TargetEpidermal growth factor receptor(Homo sapiens (Human))
Heinrich-Heine-UniversitäT
Curated by ChEMBL
Heinrich-Heine-UniversitäT
Curated by ChEMBL
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of human recombinant EGFR kinase expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of human recombinant CDK4/cyclin D1 kinase expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of CDK4/Cyclin D1 complex formationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.85E+4nMAssay Description:Inhibition of mouse recombinant PKCepsilon expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
University Of Oklahoma
Curated by ChEMBL
University Of Oklahoma
Curated by ChEMBL
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibition of CDK4/Cyclin D1 complex formationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.25E+4nMAssay Description:Inhibition of human recombinant CDK4/cyclin D1 kinase expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of mouse recombinant PKCepsilon expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Heinrich-Heine-UniversitäT
Curated by ChEMBL
Heinrich-Heine-UniversitäT
Curated by ChEMBL
Affinity DataIC50: 2.75E+4nMAssay Description:Inhibition of human recombinant EGFR kinase expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of mouse recombinant PKCepsilon expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Heinrich-Heine-UniversitäT
Curated by ChEMBL
Heinrich-Heine-UniversitäT
Curated by ChEMBL
Affinity DataIC50: 3.75E+4nMAssay Description:Inhibition of human recombinant EGFR kinase expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.75E+4nMAssay Description:Inhibition of human recombinant CDK4/cyclin D1 kinase expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Heinrich-Heine-UniversitäT
Curated by ChEMBL
Heinrich-Heine-UniversitäT
Curated by ChEMBL
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of human recombinant EGFR kinase expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.35E+4nMAssay Description:Inhibition of human recombinant CDK4/cyclin D1 kinase expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of mouse recombinant PKCepsilon expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mouse recombinant PKCepsilon expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Heinrich-Heine-UniversitäT
Curated by ChEMBL
Heinrich-Heine-UniversitäT
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant EGFR kinase expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant CDK4/cyclin D1 kinase expressed in Sf9 insect cellsMore data for this Ligand-Target Pair