Affinity DataKi: 0.440nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCdelta expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 18.4nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 205nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 319nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 529nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCdelta expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 590nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCdelta expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 661nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 915nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCdelta expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.18E+4nMAssay Description:Inhibition of human recombinant UGT2B17 assessed as reduction of scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 5.78E+4nMAssay Description:Competitive inhibition of UGT2B17-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 9.81E+4nMAssay Description:Inhibition of recombinant human C-terminal His-tagged UGT1A10 after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGAMore data for this Ligand-Target Pair
Affinity DataKi: 1.01E+5nMAssay Description:Competitive inhibition of UGT2B7-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 1.13E+5nMAssay Description:Competitive inhibition of UGT2B7-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 1.62E+5nMAssay Description:Inhibition of recombinant human C-terminal His-tagged UGT2B7 after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGAMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+5nMAssay Description:Non competitive inhibition of UGT2B17-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 1.92E+5nMAssay Description:Non competitive inhibition of UGT2B7-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 2.01E+5nMAssay Description:Competitive inhibition of UGT2B17-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 2.58E+5nMAssay Description:Non competitive inhibition of UGT2B7-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 3.01E+5nMAssay Description:Competitive inhibition of UGT2B7-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 4.27E+5nMAssay Description:Competitive inhibition of UGT2B17-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 6.08E+5nMAssay Description:Non competitive inhibition of UGT2B17-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 6.24E+5nMAssay Description:Non competitive inhibition of UGT2B7-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
TargetUDP-glucuronosyltransferase 1A9(Homo sapiens (Human))
Gdansk University Of Technology
Curated by ChEMBL
Gdansk University Of Technology
Curated by ChEMBL
Affinity DataKi: 9.58E+5nMAssay Description:Inhibition of human recombinant UGT1A9 activity expressed in baculovirus-infected Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.44E+6nMAssay Description:Non competitive inhibition of UGT2B17-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
TargetUDP-glucuronosyltransferase 1A9(Homo sapiens (Human))
Gdansk University Of Technology
Curated by ChEMBL
Gdansk University Of Technology
Curated by ChEMBL
Affinity DataKi: 1.65E+6nMAssay Description:Inhibition of human recombinant UGT1A9 activity expressed in baculovirus-infected Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Inhibition of human UGT2B7 by substrate-independent inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair