Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Columbia University Medical Center
Curated by ChEMBL
Columbia University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.776nMAssay Description:Displacement of [125I]SB-258585 from human recombinant 5HT6 receptor using methiothepin after 45 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Agonist activity assessed by stimulation of [35S]GTP-gamma-S binding to human 5HT1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]rauwolscine from adrenergic alpha2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]rauwolscine from adrenergic alpha2C receptorMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Columbia University
Curated by ChEMBL
Columbia University
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of [3H]paroxetine from 5HTT receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Affinity DataKi: 34nMAssay Description:Binding affinity to 5HT2B receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Columbia University Medical Center
Curated by ChEMBL
Columbia University Medical Center
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Binding affinity to dopamine 2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Columbia University Medical Center
Curated by ChEMBL
Columbia University Medical Center
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine 1D receptor(Bos taurus (Bovine))
Columbia University
Curated by PDSP Ki Database
Columbia University
Curated by PDSP Ki Database
Affinity DataKi: 109nMAssay Description:Binding affinity to alpha 2C adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Columbia University Medical Center
Curated by ChEMBL
Columbia University Medical Center
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Binding affinity to sigma1 opioid receptor by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Affinity DataKi: 228nMAssay Description:Binding affinity to 5HT1B receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity to alpha 2A adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Affinity DataKi: 328nMAssay Description:Binding affinity to 5HT7 receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Affinity DataKi: 378nMAssay Description:Binding affinity to alpha 1B adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Affinity DataKi: 413nMAssay Description:Binding affinity to alpha 1A adrenergic receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
Columbia University Medical Center
Curated by ChEMBL
Columbia University Medical Center
Curated by ChEMBL
Affinity DataKi: 512nMAssay Description:Binding affinity to histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
Columbia University Medical Center
Curated by ChEMBL
Columbia University Medical Center
Curated by ChEMBL
Affinity DataKi: 839nMAssay Description:Binding affinity to histamine H1 receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
Columbia University Medical Center
Curated by ChEMBL
Columbia University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.03E+3nMAssay Description:Binding affinity to histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Homo sapiens (Human))
Columbia University Medical Center
Curated by ChEMBL
Columbia University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.77E+3nMAssay Description:Binding affinity to histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Binding affinity to 5HT2A receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Homo sapiens (Human))
Columbia University Medical Center
Curated by ChEMBL
Columbia University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.13E+3nMAssay Description:Binding affinity to histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Homo sapiens (Human))
Columbia University Medical Center
Curated by ChEMBL
Columbia University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.13E+3nMAssay Description:Binding affinity to histamine H2 receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Columbia University Medical Center
Curated by ChEMBL
Columbia University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.58E+3nMAssay Description:Binding affinity to D2 dopamine receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to D5 dopamine receptor by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT5A receptor by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT1E receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to KOR by radioligand binding assayMore data for this Ligand-Target Pair
TargetTumor necrosis factor receptor superfamily member 16(Homo sapiens (Human))
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Columbia University College Of Physicians And Surgeons
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to NT by radioligand binding assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Columbia University Medical Center
Curated by ChEMBL
Columbia University Medical Center
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Columbia University Medical Center
Curated by ChEMBL
Columbia University Medical Center
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to dopamine 2 receptor (unknown origin)More data for this Ligand-Target Pair