminase type-4' and Ligand = 'BDBM454162'
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM454162(BDBM50246174 | US10716791, Code KP-286)
Affinity DataKi:  8.80E+4nMAssay Description:Inhibition of full length human GST-tagged PAD4 expressed in baculovirus infected Sf9 insect cells preincubated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
University of Toronto

Curated by ChEMBL
LigandPNGBDBM454162(BDBM50246174 | US10716791, Code KP-286)
Affinity DataKi:  7.14E+5nMAssay Description:Materials: PAD1, PAD2, PAD3 and PAD4 were purchased from commercial sources. Assay buffer: 50 mM Tris pH 7.5, 100 mM NaCl, 10 mM CaCl2, 5 mM DTT. Col...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent