Affinity DataKi: 1nM ΔG°: -51.4kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 6nM ΔG°: -46.9kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 7nM ΔG°: -46.5kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 7nM ΔG°: -46.5kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 8nM ΔG°: -46.2kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 10nM ΔG°: -45.7kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 11nM ΔG°: -45.4kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 12nM ΔG°: -47.0kJ/moleT: 2°CAssay Description:hese assays were performed at adenosine receptors transfected using a cAMP enzymeimmunoassay kit (Amersham Biosciences). CHO-A2A cells were seeded (1...More data for this Ligand-Target Pair
Affinity DataKi: 12nM ΔG°: -45.2kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 14nM ΔG°: -44.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 14nM ΔG°: -44.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 14nM ΔG°: -44.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 16nM ΔG°: -44.5kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 17nM ΔG°: -44.3kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 18nM ΔG°: -44.2kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 21nM ΔG°: -43.8kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 23.9nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 25nM ΔG°: -45.1kJ/moleT: 2°CAssay Description:hese assays were performed at adenosine receptors transfected using a cAMP enzymeimmunoassay kit (Amersham Biosciences). CHO-A2A cells were seeded (1...More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 33nM ΔG°: -42.7kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 34.5nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 35nM ΔG°: -42.6kJ/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair
Affinity DataKi: 46.1nMAssay Description:The binding assay for adenosine A2B receptor subtype was carried out on human recombinant source (HEK-293 cells) and [3H]DPCPX as radioligand, accord...More data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Biological assay using monoamine oxidase or LSD1.More data for this Ligand-Target Pair