BDBM50312464 2-(4-(3-(4-bromophenyl)-5-(4-(trifluoromethyl)phenyl)pent-2-en-4-ynyloxy)-2-methylphenoxy)acetic acid::CHEMBL1081963

SMILES Cc1cc(OC\C=C(/C#Cc2ccc(cc2)C(F)(F)F)c2ccc(Br)cc2)ccc1OCC(O)=O

InChI Key InChIKey=NWQRCIMQYXJWJG-KGENOOAVSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50312464   

TargetPeroxisome proliferator-activated receptor alpha(Human)
The Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50312464(2-(4-(3-(4-bromophenyl)-5-(4-(trifluoromethyl)phen...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human 293T cells cotransfected with Gal4-DBD by luciferase transactivation ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
The Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50312464(2-(4-(3-(4-bromophenyl)-5-(4-(trifluoromethyl)phen...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human PPARdelta ligand binding domain expressed in human 293T cells cotransfected with Gal4-DBD by luciferase transactivation ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
The Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50312464(2-(4-(3-(4-bromophenyl)-5-(4-(trifluoromethyl)phen...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human 293T cells cotransfected with Gal4-DBD by luciferase transactivation ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed