BDBM50202222 CHEMBL398714::N-tert-butyl-6,7-dichloro-3-(methylsulfonyl)quinoxalin-2-amine

SMILES CC(C)(C)Nc1nc2cc(Cl)c(Cl)cc2nc1S(C)(=O)=O

InChI Key InChIKey=GNZCSGYHILBXLL-UHFFFAOYSA-N

Data  1 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50202222   

TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50202222(CHEMBL398714 | N-tert-butyl-6,7-dichloro-3-(methyl...)
Affinity DataIC50:  32nMAssay Description:Effect on augmentation of [125]GLP1 binding to human GLP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50202222(CHEMBL398714 | N-tert-butyl-6,7-dichloro-3-(methyl...)
Affinity DataEC50:  101nMAssay Description:Agonist activity at human GLP1 receptor expressed in BHK cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50202222(CHEMBL398714 | N-tert-butyl-6,7-dichloro-3-(methyl...)
Affinity DataEC50:  155nMAssay Description:Agonist activity at human GLP1 assessed as stimulation of cAMPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed