BDBM50321821 4-((1H-Imidazol-4-yl)methyl)-1-(4-fluorophenyl)piperidine::CHEMBL1173809

SMILES Fc1ccc(cc1)N1CCC(Cc2cnc[nH]2)CC1

InChI Key InChIKey=IXNINVYBQXUWTR-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50321821   

TargetHistamine H3 receptor(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321821(4-((1H-Imidazol-4-yl)methyl)-1-(4-fluorophenyl)pip...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50321821(4-((1H-Imidazol-4-yl)methyl)-1-(4-fluorophenyl)pip...)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed