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Found 2 Enz. Inhib. hit(s) with Target = 'Synaptic vesicular amine transporter' and Ligand = 'BDBM50171947'
TargetSynaptic vesicular amine transporter(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50171947((2R,6S)-1-Methyl-2,6-bis-(2-naphthalen-1-yl-ethyl)...)
Affinity DataKi:  630nMAssay Description:Binding affinity to VMAT2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50171947((2R,6S)-1-Methyl-2,6-bis-(2-naphthalen-1-yl-ethyl)...)
Affinity DataKi:  630nMAssay Description:Inhibition of 5 nM [3H]DTBZ binding to Vesicular Monoamine Transporter (VAMT2) of rat vesicle membranes More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed