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Found 248 with Last Name = 'grembecka' and Initial = 'j'
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50017478(Amastatin | CHEMBL28650 | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataKi:  30nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetAminopeptidase N(Sus scrofa (Pig))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129681(3-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  36nMAssay Description:Binding affinity towards aminopeptidase N (APN) from pig kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50117680(CHEMBL3613792)
Affinity DataKi:  57nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129685(2-Amino-4-methyl-pentanal | CHEMBL88476)
Affinity DataKi:  60nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129683(2-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoylmet...)
Affinity DataKi:  65nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129683(2-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoylmet...)
Affinity DataKi:  65nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129684(3-[(1-amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  66nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129681(3-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  67nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129682(2-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoylme...)
Affinity DataKi:  74nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129679((1-Amino-3-methyl-butyl)-phosphonic acid | 1-amino...)
Affinity DataKi:  230nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129684(3-[(1-amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  276nMAssay Description:Binding affinity towards aminopeptidase N (APN) from pig kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50117692(CHEMBL3613791)
Affinity DataKi:  310nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129677(3-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoyl]-p...)
Affinity DataKi:  330nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129682(2-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoylme...)
Affinity DataKi:  1.01E+3nMAssay Description:Binding affinity towards aminopeptidase N (APN) from pig kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129683(2-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoylmet...)
Affinity DataKi:  1.02E+3nMAssay Description:Binding affinity towards aminopeptidase N (APN) from pig kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129677(3-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoyl]-p...)
Affinity DataKi:  1.42E+3nMAssay Description:Binding affinity towards aminopeptidase N (APN) from pig kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129680(CHEMBL423870 | {[hydroxy(1-hydroxy-3-methylbutyl)p...)
Affinity DataKi:  4.88E+3nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129679((1-Amino-3-methyl-butyl)-phosphonic acid | 1-amino...)
Affinity DataKi:  5.50E+4nMAssay Description:Binding affinity towards aminopeptidase N (APN) from pig kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129678(2-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoyloxy...)
Affinity DataKi:  5.80E+4nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455873(CHEMBL4216801)
Affinity DataIC50:  3.60nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455856(CHEMBL4218724)
Affinity DataIC50:  7.5nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455865(CHEMBL4211318)
Affinity DataIC50:  10nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455881(CHEMBL4204254)
Affinity DataIC50:  13nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455883(CHEMBL4207749)
Affinity DataIC50:  13nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455862(CHEMBL4207527)
Affinity DataIC50:  13nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455880(CHEMBL4209476)
Affinity DataIC50:  14nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455860(CHEMBL4203695)
Affinity DataIC50:  15nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin polymerization-promoting protein(Homo sapiens (Human))
University of Virginia

LigandPNGBDBM59225(Boronic acid, cis-6 | Boronic acid, trans-6)
Affinity DataIC50:  17nMAssay Description:IC50 values for inhibition of cell growth using MCF-7 cell line were obtained by measuring the amount of total cell protein with the sulforhodamine B...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455864(CHEMBL4203028)
Affinity DataIC50:  18nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455868(CHEMBL4204241)
Affinity DataIC50:  21nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455861(CHEMBL4218853)
Affinity DataIC50:  22nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455879(CHEMBL4205576)
Affinity DataIC50:  26nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455874(CHEMBL4208216)
Affinity DataIC50:  28nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455869(CHEMBL4209696)
Affinity DataIC50:  32nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455859(CHEMBL3780895)
Affinity DataIC50:  32nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin polymerization-promoting protein(Homo sapiens (Human))
University of Virginia

LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  32nMAssay Description:IC50 values for inhibition of cell growth using MCF-7 cell line were obtained by measuring the amount of total cell protein with the sulforhodamine B...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455876(CHEMBL4217916)
Affinity DataIC50:  33nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455872(CHEMBL4204591)
Affinity DataIC50:  38nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455863(CHEMBL4204941)
Affinity DataIC50:  39nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455884(CHEMBL4210554)
Affinity DataIC50:  40nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455867(CHEMBL4213678)
Affinity DataIC50:  42nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455858(CHEMBL4210798)
Affinity DataIC50:  44nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50117750(CHEMBL3586090)
Affinity DataIC50:  46nMAssay Description:Inhibition of N-terminal thioredoxin His6-tagged full-length human menin expressed in Escherichia coli Rosetta (DE3) cells assessed as reduction in m...More data for this Ligand-Target Pair
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455857(CHEMBL4218711)
Affinity DataIC50:  55nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50496327(CHEMBL3126198)
Affinity DataIC50:  56nMAssay Description:Inhibition of human His-tagged menin-biotinylated MLL (4 to 15) interaction after 1 hr by HTRF assayMore data for this Ligand-Target Pair
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455882(CHEMBL4207176)
Affinity DataIC50:  57nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50455870(CHEMBL4210221)
Affinity DataIC50:  63nMAssay Description:Displacement of fluorescein-labeled MLL4-43 from full length human menin expressed in Escherichia coli BL21 (DE3) cells after 3 hrs by fluorescence p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50117744(CHEMBL3613789)
Affinity DataIC50:  65nMAssay Description:Inhibition of N-terminal thioredoxin His6-tagged full-length human menin expressed in Escherichia coli Rosetta (DE3) cells assessed as reduction in m...More data for this Ligand-Target Pair
TargetMenin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50496346(CHEMBL3126196)
Affinity DataIC50:  67nMAssay Description:Inhibition of human His-tagged menin-biotinylated MLL (4 to 15) interaction after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
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