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Found 34 with Last Name = 'ozadali-sari' and Initial = 'k'
TargetAcetylcholinesterase(Homo sapiens (Human))
Hacettepe University

LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  6.16nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  650nMAssay Description:Inhibition of ovine recombinant COX-1 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50029593(CHEMBL7162 | N-(2-(cyclohexyloxy)-4-nitrophenyl)me...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human recombinant COX-2 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Hacettepe University

LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  4.94E+3nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
In DepthDetails
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Hacettepe University

LigandPNGBDBM225274(2-[4-(4-Ethylpiperazin-1-yl)phenyl]-1H-benzo[d]imi...)
Affinity DataIC50:  5.18E+3nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Hacettepe University

LigandPNGBDBM225276(2-[4-(4-Benzylpiperazin-1-yl)phenyl]-1H-benzo[d]im...)
Affinity DataIC50:  5.22E+3nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Hacettepe University

LigandPNGBDBM225280(5-Methoxy-2-[4-(4-benzylpiperazin-1-yl)phenyl]-1H-...)
Affinity DataIC50:  1.15E+4nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Hacettepe University

LigandPNGBDBM225273(2-[4-(4-Methylpiperazin-1-yl)phenyl]-1H-benzo[d]im...)
Affinity DataIC50:  1.57E+4nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
In DepthDetails
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50068356(CHEMBL3402334)
Affinity DataIC50:  1.73E+4nMAssay Description:Inhibition of human recombinant COX-2 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Hacettepe University

LigandPNGBDBM225277(5-Methoxy-2-[4-(4-methylpiperazin-1-yl)phenyl]-1H-...)
Affinity DataIC50:  1.78E+4nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Hacettepe University

LigandPNGBDBM225278(5-Methoxy-2-[4-(4-ethylpiperazin-1-yl)phenyl]-1H-b...)
Affinity DataIC50:  2.02E+4nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50068355(CHEMBL3402332)
Affinity DataIC50:  2.05E+4nMAssay Description:Inhibition of human recombinant COX-2 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50068351(CHEMBL3402317)
Affinity DataIC50:  2.46E+4nMAssay Description:Inhibition of human recombinant COX-2 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  2.96E+4nMAssay Description:Inhibition of human recombinant COX-2 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Hacettepe University

LigandPNGBDBM225274(2-[4-(4-Ethylpiperazin-1-yl)phenyl]-1H-benzo[d]imi...)
Affinity DataIC50:  3.49E+4nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50068356(CHEMBL3402334)
Affinity DataIC50:  3.98E+4nMAssay Description:Inhibition of ovine recombinant COX-1 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50068351(CHEMBL3402317)
Affinity DataIC50:  6.47E+4nMAssay Description:Inhibition of ovine recombinant COX-1 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50068354(CHEMBL3402326)
Affinity DataIC50:  6.82E+4nMAssay Description:Inhibition of human recombinant COX-2 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50068352(CHEMBL3402318)
Affinity DataIC50:  7.96E+4nMAssay Description:Inhibition of ovine recombinant COX-1 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50068354(CHEMBL3402326)
Affinity DataIC50:  8.56E+4nMAssay Description:Inhibition of ovine recombinant COX-1 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Hacettepe University

LigandPNGBDBM225276(2-[4-(4-Benzylpiperazin-1-yl)phenyl]-1H-benzo[d]im...)
Affinity DataIC50:  9.72E+4nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50068355(CHEMBL3402332)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ovine recombinant COX-1 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50068353(CHEMBL3402325)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ovine recombinant COX-1 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Hacettepe University

LigandPNGBDBM225279(5-Methoxy-2-[4-(4-phenylpiperazin-1-yl)phenyl]-1H-...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Hacettepe University

LigandPNGBDBM225275(2-[4-(4-Phenylpiperazin-1-yl)phenyl]-1H-benzo[d]im...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Hacettepe University

LigandPNGBDBM225279(5-Methoxy-2-[4-(4-phenylpiperazin-1-yl)phenyl]-1H-...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50068353(CHEMBL3402325)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX-2 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50068352(CHEMBL3402318)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX-2 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Hacettepe University

LigandPNGBDBM225275(2-[4-(4-Phenylpiperazin-1-yl)phenyl]-1H-benzo[d]im...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetAcetylcholinesterase(Homo sapiens (Human))
Hacettepe University

LigandPNGBDBM225273(2-[4-(4-Methylpiperazin-1-yl)phenyl]-1H-benzo[d]im...)
Affinity DataIC50:  1.17E+5nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
In DepthDetails
TargetAcetylcholinesterase(Homo sapiens (Human))
Hacettepe University

LigandPNGBDBM225278(5-Methoxy-2-[4-(4-ethylpiperazin-1-yl)phenyl]-1H-b...)
Affinity DataIC50:  1.21E+5nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetAcetylcholinesterase(Homo sapiens (Human))
Hacettepe University

LigandPNGBDBM225280(5-Methoxy-2-[4-(4-benzylpiperazin-1-yl)phenyl]-1H-...)
Affinity DataIC50:  1.44E+5nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50029593(CHEMBL7162 | N-(2-(cyclohexyloxy)-4-nitrophenyl)me...)
Affinity DataIC50:  2.13E+5nMAssay Description:Inhibition of ovine recombinant COX-1 using PGH2 as substrate incubated for 10 mins prior to arachidonic acid addition measured after 2 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Hacettepe University

LigandPNGBDBM225277(5-Methoxy-2-[4-(4-methylpiperazin-1-yl)phenyl]-1H-...)
Affinity DataIC50:  2.29E+5nMpH: 8.0 T: 2°CAssay Description:Reactions were performed in a mediumcontaining substrate (0.05-0.4 mM) combined with 0.125 mM DTNB in 100 mM 3-(N-morpholino)propanesulfonic acid buf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails