BDBM50171259 3-(2-Dimethylamino-ethyl)-1H-indol-6-ol::CHEMBL382750

SMILES CN(C)CCc1c[nH]c2cc(O)ccc12

InChI Key InChIKey=WUQMRWPLIMXBDX-UHFFFAOYSA-N

Data  6 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50171259   

Target5-hydroxytryptamine receptor 2B(Human)
Organix

Curated by ChEMBL
LigandPNGBDBM50171259(3-(2-Dimethylamino-ethyl)-1H-indol-6-ol | CHEMBL38...)
Affinity DataKi:  6.30E+3nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2B receptor using [3H]-LSD as radioligand with the compound (10 uM) dissolved in DMSOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Human)
Organix

Curated by ChEMBL
LigandPNGBDBM50171259(3-(2-Dimethylamino-ethyl)-1H-indol-6-ol | CHEMBL38...)
Affinity DataKi:  6.80E+3nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [VGI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Human)
Organix

Curated by ChEMBL
LigandPNGBDBM50171259(3-(2-Dimethylamino-ethyl)-1H-indol-6-ol | CHEMBL38...)
Affinity DataKi:  7.60E+3nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2A receptor using [3H]-ketanserin as radioligand with the compound (10 uM) dissolved in DMSOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Human)
Organix

Curated by ChEMBL
LigandPNGBDBM50171259(3-(2-Dimethylamino-ethyl)-1H-indol-6-ol | CHEMBL38...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition constant against human 5-hydroxytryptamine 2C receptor [INI isoforms] using [3H]-mesulergine as radioligand with the compound (10 uM) diss...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50171259(3-(2-Dimethylamino-ethyl)-1H-indol-6-ol | CHEMBL38...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition constant against rat 5-hydroxytryptamine 2A receptor using [3H]-ketanserin as radioligand with the compound (10 uM) dissolved in DMSOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Organix

Curated by ChEMBL
LigandPNGBDBM50171259(3-(2-Dimethylamino-ethyl)-1H-indol-6-ol | CHEMBL38...)
Affinity DataKi:  1.90E+4nMAssay Description:Inhibition constant against rat 5-hydroxytryptamine 2C receptor using [3H]-mesulergine as radioligand with the compound (10 uM) dissolved in DMSOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed