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Found 587 with Last Name = 'cui' and Initial = 'g'
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50172545((2-Iodo-phenyl)-[1-((S)-1-methyl-piperidin-2-ylmet...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity towards mouse hippocampal membranes cannabinoid receptor 1 using [131I]-(R)-8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50172553(CHEMBL68641 | [1-(1-Methyl-piperidin-2-ylmethyl)-1...)
Affinity DataKi:  0.75nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50172545((2-Iodo-phenyl)-[1-((S)-1-methyl-piperidin-2-ylmet...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity towards mouse hippocampal membranes cannabinoid receptor 1 using [3H]SR-141,716AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity towards mouse hippocampal membranes cannabinoid receptor 1 using [131I]-(R)-8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50172553(CHEMBL68641 | [1-(1-Methyl-piperidin-2-ylmethyl)-1...)
Affinity DataKi:  1.91nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50172545((2-Iodo-phenyl)-[1-((S)-1-methyl-piperidin-2-ylmet...)
Affinity DataKi:  2.80nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50172545((2-Iodo-phenyl)-[1-((S)-1-methyl-piperidin-2-ylmet...)
Affinity DataKi:  2.90nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50174549((4-Iodo-naphthalen-1-yl)-[1-(1-methyl-piperidin-2-...)
Affinity DataKi:  5.30nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50314706((R)-2-(2-naphthamido)-5-(3-fluorophenyl)pent-4-eno...)
Affinity DataKi:  6nMAssay Description:Inhibition of N-terminal His tagged human Pin1 expressed in Escherichia coli BL21 (DE3) using Suc-Ala-Glu-Pro-Phe-4-nitroanilide as substrate preincu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM34012(3-fluorophenylalanine derivative, 21b)
Affinity DataKi:  6nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50174548((2-Iodo-phenyl)-[2-methyl-1-(1-methyl-piperidin-2-...)
Affinity DataKi:  6.70nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50174547(CHEMBL436120 | [6-Iodo-1-(1-methyl-piperidin-2-ylm...)
Affinity DataKi:  9.80nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50174549((4-Iodo-naphthalen-1-yl)-[1-(1-methyl-piperidin-2-...)
Affinity DataKi:  10nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50174548((2-Iodo-phenyl)-[2-methyl-1-(1-methyl-piperidin-2-...)
Affinity DataKi:  10nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50174547(CHEMBL436120 | [6-Iodo-1-(1-methyl-piperidin-2-ylm...)
Affinity DataKi:  18nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50552327(CHEMBL4751817)
Affinity DataKi:  20nMAssay Description:Inhibition of GST-tagged Pin1 (unknown origin) using Suc-Ala-pSer-Pro-Phe-pNA as substrate preincubated with enzyme for 12 hrs followed by substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  20nMAssay Description:Binding affinity towards mouse hippocampal membranes cannabinoid receptor 1 using [3H]SR-141,716AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50174548((2-Iodo-phenyl)-[2-methyl-1-(1-methyl-piperidin-2-...)
Affinity DataKi:  34nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50174548((2-Iodo-phenyl)-[2-methyl-1-(1-methyl-piperidin-2-...)
Affinity DataKi:  34nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50174548((2-Iodo-phenyl)-[2-methyl-1-(1-methyl-piperidin-2-...)
Affinity DataKi:  34nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50174548((2-Iodo-phenyl)-[2-methyl-1-(1-methyl-piperidin-2-...)
Affinity DataKi:  34nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50552328(CHEMBL4750217)
Affinity DataKi:  48nMAssay Description:Inhibition of GST-tagged Pin1 (unknown origin) using Suc-Ala-pSer-Pro-Phe-pNA as substrate preincubated with enzyme for 12 hrs followed by substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50535516(CHEMBL4542964)
Affinity DataKi:  60nMAssay Description:Inhibition of Escherichia coli PDFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50370681(CHEMBL1788276)
Affinity DataKi:  560nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50370681(CHEMBL1788276)
Affinity DataKi:  580nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50174546((4-Iodo-phenyl)-[2-methyl-1-(1-methyl-piperidin-2-...)
Affinity DataKi:  790nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  820nMAssay Description:Inhibition of GST-tagged Pin1 (unknown origin) using Suc-Ala-pSer-Pro-Phe-pNA, Suc-Ala-Glu-Pro-Phe-pNA or Suc-Ala-Ala-Pro-Phe-pNA as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50174546((4-Iodo-phenyl)-[2-methyl-1-(1-methyl-piperidin-2-...)
Affinity DataKi:  1.80E+3nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50174545((3-Iodo-phenyl)-[2-methyl-1-(1-methyl-piperidin-2-...)
Affinity DataKi:  2.90E+3nMAssay Description:Binding affinity towards rat forebrain cannabinoid receptor 1 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50174545((3-Iodo-phenyl)-[2-methyl-1-(1-methyl-piperidin-2-...)
Affinity DataKi:  9.60E+3nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 using [3H]CP-55940More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50535514(CHEMBL4458398)
Affinity DataIC50:  0.630nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50535509(CHEMBL4457234)
Affinity DataIC50:  1nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50268281(CHEMBL4067999)
Affinity DataIC50:  1nMAssay Description:Inhibition of recombinant human PARP-2 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50535505(CHEMBL4462876)
Affinity DataIC50:  1nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50535513(CHEMBL4572153)
Affinity DataIC50:  1nMAssay Description:Inhibition of Staphylococcus aureus PDF by fluorescence detection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50268281(CHEMBL4067999)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of recombinant human PARP-1 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of recombinant human PARP-2 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
TargetPeptide deformylase(Staphylococcus aureus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50535512(CHEMBL4434997)
Affinity DataIC50:  2nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50535508(CHEMBL4518477)
Affinity DataIC50:  2nMAssay Description:Inhibition of Staphylococcus aureus PDF by fluorescence detection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50535497(CHEMBL4466084)
Affinity DataIC50:  2nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50535515(CHEMBL4559778)
Affinity DataIC50:  2nMAssay Description:Inhibition of Staphylococcus aureus PDF by fluorescence detection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50535500(CHEMBL4568739)
Affinity DataIC50:  2nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50535518(CHEMBL4448951)
Affinity DataIC50:  2nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50268267(CHEMBL4083291)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of recombinant human PARP-2 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50535504(CHEMBL4565584)
Affinity DataIC50:  3nMAssay Description:Inhibition of Staphylococcus aureus PDF by fluorescence detection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50268267(CHEMBL4083291)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of recombinant human PARP-1 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50268268(CHEMBL4061458)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of recombinant human PARP-2 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50268284(CHEMBL4100719)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of recombinant human PARP-2 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 2(Homo sapiens (Human))
Chinese Academy Of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50268277(CHEMBL4072243)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of recombinant human PARP-2 expressed in Escherichia coli BL21 (DE3) using sheared DNA as substrate in presence of biotinylated NAD after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50535501(CHEMBL4435970)
Affinity DataIC50:  5nMAssay Description:Inhibition of Staphylococcus aureus PDF by absorbance detection assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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