Found 4 Enz. Inhib. hit(s) with Target = 'Transcriptional activator protein LuxR' and Ligand = 'BDBM50266163'
Affinity DataIC50: 600nMAssay Description:Antagonist activity against LuxR mediated quorum sensing system in Vibrio fischeri ES114 expressing luxI assessed as decrease in luminescence intensi...More data for this Ligand-Target Pair
Affinity DataIC50: 860nMAssay Description:Antagonist activity at Vibrio fischeri ES114 LuxR receptor assessed as inhibition of OHHL-induced response by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 860nMAssay Description:Antagonist activity at Vibrio fischeri luxR receptor in presence of 5 uM 3-oxo-C6-HSLMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Antagonist activity at Aliivibrio fischeri ES114 LuxR after 4 to 8 hrs by luminescence methodMore data for this Ligand-Target Pair