BDBM50008710 CHEMBL3235977

SMILES Fc1ccc(NC(=O)N2CCc3cncnc3C2c2ccc(cc2)C(F)(F)F)cc1

InChI Key InChIKey=HBSIDFVCWOXNNO-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50008710   

LigandPNGBDBM50008710(CHEMBL3235977)
Affinity DataIC50:  1.17E+3nMAssay Description:Antagonist activity at rat TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced Ca2+ influx incubated 2.5 mins prior to icilin chall...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50008710(CHEMBL3235977)
Affinity DataIC50:  786nMAssay Description:Antagonist activity at human TRPM8 assessed as inhibition of icilin-induced Ca2+ influx incubated 2.5 mins prior to icilin challenge by luminometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed