BDBM20160 3-[(4-methoxyphenyl)amino]-1,4-diphenyl-2,5-dihydro-1H-pyrrole-2,5-dione::GSK3987 Analogue::Substituted Maleimide, 8

SMILES COc1ccc(cc1)N=C1C(C(=O)N(C1=O)c1ccccc1)c1ccccc1

InChI Key InChIKey=IVMIYZHBOTZWSL-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 20160   

TargetOxysterols receptor LXR-beta(Human)
Glaxosmithkline

LigandPNGBDBM20160(3-[(4-methoxyphenyl)amino]-1,4-diphenyl-2,5-dihydr...)
Affinity DataEC50:  260nMpH: 7.5 T: 22°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Human)
Glaxosmithkline

LigandPNGBDBM20160(3-[(4-methoxyphenyl)amino]-1,4-diphenyl-2,5-dihydr...)
Affinity DataEC50:  275nMpH: 7.5 T: 22°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed