Compile Data Set for Download or QSAR
maximum 50k data
Found 50 with Last Name = 'moir' and Initial = 'em'
TargetCytochrome P450 3A4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332241((S)-(1-(cyclohexylmethyl)-7-methoxy-1H-indol-3-yl)...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332241((S)-(1-(cyclohexylmethyl)-7-methoxy-1H-indol-3-yl)...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human CYP2C19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332241((S)-(1-(cyclohexylmethyl)-7-methoxy-1H-indol-3-yl)...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50332241((S)-(1-(cyclohexylmethyl)-7-methoxy-1H-indol-3-yl)...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417559(CHEMBL1642163)
Affinity DataEC50:  2.51E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417560(CHEMBL1642164)
Affinity DataEC50:  2.51E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417561(CHEMBL1642165)
Affinity DataEC50:  1.00E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417562(CHEMBL1642166)
Affinity DataEC50:  398nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417563(CHEMBL1642167)
Affinity DataEC50:  7.94E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417564(CHEMBL1642168)
Affinity DataEC50:  100nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417565(CHEMBL1642169)
Affinity DataEC50:  158nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417566(CHEMBL1642170)
Affinity DataEC50:  501nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417567(CHEMBL1642171)
Affinity DataEC50:  2.00E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417568(CHEMBL1642172)
Affinity DataEC50:  1.26E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417569(CHEMBL1642150)
Affinity DataEC50:  398nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417570(CHEMBL1642152)
Affinity DataEC50: >3.16E+4nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417571(CHEMBL1232932)
Affinity DataEC50:  501nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417572(CHEMBL1642153)
Affinity DataEC50:  1.26E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417573(CHEMBL1642154)
Affinity DataEC50:  1.26E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417574(CHEMBL1642155)
Affinity DataEC50:  100nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417089(CHEMBL1257768)
Affinity DataEC50:  1.58E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417576(CHEMBL1642157)
Affinity DataEC50:  1.58E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417577(CHEMBL1642158)
Affinity DataEC50:  3.98E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417578(CHEMBL1642159)
Affinity DataEC50:  1.26E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417073(CHEMBL1234887)
Affinity DataEC50:  794nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417069(CHEMBL1234889)
Affinity DataEC50:  251nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417070(CHEMBL1258570)
Affinity DataEC50:  251nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417071(CHEMBL1258571)
Affinity DataEC50:  794nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417072(CHEMBL1258681)
Affinity DataEC50:  126nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417073(CHEMBL1234887)
Affinity DataEC50:  794nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417074(CHEMBL1258795)
Affinity DataEC50:  501nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417075(CHEMBL1258796)
Affinity DataEC50:  3.16E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417076(CHEMBL1258915)
Affinity DataEC50:  1.58E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417077(CHEMBL1257181)
Affinity DataEC50:  631nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417078(CHEMBL1258914)
Affinity DataEC50:  631nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417079(CHEMBL1257182)
Affinity DataEC50:  1.00E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417080(CHEMBL1234888)
Affinity DataEC50:  316nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417081(CHEMBL1257298)
Affinity DataEC50:  316nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417082(CHEMBL1257414)
Affinity DataEC50:  1.58E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417083(CHEMBL1257415)
Affinity DataEC50:  794nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417084(CHEMBL1257527)
Affinity DataEC50:  1.58E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417085(CHEMBL1257528)
Affinity DataEC50:  1.58E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417086(CHEMBL1257645)
Affinity DataEC50:  2.51E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417087(CHEMBL1257646)
Affinity DataEC50:  2.00E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417088(CHEMBL1258461)
Affinity DataEC50:  1.00E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417558(CHEMBL1642162)
Affinity DataEC50:  5.01E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417557(CHEMBL1642161)
Affinity DataEC50:  398nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417556(CHEMBL1230591)
Affinity DataEC50:  1.00E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417555(CHEMBL1642160)
Affinity DataEC50:  794nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50417575(CHEMBL1642156)
Affinity DataEC50:  1.26E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed