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Targets Binding with 3 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
1-alkyl-2-acetylglycerophosphocholine esterase
IC50:
3
2
1
2D
3D
TSV
1-deoxy-D-xylulose 5-phosphate reductoisomerase, chloroplastic
IC50:
3
1
3
2D
3D
TSV
1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase delta-1
Kd:
4
1
9
2D
3D
TSV
2,6-dichloro-p-hydroquinone 1,2-dioxygenase
Ki:
4
1
1
2D
3D
TSV
3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase/7-dehydrocholesterol reductase
IC50:
3
1
7
2D
3D
TSV
3-keto-steroid reductase/17-beta-hydroxysteroid dehydrogenase 7
IC50:
3
1
6
2D
3D
TSV
5' exonuclease Apollo
IC50:
3
1
3
2D
3D
TSV
5'-3' exonuclease PLD3
IC50:
4
EC50:
2
1
4
2D
3D
TSV
5'-3' exonuclease PLD4
IC50:
4
EC50:
1
1
3
2D
3D
TSV
5,6-dihydroxyindole-2-carboxylic acid oxidase
IC50:
3
1
1
2D
3D
TSV
6-pyruvoyl tetrahydrobiopterin synthase
IC50:
3
1
4
2D
3D
TSV
Acetyl-CoA acetyltransferase/HMG-CoA reductase
IC50:
3
1
1
2D
3D
TSV
Acetyl-CoA carboxylase 1 [39-967]
IC50:
6
1
12
2D
3D
TSV
Acetyl-CoA carboxylase 2 [27-967]
IC50:
3
1
8
2D
3D
TSV
Acetyl-CoA carboxylase 2 [39-967]
IC50:
3
1
8
2D
3D
TSV
Acetylcholine receptor subunit gamma
IC50:
3
1
1
2D
3D
TSV
Acetyltransferase, GNAT family
IC50:
3
1
5
2D
3D
TSV
Actin
IC50:
3
1
6
2D
3D
TSV
Actin [R183K]
IC50:
3
1
6
2D
3D
TSV
Actin [R335K]
IC50:
3
1
6
2D
3D
TSV
ADAM metallopeptidase with thrombospondin type 1 motif 4
IC50:
6
1
1
2D
3D
TSV
Adenylosuccinate synthetase isozyme 2
IC50:
3
1
4
2D
3D
TSV
Alanine racemase, biosynthetic
Ki:
8
2
5
2D
3D
TSV
Aldehyde dehydrogenase 1, mitochondrial
IC50:
3
1
1
2D
3D
TSV
ALK tyrosine kinase receptor [G1269S]
Ki:
3
1
9
2D
3D
TSV
ALK tyrosine kinase/Hepatocyte growth factor receptor
IC50:
3
1
16
2D
3D
TSV
Alpha-(1,3)-fucosyltransferase 10
IC50:
3
1
9
2D
3D
TSV
Alpha-xylosidase
IC50:
3
1
1
2D
3D
TSV
Androgen receptor [646-919]
IC50:
2
Kd:
3
1
9
2D
3D
TSV
Asparagine synthetase [glutamine-hydrolyzing]
Ki:
14
2
12
2D
3D
TSV
ATP synthase subunit c
IC50:
5
2
1
2D
3D
TSV
ATP-sensitive inward rectifier potassium channel 10
IC50:
3
3
6
2D
3D
TSV
Aurora kinase A-interacting protein
Ki:
1
IC50:
2
2
4
2D
3D
TSV
Aurora kinase B-A
IC50:
3
1
5
2D
3D
TSV
Baculoviral IAP repeat-containing protein 3 [252-340]
Ki:
3
1
5
2D
3D
TSV
Beta-lactamase OXA-10
Ki:
2
IC50:
1
2
1
2D
3D
TSV
Beta-secretase 2 [21-466]
IC50:
3
1
9
2D
3D
TSV
Bifunctional 3'-phosphoadenosine 5'-phosphosulfate synthase 2
EC50:
3
1
7
2D
3D
TSV
Bifunctional dihydrofolate reductase-thymidylate synthase [N51I,C59R,S108N,I164L]
Ki:
3
IC50:
3
1
4
2D
3D
TSV
BirA Bifunctional Protein Mutant (V214A)
ITC:
3
1
0
2D
3D
TSV
BirA Bifunctional Protein Mutant (V219A)
ITC:
3
1
0
2D
3D
TSV
BirA Bifunctional Protein Mutant (W223A)
ITC:
3
1
0
2D
3D
TSV
Bone morphogenetic protein 2
Kd:
3
1
1
2D
3D
TSV
Bone morphogenetic protein 6
Kd:
3
1
3
2D
3D
TSV
Brain-derived neurotrophic factor
Kd:
6
1
11
2D
3D
TSV
Bromodomain testis-specific protein [21-137,251-382]
Ki:
2
Kd:
2
1
13
2D
3D
TSV
Bromodomain testis-specific protein [251-382]
Ki:
2
Kd:
1
1
12
2D
3D
TSV
Bromodomain-containing protein 2 [71-194,348-455]
Ki:
2
Kd:
1
1
14
2D
3D
TSV
Bromodomain-containing protein 2 [71-194]
Ki:
2
Kd:
1
1
13
2D
3D
TSV
Bromodomain-containing protein 3 [24-144,306-416]
Ki:
2
Kd:
1
1
8
2D
3D
TSV
Bromodomain-containing protein 3 [24-144]
Ki:
2
Kd:
1
1
7
2D
3D
TSV
Bromodomain-containing protein 3 [306-416]
Ki:
2
Kd:
1
1
7
2D
3D
TSV
Bromodomain-containing protein 4 [333-460]
Ki:
2
Kd:
2
1
6
2D
3D
TSV
C-terminal-binding protein 1 (CtBP1)
Kd:
4
ITC:
3
2
4
2D
3D
TSV
C-X-C motif chemokine 2
Kd:
3
1
4
2D
3D
TSV
Calcium/calmodulin-dependent protein kinase II inhibitor 2
IC50:
3
1
1
2D
3D
TSV
Calpain-1/Calpain-2 catalytic subunit
IC50:
3
1
11
2D
3D
TSV
cAMP-dependent protein kinase catalytic subunit alpha [V123M,T183A]
IC50:
3
1
2
2D
3D
TSV
cAMP-regulated phosphoprotein 19
EC50:
3
1
1
2D
3D
TSV
Carbonic anhydrase 1/2/5B, mitochondrial
IC50:
3
1
7
2D
3D
TSV
Casein kinase II subunit alpha
Ki:
3
1
8
2D
3D
TSV
CD81 antigen
Kd:
6
2
4
2D
3D
TSV
CDGSH iron-sulfur domain-containing protein 2
IC50:
3
1
3
2D
3D
TSV
Cell division control protein 45 homolog
IC50:
3
1
9
2D
3D
TSV
cGMP-dependent protein kinase 2 [41-418,G232E]
EC50:
4
1
7
2D
3D
TSV
cGMP-dependent protein kinase 2 [41-418,G356E]
EC50:
4
1
7
2D
3D
TSV
cGMP-dependent protein kinase 2 [41-418]
EC50:
4
1
6
2D
3D
TSV
cGMP-specific 3',5'-cyclic phosphodiesterase [1-660,682-875]
IC50:
3
1
10
2D
3D
TSV
cGMP-specific 3',5'-cyclic phosphodiesterase [1-662,679-875]
IC50:
3
1
10
2D
3D
TSV
cGMP-specific 3',5'-cyclic phosphodiesterase [535-860]
IC50:
3
1
9
2D
3D
TSV
Choline kinase
IC50:
3
1
1
2D
3D
TSV
Class A beta-lactamase BCL-1
IC50:
3
1
1
2D
3D
TSV
Class D beta-lactamase
IC50:
3
1
1
2D
3D
TSV
CMP-N-acetylneuraminate-beta-galactosamide-alpha-2,3-sialyltransferase 1
IC50:
3
1
4
2D
3D
TSV
Collagenase ColH
IC50:
3
1
1
2D
3D
TSV
Complement component C9
IC50:
3
1
1
2D
3D
TSV
Conantokin-G
ITC:
6
1
0
2D
3D
TSV
Conantokin-T
ITC:
4
1
0
2D
3D
TSV
Cyclin-dependent kinase 18
IC50:
3
3
6
2D
3D
TSV
Cystic fibrosis transmembrane conductance regulator [G550E]
IC50:
3
1
6
2D
3D
TSV
Cytochrome P450 2A2
IC50:
4
1
3
2D
3D
TSV
Cytochrome P450 2C23
IC50:
3
1
4
2D
3D
TSV
Cytochrome P450 3A4/3A43/3A5/3A7
IC50:
4
3
21
2D
3D
TSV
Cytochrome P450 7A1
IC50:
4
1
3
2D
3D
TSV
D(4) dopamine receptor [281-332]
IC50:
3
1
5
2D
3D
TSV
Dehaloperoxidase B
Kd:
3
1
1
2D
3D
TSV
Deoxyribonuclease gamma
IC50:
5
2
5
2D
3D
TSV
Dimer of Gag-Pol polyprotein [489-587,V571A]
Ki:
3
1
4
2D
3D
TSV
Dimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A,G574S]
Ki:
3
1
7
2D
3D
TSV
Dimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A,L525I]
Ki:
3
1
7
2D
3D
TSV
Dimer of Gag-Pol polyprotein [600-1159,L699I,K702N,C879S]
IC50:
3
1
5
2D
3D
TSV
Dimer of Growth hormone secretagogue receptor type 1
Ki:
4
1
5
2D
3D
TSV
Disabled homolog 2
Ki:
3
1
6
2D
3D
TSV
DNA cross-link repair 1A protein
IC50:
3
2
6
2D
3D
TSV
DNA polymerase nu
IC50:
3
1
6
2D
3D
TSV
DNA repair endonuclease XPF
IC50:
4
Kd:
2
2
6
2D
3D
TSV
Ecdysone receptor/Ultraspiracle
Ki:
3
IC50:
2
1
9
2D
3D
TSV
Efflux pump membrane transporter
Kd:
4
2
1
2D
3D
TSV
Elongation factor 1-alpha 1
Kd:
3
1
5
2D
3D
TSV
Elongation factor 1-alpha 2
Kd:
3
1
6
2D
3D
TSV
Endo-beta-N-acetylglucosaminidase
IC50:
3
1
1
2D
3D
TSV
Endochitinase B1 [A217G]
Kd:
3
2
3
2D
3D
TSV
Endochitinase B1 [D175A]
Kd:
3
2
3
2D
3D
TSV
Endochitinase B1 [E322A]
Kd:
3
2
3
2D
3D
TSV
Endochitinase B1 [M243A]
Kd:
3
2
3
2D
3D
TSV
Endochitinase B1 [R301K]
Kd:
3
2
3
2D
3D
TSV
Endochitinase B1 [T138A]
Kd:
3
2
3
2D
3D
TSV
Enoyl-ACP Reductase (FabI) Mutant (F203L)
ITC:
9
1
0
2D
3D
TSV
Enterobactin synthase component E
Ki:
4
1
5
2D
3D
TSV
Eotaxin
Kd:
3
1
5
2D
3D
TSV
Epidermal growth factor receptor [G719S]
IC50:
2
Kd:
1
2
15
2D
3D
TSV
Epidermal growth factor receptor [L861Q]
IC50:
2
Kd:
1
2
15
2D
3D
TSV
Epidermal/Hepatocyte growth factor receptor
IC50:
3
1
22
2D
3D
TSV
Eyes absent homolog 2 [253-538]
IC50:
3
Kd:
3
1
13
2D
3D
TSV
Eyes absent homolog 3 [223-510]
IC50:
6
2
11
2D
3D
TSV
Fatty acid-binding protein, liver [T94A]
Ki:
3
1
1
2D
3D
TSV
Fibroblast growth factor 7
Kd:
3
1
5
2D
3D
TSV
Flap endonuclease 1 [1-336]
IC50:
3
1
1
2D
3D
TSV
Frizzled-1
Kd:
3
1
5
2D
3D
TSV
G protein-coupled receptor 34a
EC50:
6
1
1
2D
3D
TSV
G protein-coupled receptor 34b
EC50:
6
1
1
2D
3D
TSV
Gag-Pol polyprotein [588-1027,V694A]/[588-1147,V694A]
Ki:
3
1
7
2D
3D
TSV
Gag-Pol polyprotein [588-1027,Y776L]/[588-1147,Y776L]
Ki:
3
1
7
2D
3D
TSV
Gag-Pol polyprotein [600-1159,Y780C]/Imidazoleglycerol-phosphate dehydratase [600-1029,Y780C]
IC50:
3
1
10
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-200],P14867[176-456]
Ki:
3
1
19
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,A118C]
Ki:
3
1
17
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,D95C]
Ki:
3
1
17
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,L179C]
Ki:
3
1
17
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,M169C]
Ki:
3
1
17
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R171C]
Ki:
3
1
17
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R183C]
Ki:
3
1
17
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R224C]
Ki:
3
1
17
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R233C]
Ki:
3
1
17
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T120C]
Ki:
3
1
17
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T165C]
Ki:
3
1
17
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T181C]
Ki:
3
1
17
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
16
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [A160C]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
16
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [F99C]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
16
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [G157C]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
16
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [G200C]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
16
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [S204C]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
16
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [S205C]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
16
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [T162C]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
16
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [T206C]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
16
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [V202C]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
16
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-1 [V211C]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
16
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-2 [29-451]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
17
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-3 [29-492]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
15
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-4 [36-554]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
15
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-5 [32-462]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
20
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-6 [20-453]/beta-2 [26-512]/gamma-2 [40-467]
Ki:
3
1
16
2D
3D
TSV
Genome polyprotein [1027-1207,C159S]
IC50:
4
1
4
2D
3D
TSV
Genome polyprotein [1027-1207,R155K]
IC50:
4
1
4
2D
3D
TSV
Genome polyprotein [2420-3010,S282T]
IC50:
3
1
2
2D
3D
TSV
GLRA1 protein
Ki:
6
3
1
2D
3D
TSV
Glucan 1,4-alpha-glucosidase
IC50:
3
1
1
2D
3D
TSV
Glutamate transporter homolog
Kd:
3
1
1
2D
3D
TSV
Glutathione S-transferase
IC50:
3
1
5
2D
3D
TSV
Glycerophosphocholine phosphodiesterase GPCPD1
Ki:
3
2
6
2D
3D
TSV
GMP synthase [glutamine-hydrolyzing]
IC50:
3
2
11
2D
3D
TSV
Granzyme K
Ki:
4
3
3
2D
3D
TSV
Growth hormone secretagogue receptor type 1/Isoform 1B of Growth hormone secretagogue receptor type 1 (1B)
Ki:
4
1
10
2D
3D
TSV
HbpA
Kd:
3
1
1
2D
3D
TSV
Heme-binding protein A
Kd:
6
1
2
2D
3D
TSV
Hepatocyte growth factor receptor/Proto-oncogene tyrosine-protein kinase receptor Ret
IC50:
3
1
13
2D
3D
TSV
Histamine oxidase
IC50:
3
1
1
2D
3D
TSV
Histo-blood group ABO system transferase
Ki:
7
IC50:
2
Kd:
3
1
14
2D
3D
TSV
Histone acetyltransferase
IC50:
3
3
1
2D
3D
TSV
Histone deacetylase 1/REST corepressor 3
Ki:
3
1
9
2D
3D
TSV
Histone H3.1
EC50:
3
1
13
2D
3D
TSV
Histone H3.1 [22-45]
IC50:
6
1
13
2D
3D
TSV
Histone-lysine N-methyltransferase SETD2
IC50:
3
3
16
2D
3D
TSV
Histone-lysine N-methyltransferase SETMAR
IC50:
3
1
7
2D
3D
TSV
Homeobox C9
Ki:
4
1
3
2D
3D
TSV
Inositol 1,4,5-trisphosphate receptor type 2
IC50:
6
1
3
2D
3D
TSV
Inositol phosphorylceramide synthase catalytic subunit AUR1
Ki:
2
IC50:
6
1
4
2D
3D
TSV
Integrin alpha-2
IC50:
3
2
3
2D
3D
TSV
Integrin alpha-5/beta-8
IC50:
3
1
5
2D
3D
TSV
Interferon gamma
Kd:
3
1
4
2D
3D
TSV
Interleukin-1 receptor type 1
IC50:
3
3
3
2D
3D
TSV
Inward rectifier potassium channel 13
IC50:
3
3
6
2D
3D
TSV
Isoform Beta of cGMP-dependent protein kinase 1 [1-351,G182E]
EC50:
4
1
10
2D
3D
TSV
Isoform Beta of cGMP-dependent protein kinase 1 [1-351,G306E]
EC50:
4
1
10
2D
3D
TSV
Isoform Beta of cGMP-dependent protein kinase 1 [1-351]
EC50:
4
1
9
2D
3D
TSV
Isoform Beta of cGMP-dependent protein kinase 1 [5-676,G306E]
EC50:
4
1
10
2D
3D
TSV
Kallikrein-12
Ki:
3
1
4
2D
3D
TSV
Kaposi's sarcoma-associated herpesvirus cyclin homolog
IC50:
3
1
1
2D
3D
TSV
Kinesin-like protein KIF11 [15-368]
IC50:
3
1
6
2D
3D
TSV
Kinesin-like protein KIF11 [D130V]
IC50:
12
1
6
2D
3D
TSV
Kinesin-like protein KIF15
IC50:
5
1
6
2D
3D
TSV
Kv channel-interacting protein 2
IC50:
3
1
19
2D
3D
TSV
Large neutral amino acids transporter small subunit 3
IC50:
3
1
1
2D
3D
TSV
Lecithin retinol acyltransferase
IC50:
7
1
4
2D
3D
TSV
Leucine-rich repeat serine/threonine-protein kinase 2 [970-2527,I2020T]
IC50:
3
1
6
2D
3D
TSV
Lysine-specific histone demethylase 1B
Ki:
3
1
4
2D
3D
TSV
LysP-related transporter STM2200 (STM2200)
Kd:
2
ITC:
4
1
1
2D
3D
TSV
Macrophage scavenger receptor types I and II
IC50:
3
2
10
2D
3D
TSV
Mannan-binding lectin serine protease 1
Ki:
2
IC50:
3
1
10
2D
3D
TSV
Mast cell protease 9
Ki:
3
2
1
2D
3D
TSV
Matrix metalloproteinase-24
Ki:
2
IC50:
1
3
4
2D
3D
TSV
Metallo-beta-lactamase AIM-1
Ki:
3
1
1
2D
3D
TSV
Methylcytosine dioxygenase TET1
IC50:
4
2
6
2D
3D
TSV
Mitochondrial carnitine/acylcarnitine carrier protein
IC50:
3
1
4
2D
3D
TSV
Mitogen-activated protein kinase
IC50:
3
2
2
2D
3D
TSV
N-methyl-D-aspartate receptor
IC50:
9
1
1
2D
3D
TSV
N-terminal Xaa-Pro-Lys N-methyltransferase 2
Kd:
3
1
3
2D
3D
TSV
Neuronal acetylcholine receptor subunit alpha-3/alpha-5/beta-4
Ki:
3
2
22
2D
3D
TSV
Neuropeptide Y-Y2 receptor
Ki:
3
1
1
2D
3D
TSV
Neurotensin/neuromedin N
Ki:
3
3
1
2D
3D
TSV
Ninein
Ki:
3
1
18
2D
3D
TSV
Nitric oxide synthase, endothelial [N368D]
Ki:
3
1
1
2D
3D
TSV
Non-structural protein 4A
IC50:
3
1
1
2D
3D
TSV
ORF1a
Ki:
1
IC50:
2
Kd:
2
1
1
2D
3D
TSV
Ornithine aminotransferase, mitochondrial
Ki:
3
2
8
2D
3D
TSV
Outer capsid protein sigma-1
Ki:
3
3
4
2D
3D
TSV
OXA23 carbapenemase
Ki:
3
1
1
2D
3D
TSV
Peptidyl-prolyl cis-trans isomerase C
Ki:
3
2
3
2D
3D
TSV
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 4
Ki:
1
IC50:
2
3
10
2D
3D
TSV
Peroxiredoxin-1
IC50:
1
Kd:
2
2
8
2D
3D
TSV
Peroxisomal sarcosine oxidase
Ki:
2
IC50:
1
3
5
2D
3D
TSV
PH domain leucine-rich repeat-containing protein phosphatase 1
Kd:
3
1
9
2D
3D
TSV
Phosphatidylinositol 3,4,5-trisphosphate 3-phosphatase and dual-specificity protein phosphatase PTEN
IC50:
3
2
7
2D
3D
TSV
Phosphatidylinositol 3-kinase regulatory subunit beta/4,5-bisphosphate 3-kinase catalytic subunit beta isoform
IC50:
3
2
6
2D
3D
TSV
Phospho-2-dehydro-3-deoxyheptonate aldolase, Phe-sensitive
Ki:
5
1
3
2D
3D
TSV
Phosphoribosyl pyrophosphate synthase-associated protein 2
Ki:
3
1
7
2D
3D
TSV
Polyprotein II
IC50:
3
2
1
2D
3D
TSV
Polyunsaturated fatty acid lipoxygenase ALOX8
IC50:
3
1
3
2D
3D
TSV
Potassium voltage-gated channel subfamily H member 8
Ki:
3
3
3
2D
3D
TSV
Potassium-transporting ATPase subunit beta
IC50:
3
1
1
2D
3D
TSV
POU domain, class 5, transcription factor 1
IC50:
3
1
11
2D
3D
TSV
Pro-thyrotropin-releasing hormone-B
Ki:
4
1
1
2D
3D
TSV
Probable arabinosyltransferase A
IC50:
3
1
6
2D
3D
TSV
Proheparin-binding EGF-like growth factor
Kd:
3
1
3
2D
3D
TSV
Proline racemase
Ki:
2
IC50:
2
1
1
2D
3D
TSV
Protein ABHD11
IC50:
3
1
9
2D
3D
TSV
Protein disulfide-isomerase A3
IC50:
3
1
6
2D
3D
TSV
Protein disulfide-isomerase A4
IC50:
3
1
4
2D
3D
TSV
Protein disulfide-isomerase A6
IC50:
3
1
10
2D
3D
TSV
Protein mono-ADP-ribosyltransferase PARP8
IC50:
3
3
5
2D
3D
TSV
Protein translocase subunit SecA 1
IC50:
7
1
3
2D
3D
TSV
Protein translocase subunit SecA 2
IC50:
3
1
1
2D
3D
TSV
Protein UL24 homolog
IC50:
3
1
1
2D
3D
TSV
Proto-oncogene tyrosine-protein kinase Src [251-533,V323A,T338C]
IC50:
3
1
10
2D
3D
TSV
Proto-oncogene tyrosine-protein kinase Src [251-533,V323S,T338C]
IC50:
3
1
10
2D
3D
TSV
Putative cathepsin L 3
Ki:
3
IC50:
3
1
3
2D
3D
TSV
Putative farnesyl pyrophosphate synthase
Ki:
3
IC50:
3
1
1
2D
3D
TSV
Putative polyamine transporter
IC50:
7
1
1
2D
3D
TSV
RAR related orphan receptor B isoform 1
Ki:
3
1
1
2D
3D
TSV
RCG38204, isoform CRA_d
Ki:
3
1
1
2D
3D
TSV
Replicase polyprotein 1ab [3264-3569]
IC50:
3
1
1
2D
3D
TSV
Ribosomal protein S6 kinase alpha-1/alpha-2/alpha-3/alpha-4/alpha-5/alpha-6/beta-1/beta-2
Ki:
1
IC50:
2
3
50
2D
3D
TSV
RNA demethylase ALKBH5
IC50:
3
2
5
2D
3D
TSV
S-formylglutathione hydrolase
Ki:
4
Kd:
2
2
8
2D
3D
TSV
Saccharopepsin
Ki:
3
1
3
2D
3D
TSV
Segment polarity protein dishevelled homolog DVL-2
Ki:
3
1
4
2D
3D
TSV
Serine/threonine-protein kinase PAK 1 [249-545,K299R]
IC50:
3
1
8
2D
3D
TSV
Serine/threonine-protein kinase WNK1 [1-491]
IC50:
6
2
15
2D
3D
TSV
Serum paraoxonase/arylesterase 2
IC50:
3
1
10
2D
3D
TSV
Serum paraoxonase/lactonase 3
IC50:
3
1
8
2D
3D
TSV
SH2 domain-containing protein 1A
IC50:
3
1
9
2D
3D
TSV
Sialin
Ki:
3
IC50:
2
1
5
2D
3D
TSV
Sigma-54-dependent Fis family transcriptional regulator
IC50:
3
1
3
2D
3D
TSV
Sodium channel protein type 11 subunit alpha
IC50:
4
3
9
2D
3D
TSV
Sodium/myo-inositol cotransporter 2
IC50:
3
1
8
2D
3D
TSV
Sodium/nucleoside cotransporter
Ki:
3
2
1
2D
3D
TSV
Solute carrier organic anion transporter family member 4C1
IC50:
3
1
3
2D
3D
TSV
Stanniocalcin-1
IC50:
6
1
5
2D
3D
TSV
Steroid 11-beta-monooxygenase
IC50:
4
1
1
2D
3D
TSV
Sterol carrier protein 2
Kd:
2
EC50:
2
2
15
2D
3D
TSV
Streptavidin
Kd:
3
ITC:
3
4
1
2D
3D
TSV
Succinate dehydrogenase [ubiquinone] flavoprotein subunit, mitochondrial
IC50:
3
1
9
2D
3D
TSV
SugE
IC50:
3
1
1
2D
3D
TSV
Sulfotransferase 2A1
Ki:
2
IC50:
1
2
4
2D
3D
TSV
Superoxide dismutase
IC50:
3
1
1
2D
3D
TSV
Synapsin-1
IC50:
3
1
1
2D
3D
TSV
Thiamine-binding periplasmic protein
Kd:
3
1
3
2D
3D
TSV
Thioredoxin domain-containing protein 5
IC50:
3
1
7
2D
3D
TSV
Thyrotropin subunit beta
IC50:
3
1
1
2D
3D
TSV
Tolloid-like protein 1
Ki:
2
IC50:
1
1
5
2D
3D
TSV
Tolloid-like protein 2
Ki:
2
IC50:
1
1
6
2D
3D
TSV
Trehalose synthase/amylase TreS
Ki:
3
1
5
2D
3D
TSV
Tryptase
Ki:
5
2
5
2D
3D
TSV
Tuberculosinyl adenosine transferase
IC50:
3
1
6
2D
3D
TSV
Tumor necrosis factor receptor superfamily member 10A
IC50:
3
1
5
2D
3D
TSV
Tumor necrosis factor receptor superfamily member 5
IC50:
3
1
9
2D
3D
TSV
Tyrosine-protein kinase ABL1 [131-238]
Kd:
3
1
8
2D
3D
TSV
Tyrosine-protein kinase ABL2 [121-226]
Kd:
3
1
11
2D
3D
TSV
Tyrosine-protein phosphatase non-receptor type 1 [1-321]
IC50:
3
1
5
2D
3D
TSV
Tyrosine-protein phosphatase non-receptor type 9 [277-582]
Ki:
1
IC50:
3
1
3
2D
3D
TSV
Ubiquitin carboxyl-terminal hydrolase 17
IC50:
3
1
1
2D
3D
TSV
Ubiquitin carboxyl-terminal hydrolase 4
IC50:
3
3
7
2D
3D
TSV
UDP-glucuronosyltransferase 1A7
Ki:
3
2
4
2D
3D
TSV
UDP-glucuronosyltransferase 1A8
Ki:
4
3
8
2D
3D
TSV
Ultraspiracle isoform-A
Ki:
1
EC50:
2
2
1
2D
3D
TSV
Valine--tRNA ligase
IC50:
3
1
7
2D
3D
TSV
VIM-13
IC50:
3
1
1
2D
3D
TSV
Voltage-dependent calcium channel alpha-1 subunit
IC50:
6
1
1
2D
3D
TSV
Voltage-dependent L-type calcium channel subunit beta-2
Ki:
1
IC50:
2
2
23
2D
3D
TSV
Voltage-dependent P/Q-type calcium channel subunit alpha-1A
IC50:
2
EC50:
1
3
13
2D
3D
TSV