BDBM50008712 CHEMBL3235979

SMILES FC(F)(F)c1ccc(cc1)[C@H]1N(CCc2cccnc12)C(=O)Nc1cccnc1

InChI Key InChIKey=GFCKYRRYSOERHO-LJQANCHMSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50008712   

LigandPNGBDBM50008712(CHEMBL3235979)
Affinity DataIC50:  48nMAssay Description:Antagonist activity at rat TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced Ca2+ influx incubated 2.5 mins prior to icilin chall...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50008712(CHEMBL3235979)
Affinity DataIC50:  24nMAssay Description:Antagonist activity at human TRPM8 assessed as inhibition of icilin-induced Ca2+ influx incubated 2.5 mins prior to icilin challenge by luminometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed