Affinity DataKi: 0.300nMAssay Description:Competitive inhibition of recombinant mouse aurora kinase A expressed in insect Sf9 cells in presence of ATPMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Competitive inhibition of recombinant mouse aurora kinase A expressed in insect Sf9 cells in presence of ATPMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Antagonistic activity of the compound was determined against mice melanocortin 4 receptor using [125I]-[NDP]-R-MSH as radioligand in a membranefiltra...More data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Antagonistic activity of the compound was determined against mice melanocortin 4 receptor using [125I]-[NDP]-R-MSH as radioligand in a membranefiltra...More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Antagonistic activity of the compound was determined against mice melanocortin 4 receptor using [125I]-[NDP]-R-MSH as radioligand in a membranefiltra...More data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Antagonistic activity of the compound was determined against mice melanocortin 4 receptor using [125I]-[NDP]-R-MSH as radioligand in a membranefiltra...More data for this Ligand-Target Pair
Affinity DataKi: 690nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 770nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 840nMAssay Description:Binding affinity to hERGMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 920nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Antagonistic activity of the compound was determined against mice melanocortin 4 receptor using [125I]-[NDP]-R-MSH as radioligand in a membranefiltra...More data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+3nMAssay Description:Antagonistic activity of the compound was determined against mice melanocortin 4 receptor using [125I]-[NDP]-R-MSH as radioligand in a membranefiltra...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 3.15E+3nMAssay Description:Binding affinity to hERGMore data for this Ligand-Target Pair
Affinity DataKi: 4.10E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.30E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.58E+4nMAssay Description:Antagonistic activity of the compound was determined against mice melanocortin 4 receptor using [125I]-[NDP]-R-MSH as radioligand in a membranefiltra...More data for this Ligand-Target Pair
Affinity DataKi: 2.60E+4nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant mouse aurora kinase A expressed in insect Sf9 cells using biotin-GLRRASLG as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Merck Research Laboratories
Merck Research Laboratories
Affinity DataIC50: 3nMpH: 8.2Assay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of mouse recombinant Aurora A kinase expressed in insect Sf9 cells by radioactive flashplate assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of aurora kinase A autophosphorylation at T288 in human HCT116 cells by immunofluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant mouse aurora kinase A expressed in insect Sf9 cells using biotin-GLRRASLG as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Merck Research Laboratories
Merck Research Laboratories
Affinity DataIC50: 14nMpH: 8.2Assay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of aurora kinase A autophosphorylation at T288 in human HCT116 cells by immunofluorescence analysisMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Merck Research Laboratories
Merck Research Laboratories
Affinity DataIC50: 22nMpH: 8.2Assay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Merck Research Laboratories
Merck Research Laboratories
Affinity DataIC50: 23nMpH: 8.2Assay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant mouse aurora kinase A expressed in insect Sf9 cells using biotin-GLRRASLG as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of recombinant mouse aurora kinase A expressed in insect Sf9 cells using biotin-GLRRASLG as substrate in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair