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Found 24 with Last Name = 'pomponi' and Initial = 'sa'
TargetCaspase-3(Homo sapiens (Human))
Harbor Branch Oceanographic Institution

Curated by ChEMBL
LigandPNGBDBM50478882(SECOBATZELLINE A)
Affinity DataIC50:  78.2nMAssay Description:Inhibition of peptidase activity of CPP32More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286606((4aS,12bR)-11-Chloro-10-hydroxy-4,4,4a,12b-tetrame...)
Affinity DataIC50:  300nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50127868(CHEMBL299895 | Sterol sulfate)
Affinity DataIC50:  480nMAssay Description:Binding affinity against Purinergic receptor P2Y12 using [3H]-2-methylthio-ADP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50070217(3-(3-Bromo-4-methoxy-phenyl)-2-[(E)-hydroxyimino]-...)
Affinity DataIC50:  500nMAssay Description:Binding affinity to histamine H3 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50276581((+/-)-wiedendiol B | CHEMBL456619)
Affinity DataIC50:  600nMAssay Description:Compound was tested for CETP inhibition by a precipitation method to separate lipoproteins after incubation of radiolabeled HDL with LDL and CETP.More data for this Ligand-Target Pair
In DepthDetails Article
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Harbor Branch Oceanographic Institution

Curated by ChEMBL
LigandPNGBDBM50478457(PLAKOLIDE A)
Affinity DataIC50:  723nMAssay Description:Inhibition of iNOS-mediated NO production in LPS-stimulated mouse RAW264.7 cells by Griess methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
Harbor Branch Oceanographic Institution

Curated by ChEMBL
LigandPNGBDBM50478844(DISCORHABDIN | Discorhabdin P | Discorhabdine C)
Affinity DataIC50:  775nMAssay Description:Inhibition of CPP32 peptidase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285079(4-Methoxy-3-((S)-2,5,5,8a-tetramethyl-3,4,4a,5,6,7...)
Affinity DataIC50:  1.00E+3nMAssay Description:Compound was tested for CETP inhibition by a precipitation method to separate lipoproteins after incubation of radiolabeled HDL with LDL and CETP.More data for this Ligand-Target Pair
In DepthDetails Article
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50127869(CHEMBL299307 | Sterol sulfate)
Affinity DataIC50:  2.20E+3nMAssay Description:Binding affinity against Purinergic receptor P2Y12 using [3H]-2-methylthio-ADP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
Harbor Branch Oceanographic Institution

Curated by ChEMBL
LigandPNGBDBM50478883(Secobatzelline A Diacetate)
Affinity DataIC50:  2.35E+3nMAssay Description:Inhibition of peptidase activity of CPP32More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50276581((+/-)-wiedendiol B | CHEMBL456619)
Affinity DataIC50:  5.00E+3nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285079(4-Methoxy-3-((S)-2,5,5,8a-tetramethyl-3,4,4a,5,6,7...)
Affinity DataIC50:  5.00E+3nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50240865((4aS,6aS,12aR,12bS)-10-Hydroxy-4,4,6a,12b-tetramet...)
Affinity DataIC50:  6.00E+3nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50292430(CHEMBL479515 | aerophobin-1)
Affinity DataIC50:  9.00E+3nMAssay Description:Binding affinity to histamine H3 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50292440(Aplysiillin A | CHEMBL462733)
Affinity DataIC50:  2.00E+4nMAssay Description:Displacement of [125I]thrombin from thrombin receptor in human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286611(5,5,9,10-tetramethyl-18-oxatetracyclo[8.8.0.01,6.0...)
Affinity DataIC50:  2.20E+4nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286609(1-((4aS,12bR)-9,10-Diacetyl-4,4,4a,12b-tetramethyl...)
Affinity DataIC50:  2.30E+4nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50242257(2-((1R,2S,4aS)-1,2,4a,5-Tetramethyl-1,2,3,4,4a,7,8...)
Affinity DataIC50:  2.50E+4nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-3(Homo sapiens (Human))
Harbor Branch Oceanographic Institution

Curated by ChEMBL
LigandPNGBDBM50478884(Secobatzelline B Diacetate)
Affinity DataIC50:  2.58E+4nMAssay Description:Inhibition of peptidase activity of CPP32More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50292412(34-sulfatobastadin 13 | CHEMBL465400)
Affinity DataIC50:  3.90E+4nMAssay Description:Displacement of [125]ET1 from ETA receptor in pig thoracic aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286610(13-methoxy-5,5,9,10-tetramethyl-18-oxatetracyclo[8...)
Affinity DataIC50:  4.60E+4nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50240866((-)-ilimaquinone | 2-Hydroxy-5-methoxy-3-((1R,2S,4...)
Affinity DataIC50:  1.00E+5nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286608(CHEMBL60072 | Sulfircin analogue | Sulfuric acid m...)
Affinity DataIC50: >1.90E+5nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286607((3bR,5aR,6S,7S,9aR,9bR)-7-Hydroxy-6-hydroxymethyl-...)
Affinity DataIC50:  1.96E+5nMAssay Description:Compound was tested for Cholesteryl ester transfer protein (CETP) inhibition by CETP-SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article