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Found 1 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50313264'
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50313264(CHEMBL1087773 | N-(3-(4-(2,3-dimethylphenyl)pipera...)
Affinity DataIC50:  53.6nMAssay Description:Displacement of [3H]imipramine from human SERT expressed in HEK293 cells after 30 mins by rapid filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed