BindingDB PrimarySearch

BDBM158154 US9029356, 11::US9255087, 11

SMILES: CN1CCN(CC1)c1ccc(C(=O)Nc2n[nH]c3ccc(Cc4cc(F)cc(F)c4)cc23)c(NC2CCOCC2)c1

InChI Key: InChIKey=HAYYBYPASCDWEQ-UHFFFAOYSA-N

Data: 1 KI 60 IC50

PDB links: 1 PDB ID matches this monomer.

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 61 hits for monomerid = 158154
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
NPM/ALK (Nucleophosmin/ALK tyrosine kinase receptor) (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PDB PubMed	6.20	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of recombinant ALK (unknown origin)				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Aurora kinase B/Inner centromere protein (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	US Patent	n/a	n/a	338	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences S.R.L. US Patent					Assay Description The inhibitory activity of putative kinase inhibitors and the potency of selected compounds were determined using a trans-phosphorylation assay.A spe...				Citation and Details
Nerviano Medical Sciences S.R.L. US Patent					More data for this Ligand-Target Pair
NPM/ALK (Nucleophosmin/ALK tyrosine kinase receptor) (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PDB US Patent	n/a	n/a	55	n/a	n/a	n/a	n/a	n/a	n/a
NERVIANO MEDICAL SCIENCES S.R.L. US Patent					Assay Description BioKinase buffer was composed of 50 mM HEPES pH 7.5 containing 1 mM MnCl2, 5 mM MgCl2, 1 mM DTT, 3 microM Na3VO4, and 0.2 mg/mL BSA. 3x KB is buffer ...				Citation and Details
NERVIANO MEDICAL SCIENCES S.R.L. US Patent					More data for this Ligand-Target Pair				3D Structure (crystal)
Insulin-like growth factor I receptor (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	US Patent	n/a	n/a	263	n/a	n/a	n/a	n/a	n/a	n/a
NERVIANO MEDICAL SCIENCES S.R.L. US Patent					Assay Description Kinase buffer was composed of 50 mM HEPES pH 7.9 containing 3 mM MnCl2, 1 mM DTT, 3 microM Na3VO4, and 0.2 mg/mL BSA. 3x KB is buffer of the same com...				Citation and Details
NERVIANO MEDICAL SCIENCES S.R.L. US Patent					More data for this Ligand-Target Pair
Serine/threonine-protein kinase Aurora (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	US Patent	n/a	n/a	338	n/a	n/a	n/a	n/a	n/a	n/a
NERVIANO MEDICAL SCIENCES S.R.L. US Patent					Assay Description The kinase buffer was composed of 50 mM HEPES, pH 7.0, 10 mM MnCl2, 1 mM DTT, 3 microM Na3VO4, and 0.2 mg/mL BSA. The kinase assay was run with an en...				Citation and Details
NERVIANO MEDICAL SCIENCES S.R.L. US Patent					More data for this Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase ROS (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	5	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of human TEL (336 residues) fused-ROS1 (1891 to 2347 residues) (unknown origin) expressed in mouse BAF3 cells assessed as cell growth inhi...				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Neurotrophic tyrosine kinase receptor (Homo Sapiens)	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	3	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of human TEL (336 residues) fused-TRKA (440 to 796 residues) (unknown origin) expressed in mouse BAF3 cells assessed as cell growth inhibi...				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Neurotrophic tyrosine kinase receptor type 2 (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	3	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of human TEL (336 residues) fused-TRKB (455 to 822 residues) (unknown origin) expressed in mouse BAF3 cells assessed as cell growth inhibi...				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
NT-3 growth factor receptor (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	3	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of human TEL (336 residues) fused-TRKC (454 to 825 residues) (unknown origin) expressed in mouse BAF3 cells assessed as cell growth inhibi...				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Neurotrophic tyrosine kinase receptor (Homo Sapiens)	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	1	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of TRKA (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Neurotrophic tyrosine kinase receptor type 2 (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	3	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of recombinant human TRKB incubated for 90 mins by selectscreen kinase assay				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
NT-3 growth factor receptor (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	5	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of recombinant human TRKC incubated for 90 mins by selectscreen kinase assay				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase ROS (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	7	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of ROS1 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK2 (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	40	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of JAK2 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine kinase non-receptor protein 2 (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	70	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of ACK1 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK1 (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	112	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of JAK1 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Insulin-like growth factor I receptor (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	122	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of IGF1R (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Focal adhesion kinase 1/vascular endothelial growth factor receptor 3 (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	140	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of FAK (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase receptor FLT3 (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	164	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of FLT3 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase BRK (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	195	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of BRK (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Insulin receptor (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	209	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of IR (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
NPM/ALK (Nucleophosmin/ALK tyrosine kinase receptor) (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PDB PubMed	n/a	n/a	12	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of recombinant ALK (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Serine/threonine-protein kinase Aurora (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	215	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of AUR2 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
JAK3/JAK1 (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	349	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of JAK3 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Kinesin-1 heavy chain/ Tyrosine-protein kinase receptor RET (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	393	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of RET (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Fibroblast growth factor receptor (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of FGFR1 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of VEGFR2 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Focal adhesion kinase 1/vascular endothelial growth factor receptor 3 (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of VEGFR3 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
SRC (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of LCK (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase Kit (Kit) (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of KIT (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Aurora kinase B/Inner centromere protein (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of AUR1 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase ABL1 (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of ABL (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
PKC alpha and beta-2 (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of PKCbeta (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Cyclin-Dependent Kinase 2 (CDK2) (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of CDK2/CycA (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Tyrosine-protein kinase SYK (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of SYK (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
AKT/p21CIP1 (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of AKT1 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Activator of S phase kinase DBF4/Cell division cycle 7-related protein kinase (Homo sapiens (Human)-Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of CDC7/DBF4 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Serine/threonine-protein kinase Chk1 (Homo sapiens)	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of CHK1 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Serine/threonine-protein kinase EEF2K (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of EEF2K (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Epidermal growth factor receptor (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of EGFR1 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
MAP kinase ERK2 (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of ERK2 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Glycogen synthase kinase-3 (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of GSK3beta (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Inhibitor of NF-kappa-B kinase (IKK) (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of IKK2 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
MAP kinase-activated protein kinase 2 (Homo sapiens (human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of MAPKAPK2 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Maternal embryonic leucine zipper kinase (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of MELK (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of MET (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Dual specificity protein kinase TTK (Homo sapiens (Human))	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of MPS1 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Serine/threonine-protein kinase MST4 (Homo sapiens)	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of MST4 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Serine/threonine-protein kinase NEK6 (Homo sapiens)	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of NEK6 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair
Serine/threonine-protein kinase NIM1 (Homo sapiens)	BDBM158154 (US9029356, 11 \| US9255087, 11) Show SMILES Show InChI	KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase PC cid PC sid PDB UniChem Similars	PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Nerviano Medical Sciences Srl Curated by ChEMBL					Assay Description Inhibition of NIM1 (unknown origin) in presence of gamma33-ATP				Citation and Details
Nerviano Medical Sciences Srl Curated by ChEMBL					More data for this Ligand-Target Pair

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