BDBM50323838 5-(trifluoromethyl)-6-(8-(5-(trifluoromethyl)pyridin-2-ylamino)pyrido[2,3-b]pyrazin-3-yl)nicotinonitrile::CHEMBL1214401

SMILES FC(F)(F)c1ccc(Nc2ccnc3nc(cnc23)-c2ncc(cc2C(F)(F)F)C#N)nc1

InChI Key InChIKey=XCKZSCJEDORJGO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50323838   

LigandPNGBDBM50323838(5-(trifluoromethyl)-6-(8-(5-(trifluoromethyl)pyrid...)
Affinity DataIC50:  15nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed