Found 167 with Last Name = 'kihlberg' and Initial = 'j' 
Affinity DataKi: 0.5nMAssay Description:Inhibition of human alpha-thrombin using S-2366 as substrate after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of human alpha-thrombin using S-2366 as substrate after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Inhibition of human alpha-thrombin using S-2366 as substrate after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Inhibition of human alpha-thrombin using S-2366 as substrate after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1A receptor expressed in human CHO cell membranes incubated for 60 mins by scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibition of human alpha-thrombin using S-2366 as substrate after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibition of human alpha-thrombin using S-2366 as substrate after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 550nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1A receptor expressed in human CHO cell membranes incubated for 60 mins by scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 4.90E+3nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >5.40E+3nMAssay Description:Inhibition of human trypsin 1 using S-2222 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >5.40E+3nMAssay Description:Inhibition of human trypsin 1 using S-2222 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >5.40E+3nMAssay Description:Inhibition of human trypsin 1 using S-2222 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >5.40E+3nMAssay Description:Inhibition of human trypsin 1 using S-2222 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >5.40E+3nMAssay Description:Inhibition of human trypsin 1 using S-2222 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >5.40E+3nMAssay Description:Inhibition of human trypsin 1 using S-2222 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >1.70E+4nMAssay Description:Inhibition of human F10a using S-2765 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >1.70E+4nMAssay Description:Inhibition of human F10a using S-2765 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >1.70E+4nMAssay Description:Inhibition of human F10a using S-2765 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >1.70E+4nMAssay Description:Inhibition of human F10a using S-2765 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >1.90E+4nMAssay Description:Inhibition of human plasmin using S-2366 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >1.90E+4nMAssay Description:Inhibition of human F11a using S-2366 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >1.90E+4nMAssay Description:Inhibition of human F11a using S-2366 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >1.90E+4nMAssay Description:Inhibition of human plasmin using S-2366 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >1.90E+4nMAssay Description:Inhibition of human F11a using S-2366 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >1.90E+4nMAssay Description:Inhibition of human plasmin using S-2366 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >1.90E+4nMAssay Description:Inhibition of human F11a using S-2366 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >1.90E+4nMAssay Description:Inhibition of human plasmin using S-2366 as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >2.90E+4nMAssay Description:Inhibition of human F9a using pefachrome F9a as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >2.90E+4nMAssay Description:Inhibition of human F9a using pefachrome F9a as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >2.90E+4nMAssay Description:Inhibition of human F9a using pefachrome F9a as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataKi: >2.90E+4nMAssay Description:Inhibition of human F9a using pefachrome F9a as substrate preincubated for 300 secs followed by substrate addition measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of His6-tagged recombinant human BRD4 BD1 using (SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHGSGSK-biotin) as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of His6-tagged recombinant human BRD4 BD1 using (SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHGSGSK-biotin) as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of His6-tagged recombinant human BRD4 BD1 using (SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHGSGSK-biotin) as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 108nMAssay Description:Inhibition of His6-tagged recombinant human BRD4 BD2 using (SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHGSGSK-biotin) as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 118nMAssay Description:Inhibition of His6-tagged recombinant human BRD4 BD2 using (SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHGSGSK-biotin) as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 188nMAssay Description:Inhibition of His6-tagged recombinant human BRD4 BD2 using (SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHGSGSK-biotin) as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Targetvon Hippel-Lindau disease tumor suppressor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataIC50: 307nMAssay Description:Inhibition of VHL (unknown origin) assessed as phosphorylated peptide substrate incubated for 60 mins by TR-FRET based biochemical assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of recombinant human GST-tagged ERK5 (1 to 398 assessed as phosphorylated peptide substrate incubated for 60 mins by TR-FRET based biochem...More data for this Ligand-Target Pair
Targetvon Hippel-Lindau disease tumor suppressor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataIC50: 4.31E+3nMAssay Description:Inhibition of NanoLuc-tagged VHL in HEK293 cells incubated for 2 hrs by NanoBRET live cell assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Activity at human dopamine D2 receptor in NIH/3T3 cells assessed as beta-galactosidase activity after 5 days by R-SAT assayChecked by AuthorMore data for this Ligand-Target Pair
