Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50101416'
TargetSubstance-P receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50101416(CHEMBL307488 | [(R)-2-(3H-Indol-3-yl)-1-methyl-1-(...)
Affinity DataIC50:  0.550nMAssay Description:Binding affinity towards tachykinin receptor 1 in human IM9 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50101416(CHEMBL307488 | [(R)-2-(3H-Indol-3-yl)-1-methyl-1-(...)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at NK1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50101416(CHEMBL307488 | [(R)-2-(3H-Indol-3-yl)-1-methyl-1-(...)
Affinity DataIC50:  1.05nMAssay Description:Inhibition of specific binding at tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50101416(CHEMBL307488 | [(R)-2-(3H-Indol-3-yl)-1-methyl-1-(...)
Affinity DataIC50:  5.90nMAssay Description:In vitro affinity for specific binding at Gerbil tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed