BDBM50167161 (E)-3-{3-[Cyclohexanecarbonyl-(4'-dimethylamino-biphenyl-4-ylmethyl)-amino]-phenyl}-acrylic acid methyl ester::CHEMBL192966
SMILES COC(=O)\C=C\c1cccc(c1)N(Cc1ccc(cc1)-c1ccc(cc1)N(C)C)C(=O)C1CCCCC1
InChI Key InChIKey=VLQTUNDJHLEFEQ-KGENOOAVSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50167161
Affinity DataEC50: 25nMAssay Description:Effective concentration against farnesoid X receptor (FXR)More data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Effective concentration towards farnesoid X receptor (FXR)More data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Effective concentration against farnesoid X receptor (FXR)More data for this Ligand-Target Pair
Affinity DataEC50: 800nMAssay Description:Agonist activity at human FXR transfected in CHO-K1 cells coexpressed with beta-galactosidase incubated for 3 to 16 hrs by PathHunter chemiluminescen...More data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Agonist activity at FXRMore data for this Ligand-Target Pair
Affinity DataKd: 1.22E+6nMAssay Description:Binding affinity to FXR (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Agonist activity at FXRMore data for this Ligand-Target Pair