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Found 7 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 8285
TargetCannabinoid receptor 1(Mus musculus (Mouse))
University of Arkansas

US Patent
LigandPNGBDBM239073(US9416103, CP-55,940)
Affinity DataKi:  0.370nM ΔG°:  -53.8kJ/moleT: 2°CAssay Description:Competition receptor binding was performed as previously described [Shoemaker et al., J. Pharmacol. Exp. Ther., 314:868-75]. Briefly, 50 μg of mou...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Mus musculus (Mouse))
University of Arkansas

US Patent
LigandPNGBDBM85804(1-Naphthyl(1-butyl-1H-indole-3-yl)methanone | JWH-...)
Affinity DataKi:  12.9nM ΔG°:  -45.0kJ/moleT: 2°CAssay Description:Competition receptor binding was performed as previously described [Shoemaker et al., J. Pharmacol. Exp. Ther., 314:868-75]. Briefly, 50 μg of mou...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Mus musculus (Mouse))
University of Arkansas

US Patent
LigandPNGBDBM239074(US9416103, JWH-073-M1)
Affinity DataKi:  14.1nM ΔG°:  -44.8kJ/moleT: 2°CAssay Description:Competition receptor binding was performed as previously described [Shoemaker et al., J. Pharmacol. Exp. Ther., 314:868-75]. Briefly, 50 μg of mou...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Mus musculus (Mouse))
University of Arkansas

US Patent
LigandPNGBDBM239075(US9416103, JWH-073-M4)
Affinity DataKi:  122nM ΔG°:  -39.5kJ/moleT: 2°CAssay Description:Competition receptor binding was performed as previously described [Shoemaker et al., J. Pharmacol. Exp. Ther., 314:868-75]. Briefly, 50 μg of mou...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Mus musculus (Mouse))
University of Arkansas

US Patent
LigandPNGBDBM60993(US9416103, JWH-073-M5)
Affinity DataKi:  224nM ΔG°:  -38.0kJ/moleT: 2°CAssay Description:Competition receptor binding was performed as previously described [Shoemaker et al., J. Pharmacol. Exp. Ther., 314:868-75]. Briefly, 50 μg of mou...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 2(Homo sapiens (Human))
University of Arkansas

US Patent
LigandPNGBDBM239075(US9416103, JWH-073-M4)
Affinity DataKi:  251nM ΔG°:  -37.7kJ/moleT: 2°CAssay Description:Competition receptor binding was performed as previously described [Shoemaker et al., J. Pharmacol. Exp. Ther., 314:868-75]. Briefly, 50 μg of mou...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Mus musculus (Mouse))
University of Arkansas

US Patent
LigandPNGBDBM60992(US9416103, JWH-073-M3)
Affinity DataKi:  1.28E+3nM ΔG°:  -33.6kJ/moleT: 2°CAssay Description:Competition receptor binding was performed as previously described [Shoemaker et al., J. Pharmacol. Exp. Ther., 314:868-75]. Briefly, 50 μg of mou...More data for this Ligand-Target Pair
In DepthDetails US Patent