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BindingDB Data by Target
Target Name
contains
starts with
ends with
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Target Name
Affinity Link(s)
Article(s)
UniProt
Files
(1->4)-alpha-D-glucan:maltose-1-phosphate alpha-D-maltosyltransferase
IC50:
1
1
5
2D
3D
TSV
(ARTD1 or PARP1)
Ki:
1174
IC50:
3474
Kd:
178
EC50:
309
171
5
2D
3D
TSV
(ARTD2 or PARP2)
Ki:
20
IC50:
599
Kd:
82
58
6
2D
3D
TSV
(ARTD3 or PARP3)
IC50:
34
Kd:
20
13
0
2D
3D
TSV
(ARTD4 or PARP4)
IC50:
40
11
6
2D
3D
TSV
(ARTD5 or PARP5a)
IC50:
697
Kd:
7
48
4
2D
3D
TSV
(ARTD6 or PARP5b)
IC50:
819
Kd:
14
EC50:
9
50
5
2D
3D
TSV
(ARTD7 or PARP15)
IC50:
59
12
4
2D
3D
TSV
(ARTD7 or PARP15, Y598L)
IC50:
59
12
4
2D
3D
TSV
(ARTD8 or PARP14)
IC50:
197
Kd:
11
13
8
2D
3D
TSV
(ARTD8 or PARP14, Y1660L)
IC50:
197
Kd:
11
13
8
2D
3D
TSV
A disintegrin and metalloproteinase domain 17
Ki:
108
IC50:
402
28
1
2D
3D
TSV
A disintegrin and metalloproteinase with thrombospondin motifs 13
IC50:
3
2
8
2D
3D
TSV
A disintegrin and metalloproteinase with thrombospondin motifs 4 (ADAMTS-4)
Ki:
11
IC50:
478
Other:
2
35
7
2D
3D
TSV
A disintegrin and metalloproteinase with thrombospondin motifs 5
IC50:
57
Other:
8
2
0
2D
3D
TSV
A disintegrin and metalloproteinase with thrombospondin motifs 5 (ADAMTS-5)
Ki:
14
IC50:
1321
35
4
2D
3D
TSV
A disintegrin and metalloproteinase with thrombospondin motifs 6
IC50:
265
2
7
2D
3D
TSV
A transferase
Ki:
7
IC50:
2
Kd:
3
1
15
2D
3D
TSV
A-esterase 1
Ki:
22
IC50:
46
8
6
2D
3D
TSV
A-esterase 2
IC50:
3
1
10
2D
3D
TSV
A-FABP
Ki:
116
IC50:
538
Kd:
34
24
5
2D
3D
TSV
A-kinase anchor protein 18
EC50:
23
1
0
2D
3D
TSV
A-kinase anchor protein 18 kDa
EC50:
23
1
4
2D
3D
TSV
A-kinase anchor protein 7 isoform gamma
EC50:
46
2
4
2D
3D
TSV
A-T mutated
Ki:
20
IC50:
655
EC50:
1
33
10
2D
3D
TSV
A-type potassium channel modulatory protein 2
IC50:
3
1
19
2D
3D
TSV
A085R
Ki:
7
IC50:
28
1
1
2D
3D
TSV
A1 adenosine receptor
Ki:
393
IC50:
6
EC50:
125
23
1
2D
3D
TSV
A1 adenosine receptor (hA1)
Ki:
5130
IC50:
462
Kd:
93
EC50:
365
Koff:
2
Kon:
2
Other:
10
389
9
2D
3D
TSV
A1-A
IC50:
584
4
1
2D
3D
TSV
A190
IC50:
32
1
7
2D
3D
TSV
A1AR
Ki:
5130
IC50:
462
Kd:
93
EC50:
365
Koff:
2
Kon:
2
Other:
10
389
9
2D
3D
TSV
A2A adenosine receptor (hA2A)
Ki:
6616
IC50:
633
Kd:
44
EC50:
288
405
4
2D
3D
TSV
A2M
IC50:
2
1
8
2D
3D
TSV
A3 adenosine receptor (hA3)
Ki:
5929
IC50:
554
Kd:
15
EC50:
184
353
6
2D
3D
TSV
A3AR
Ki:
131
IC50:
2
EC50:
11
13
3
2D
3D
TSV
A4T40_06800
IC50:
12
2
1
2D
3D
TSV
A6592_09565
IC50:
661
7
1
2D
3D
TSV
A7M90_02080
IC50:
2
1
1
2D
3D
TSV
A8C65_01575
IC50:
661
7
1
2D
3D
TSV
A8C65_01580
IC50:
58
Kd:
1
1
1
2D
3D
TSV
A8C65_06565
IC50:
12
2
1
2D
3D
TSV
A8G17_01625
IC50:
58
Kd:
1
1
1
2D
3D
TSV
A8G17_01630
IC50:
661
7
1
2D
3D
TSV
A8M42_07845
IC50:
661
7
1
2D
3D
TSV
A8M42_07850
IC50:
58
Kd:
1
1
1
2D
3D
TSV
A8M42_10590
IC50:
12
2
1
2D
3D
TSV
A8M81_11475
IC50:
12
2
1
2D
3D
TSV
A9819_23720
IC50:
661
7
1
2D
3D
TSV
A9843_06625
IC50:
2
1
1
2D
3D
TSV
A9843_09540
Ki:
3
1
1
2D
3D
TSV
A9R57_11170
IC50:
12
2
1
2D
3D
TSV
A9R57_13540
IC50:
661
7
1
2D
3D
TSV
A9R57_13545
IC50:
58
Kd:
1
1
1
2D
3D
TSV
A9X62_17950
IC50:
12
2
1
2D
3D
TSV
AA 1-650
IC50:
993
19
10
2D
3D
TSV
AA1-1162
Ki:
10
IC50:
169
Kd:
4
EC50:
6
19
12
2D
3D
TSV
AA102_13090
IC50:
661
7
1
2D
3D
TSV
AA102_13095
IC50:
58
Kd:
1
1
1
2D
3D
TSV
AA102_17575
IC50:
12
2
1
2D
3D
TSV
AA954_14460
IC50:
2
1
1
2D
3D
TSV
AAA nuclear coregulator cancer-associated protein
Ki:
2
IC50:
243
Kd:
62
22
9
2D
3D
TSV
AAC2
IC50:
1
1
2
2D
3D
TSV
AAD21956.1
IC50:
63
1
1
2D
3D
TSV
AADAC
Ki:
5
IC50:
3
2
5
2D
3D
TSV
AADAT
Ki:
13
IC50:
398
9
5
2D
3D
TSV
AADC
IC50:
15
1
9
2D
3D
TSV
AaEcR
EC50:
34
1
4
2D
3D
TSV
AAG
IC50:
7
1
11
2D
3D
TSV
AAK1
Ki:
22
IC50:
1686
Kd:
149
24
5
2D
3D
TSV
AAO92295.1
Ki:
304
IC50:
1395
Kd:
3
EC50:
56
39
7
2D
3D
TSV
AARE
Ki:
1
IC50:
1
1
3
2D
3D
TSV
Ab N1G9
ITC:
4
1
0
2D
3D
TSV
AB164_07585
Ki:
12
IC50:
17
1
3
2D
3D
TSV
AB165_01610
Ki:
12
IC50:
17
1
3
2D
3D
TSV
AB166_11280
Ki:
12
IC50:
17
1
3
2D
3D
TSV
AB167_18060
Ki:
12
IC50:
17
1
3
2D
3D
TSV
AB168_06335
Ki:
12
IC50:
17
1
3
2D
3D
TSV
AB169_08740
Ki:
12
IC50:
17
1
3
2D
3D
TSV
AB170_00090
Ki:
12
IC50:
17
1
3
2D
3D
TSV
AB171_19425
Ki:
12
IC50:
17
1
3
2D
3D
TSV
AB552B1_00058
IC50:
2
1
1
2D
3D
TSV
AB719_18095
Ki:
3
1
1
2D
3D
TSV
AB893_00065
Ki:
12
IC50:
17
1
3
2D
3D
TSV
AB945B12_03757
IC50:
2
1
1
2D
3D
TSV
Abat
IC50:
4
1
3
2D
3D
TSV
ABC-1
EC50:
57
1
3
2D
3D
TSV
ABC003_03708
Ki:
3
1
1
2D
3D
TSV
ABCAM1_2216
IC50:
2
1
1
2D
3D
TSV
ABCB11
Ki:
16
IC50:
1673
21
4
2D
3D
TSV
ABCC1
Ki:
40
IC50:
542
Kd:
2
EC50:
1006
62
11
2D
3D
TSV
Abcc2
Ki:
66
IC50:
19
EC50:
6
18
3
2D
3D
TSV
Abcc3
Ki:
4
1
3
2D
3D
TSV
ABCC4
Ki:
2
IC50:
644
5
8
2D
3D
TSV
ABCC5
Ki:
3
IC50:
6
3
11
2D
3D
TSV
ABCC7
Ki:
1
IC50:
161
Kd:
11
EC50:
707
37
7
2D
3D
TSV
Abcc9
Kd:
51
1
3
2D
3D
TSV
ABCP
Ki:
4
IC50:
1356
EC50:
516
Other:
2
77
16
2D
3D
TSV
AbDsbA(ox)/AFDQIDNAPEE
Kd:
1
ITC:
1
2
0
2D
3D
TSV
Abelson murine leukemia viral oncogene homolog 1
Ki:
832
IC50:
2205
Kd:
1576
EC50:
100
324
23
2D
3D
TSV
Abelson murine leukemia viral oncogene homolog 2
Ki:
2
IC50:
85
Kd:
149
31
11
2D
3D
TSV
Abelson tyrosine-kinase 1 SH2 domain (ABL SH2)
Kd:
3
1
0
2D
3D
TSV
Abelson tyrosine-kinase 2 SH2 domain (Arg SH2)
Kd:
3
1
0
2D
3D
TSV
Abelson tyrosine-protein kinase 1
IC50:
111
6
15
2D
3D
TSV
Abelson-related gene protein
Ki:
2
IC50:
85
Kd:
149
31
11
2D
3D
TSV
Abeta-degrading protease
Ki:
37
IC50:
195
Kd:
1
EC50:
1
10
6
2D
3D
TSV
ABH3
IC50:
74
Kd:
1
2
6
2D
3D
TSV
Abh6
IC50:
287
9
4
2D
3D
TSV
ABHD11
IC50:
3
1
9
2D
3D
TSV
Abhd2
IC50:
196
1
5
2D
3D
TSV
ABHD6
Ki:
4
IC50:
170
11
5
2D
3D
TSV
Abhydrolase domain-containing protein 11
IC50:
3
1
9
2D
3D
TSV
Abhydrolase domain-containing protein 2
IC50:
196
1
5
2D
3D
TSV
Abhydrolase Domain-Containing Protein 6
IC50:
287
9
4
2D
3D
TSV
ABI1-binding protein 6
1
3
2D
3D
TSV
ABKPCSM17A_03582
IC50:
2
1
1
2D
3D
TSV
ABL
Ki:
825
IC50:
2141
Kd:
1555
EC50:
100
321
10
2D
3D
TSV
ABL1
Ki:
825
IC50:
2061
Kd:
1548
EC50:
100
316
9
2D
3D
TSV
ABL1(Q252H)
IC50:
32
Kd:
18
2
0
2D
3D
TSV
ABO
Ki:
7
IC50:
2
Kd:
3
1
15
2D
3D
TSV
ABP
Ki:
12
IC50:
83
9
12
2D
3D
TSV
ABP1
IC50:
17
1
4
2D
3D
TSV
ABPP
Ki:
516
IC50:
1191
Kd:
31
EC50:
105
129
26
2D
3D
TSV
Abrineurin
Kd:
6
1
12
2D
3D
TSV
Absent small and homeotic disks protein 1 homolog
IC50:
2
1
6
2D
3D
TSV
ABUW_0563
Ki:
3
1
1
2D
3D
TSV
ABW01_29210
Ki:
12
IC50:
17
1
3
2D
3D
TSV
ABW28_08200
IC50:
2
Kd:
73
2
1
2D
3D
TSV
ABW29_07060
IC50:
2
Kd:
73
2
1
2D
3D
TSV
ABW30_08355
IC50:
2
Kd:
73
2
1
2D
3D
TSV
ABW31_07355
IC50:
2
Kd:
73
2
1
2D
3D
TSV
ABW32_09260
IC50:
2
Kd:
73
2
1
2D
3D
TSV
ABW33_07270
IC50:
2
Kd:
73
2
1
2D
3D
TSV
AC
IC50:
49
3
3
2D
3D
TSV
Ac-DEVD-AFC
1
0
2D
3D
TSV
Ac-DEVD-AMC
1
0
2D
3D
TSV
Ac-IETD-AMC
1
0
2D
3D
TSV
AC-III
1
5
2D
3D
TSV
Ac-LEED-AMC
1
0
2D
3D
TSV
Ac-LEHD-AFC
1
0
2D
3D
TSV
Ac-Val-Asp-Val-Ala-Asp-AFC
1
0
2D
3D
TSV
Ac-VDVAD-AMC
1
0
2D
3D
TSV
Ac-VEID-AMC
1
0
2D
3D
TSV
Ac-YVAD-AMC
1
0
2D
3D
TSV
AC067_05500
IC50:
661
7
1
2D
3D
TSV
AC067_05505
IC50:
58
Kd:
1
1
1
2D
3D
TSV
AC067_14880
IC50:
12
2
1
2D
3D
TSV
AC3
1
5
2D
3D
TSV
AC6
1
1
2D
3D
TSV
AC789_1c06740
IC50:
12
2
1
2D
3D
TSV
AC789_1c45560
IC50:
661
7
1
2D
3D
TSV
AC789_1c45570
IC50:
58
Kd:
1
1
1
2D
3D
TSV
AC8
IC50:
33
EC50:
2
2
2
2D
3D
TSV
AC9
Ki:
2
2
10
2D
3D
TSV
ACACA kinase
IC50:
13
Kd:
258
EC50:
1047
27
15
2D
3D
TSV
Acacb
IC50:
3
2
3
2D
3D
TSV
ACAN
Kd:
12
1
5
2D
3D
TSV
ACAS2
IC50:
12
1
9
2D
3D
TSV
ACAT
IC50:
1062
32
2
2D
3D
TSV
ACAT-1
IC50:
1178
43
7
2D
3D
TSV
ACAT-2
IC50:
217
27
9
2D
3D
TSV
ACAT-related gene product 1
Ki:
17
IC50:
1715
EC50:
45
59
5
2D
3D
TSV
ACAT1
IC50:
31
5
3
2D
3D
TSV
ACAT2
IC50:
28
4
1
2D
3D
TSV
ACBD3 protein
Ki:
1
1
1
2D
3D
TSV
ACC
IC50:
29
2
5
2D
3D
TSV
ACC synthase 5
Ki:
2
IC50:
4
1
6
2D
3D
TSV
ACC-alpha
IC50:
737
34
15
2D
3D
TSV
ACC-beta
IC50:
3672
Kd:
1
42
8
2D
3D
TSV
ACC5
Ki:
2
IC50:
4
1
6
2D
3D
TSV
ACCase
IC50:
39
2
1
2D
3D
TSV
AccB
1
5
2D
3D
TSV
accC
IC50:
15
1
1
2D
3D
TSV
Accessory gene regulator protein A
IC50:
15
3
4
2D
3D
TSV
Accn1
IC50:
49
1
5
2D
3D
TSV
Accn2
IC50:
42
3
7
2D
3D
TSV
ACDase
IC50:
49
3
3
2D
3D
TSV
ACE
Ki:
143
IC50:
1521
EC50:
3
132
14
2D
3D
TSV
ace-1
IC50:
19
1
1
2D
3D
TSV
ACE-related carboxypeptidase
Ki:
44
IC50:
26
EC50:
3
9
8
2D
3D
TSV
ACE2
Ki:
44
IC50:
26
EC50:
3
9
8
2D
3D
TSV
AceCS
IC50:
12
1
9
2D
3D
TSV
AceCS1
IC50:
12
1
9
2D
3D
TSV
ACEH
Ki:
44
IC50:
26
EC50:
3
9
8
2D
3D
TSV
ACEI-ACE2
Ki:
1
IC50:
105
10
2
2D
3D
TSV
ACER2
IC50:
1
1
6
2D
3D
TSV
Acetate Operon Repressor (C-IclR)
ITC:
4
1
5
2D
3D
TSV
Acetate Operon Repressor (IclR)
ITC:
4
1
5
2D
3D
TSV
Acetate--CoA ligase
IC50:
12
1
9
2D
3D
TSV
Acetoacetyl-CoA thiolase
IC50:
163
6
5
2D
3D
TSV
Acetohydroxy-acid isomeroreductase
Ki:
4
1
3
2D
3D
TSV
Acetolactate synthase
Ki:
61
IC50:
31
7
8
2D
3D
TSV
Acetolactate synthase catalytic subunit, mitochondrial
Ki:
8
IC50:
1
2
3
2D
3D
TSV
Acetyl-CoA acetyltransferase, cytosolic
IC50:
189
23
8
2D
3D
TSV
Acetyl-CoA acetyltransferase, mitochondrial
IC50:
688
52
12
2D
3D
TSV
acetyl-CoA acetyltransferase/HMG-CoA reductase
IC50:
3
1
1
2D
3D
TSV
Acetyl-CoA carboxylase
IC50:
3746
Kd:
1
45
10
2D
3D
TSV
Acetyl-CoA carboxylase 1
IC50:
810
35
15
2D
3D
TSV
Acetyl-CoA carboxylase 1 (ACC1)
IC50:
743
35
15
2D
3D
TSV
Acetyl-CoA carboxylase 2
IC50:
3748
Kd:
1
43
10
2D
3D
TSV
Acetyl-CoA carboxylase 2 (ACC)
IC50:
3672
Kd:
1
42
8
2D
3D
TSV
Acetyl-CoA carboxylase 2 (ACC2)
IC50:
4090
Kd:
1
47
9
2D
3D
TSV
Acetyl-CoA carboxylase kinase
IC50:
3
Kd:
126
EC50:
1007
13
8
2D
3D
TSV
Acetyl-CoA carboxylase subunit A
IC50:
29
2
5
2D
3D
TSV
Acetyl-CoA synthetase
IC50:
12
1
9
2D
3D
TSV
Acetyl-CoA synthetase 1
IC50:
12
1
9
2D
3D
TSV
Acetyl-CoA transferase-like protein
IC50:
189
23
8
2D
3D
TSV
Acetyl-Coenzyme A carboxylase
IC50:
3
2
13
2D
3D
TSV
Acetyl-Coenzyme A carboxylase 2
IC50:
7
4
1
2D
3D
TSV
Acetyl-coenzyme A synthetase, cytoplasmic
IC50:
12
1
9
2D
3D
TSV
Acetyl-coenzyme A transporter 1 (AT1)
IC50:
151
1
4
2D
3D
TSV
acetylated histone H4 lysine-16
1
0
2D
3D
TSV
Acetylcholine Binding protein
Ki:
329
IC50:
3
Kd:
45
16
2
2D
3D
TSV
Acetylcholine receptor
Ki:
30
IC50:
14
Kd:
3
EC50:
16
11
5
2D
3D
TSV
Acetylcholine receptor protein alpha chain
Ki:
8
IC50:
29
EC50:
6
15
5
2D
3D
TSV
Acetylcholine receptor protein alpha chain/beta chain/delta chain /gamma chain
Ki:
3
IC50:
72
EC50:
21
7
4
2D
3D
TSV
Acetylcholine receptor protein alpha/beta/delta/gamma chain
Ki:
25
IC50:
14
Kd:
3
EC50:
4
8
4
2D
3D
TSV
Acetylcholine receptor protein delta chain
Ki:
1
IC50:
12
EC50:
12
4
6
2D
3D
TSV
Acetylcholine receptor protein epsilon chain
Ki:
2
IC50:
47
5
5
2D
3D
TSV
Acetylcholine receptor subunit alpha
Ki:
44
IC50:
29
EC50:
6
16
7
2D
3D
TSV
Acetylcholine receptor subunit beta
1
6
2D
3D
TSV
Acetylcholine receptor subunit beta-like 2
Ki:
8
IC50:
31
4
6
2D
3D
TSV
Acetylcholine receptor subunit delta
EC50:
1
1
1
2D
3D
TSV
Acetylcholine receptor subunit gamma
1
6
2D
3D
TSV
Acetylcholine receptor; alpha1/beta1/delta/gamma
Ki:
3
IC50:
72
EC50:
21
7
4
2D
3D
TSV
Acetylcholine-binding protein
Ki:
188
IC50:
1
Kd:
45
14
1
2D
3D
TSV
Acetylcholine-binding protein (AchBP)
Ki:
188
IC50:
1
Kd:
45
14
1
2D
3D
TSV
Acetylcholine-binding protein (Ls-AchBP)
Ki:
188
IC50:
1
Kd:
45
14
1
2D
3D
TSV
Acetylchol-nesterase
Ki:
1719
IC50:
15819
Kd:
248
EC50:
51
Koff:
3
Kon:
11
956
31
2D
3D
TSV
Acetylchol-nesterase (AChE)
Ki:
1719
IC50:
15640
Kd:
248
EC50:
51
Koff:
3
Kon:
11
955
22
2D
3D
TSV
Acetylchol-nesterase (EeAChE)
Ki:
650
IC50:
6290
Kd:
20
EC50:
2
435
1
2D
3D
TSV
Acetylchol-nesterase (human AChE)
Ki:
874
IC50:
6184
Kd:
204
EC50:
49
Kon:
5
496
13
2D
3D
TSV
Acetylchol-nesterase (mouse AChE)
Ki:
66
IC50:
545
Kd:
19
42
2
2D
3D
TSV
Acetylchol-nesterase 16 kDa subunit
IC50:
18
1
3
2D
3D
TSV
Acetylchol-nesterase 55 kDa subunit
IC50:
18
1
3
2D
3D
TSV
Acetylchol-nesterase and butyrylcholinesterase (AChE and BChE)
Ki:
18
IC50:
2121
Kd:
2
105
3
2D
3D
TSV
Acetylchol-nesterase precursor
Ki:
195
IC50:
3161
Kd:
24
Koff:
3
Kon:
6
210
8
2D
3D
TSV
Acetylchol-nesterase, AChE
Ki:
18
IC50:
1656
Kd:
2
99
1
2D
3D
TSV
Acetylpolyamine amidohydrolase (APAH)
IC50:
15
3
1
2D
3D
TSV
Acetylpolyamine aminohydrolase
IC50:
15
3
1
2D
3D
TSV
Acetylpolyamine oxidase (APAO)
Ki:
23
3
18
2D
3D
TSV
Acetyltransferase
EC50:
2
1
1
2D
3D
TSV
ACh-binding protein
Ki:
188
IC50:
1
Kd:
45
14
1
2D
3D
TSV
AchBP
Ki:
188
IC50:
1
Kd:
45
14
1
2D
3D
TSV
AChE
Ki:
1069
IC50:
9483
Kd:
228
EC50:
49
Koff:
3
Kon:
11
637
28
2D
3D
TSV
ACHE1
IC50:
120
4
7
2D
3D
TSV
Acid beta-galactosidase
Ki:
15
IC50:
73
19
7
2D
3D
TSV
Acid beta-glucosidase
Ki:
281
IC50:
872
Kd:
3
EC50:
163
63
13
2D
3D
TSV
Acid CDase
IC50:
49
3
3
2D
3D
TSV
Acid ceramidase
Ki:
3
IC50:
253
EC50:
1
15
7
2D
3D
TSV
Acid ceramidase (AC)
Ki:
3
IC50:
253
EC50:
1
15
7
2D
3D
TSV
Acid ceramidase-like protein
IC50:
494
19
5
2D
3D
TSV
Acid DNase
Ki:
1
1
6
2D
3D
TSV
Acid maltase
Ki:
18
IC50:
173
Kd:
2
EC50:
18
28
10
2D
3D
TSV
Acid phosphatase (acpA)
Ki:
8
1
2
2D
3D
TSV
Acid phosphatase (acpB)
Ki:
8
1
2
2D
3D
TSV
Acid phosphatase (acpC)
Ki:
8
1
2
2D
3D
TSV
Acid sphingomyelinase
Ki:
1
IC50:
140
3
9
2D
3D
TSV
Acid-sensing ion channel
IC50:
25
1
3
2D
3D
TSV
Acid-sensing ion channel 1
IC50:
45
EC50:
3
5
12
2D
3D
TSV
Acid-sensing ion channel 1/2
IC50:
1
1
3
2D
3D
TSV
Acid-sensing ion channel 2
IC50:
49
1
5
2D
3D
TSV
Acid-sensing ion channel 5
EC50:
5
1
1
2D
3D
TSV
Acid-sensitive potassium channel protein TASK-1
IC50:
1151
11
4
2D
3D
TSV
Acid-sensitive potassium channel protein TASK-2
IC50:
1
1
6
2D
3D
TSV
Acid-sensitive potassium channel protein TASK-3
IC50:
226
5
8
2D
3D
TSV
Acid-sensitive potassium channel protein TASK-4
IC50:
1
1
7
2D
3D
TSV
Acid-sensitive potassium channel TASK-1
IC50:
1149
11
3
2D
3D
TSV
Acidic alpha-glucosidase
Ki:
15
IC50:
277
30
1
2D
3D
TSV
Acidic fibroblast growth factor
IC50:
2
Kd:
116
9
6
2D
3D
TSV
Acidic mammalian chitinase
Ki:
3
IC50:
76
5
8
2D
3D
TSV
Acidic mammalian chitinase (AMCase)
Ki:
4
IC50:
287
Kd:
3
12
10
2D
3D
TSV
Acinetobacter trimeric autotransporter
IC50:
55
1
1
2D
3D
TSV
ACIX
Ki:
2
2
10
2D
3D
TSV
ACK-1
IC50:
40
1
5
2D
3D
TSV
Ack1
IC50:
40
1
5
2D
3D
TSV
ACKR2
IC50:
1
EC50:
1
1
8
2D
3D
TSV
Ackr3
Ki:
2
1
3
2D
3D
TSV
ACMSD
IC50:
57
3
5
2D
3D
TSV
ACN002_0164
Ki:
3
1
1
2D
3D
TSV
ACN002_0653
IC50:
12
2
1
2D
3D
TSV
ACN002_4371
IC50:
661
7
1
2D
3D
TSV
ACN002_4372
IC50:
58
Kd:
1
1
1
2D
3D
TSV
ACN77_13920
IC50:
661
7
1
2D
3D
TSV
ACN77_13925
IC50:
58
Kd:
1
1
1
2D
3D
TSV
ACN77_23585
IC50:
12
2
1
2D
3D
TSV
ACN81_02930
IC50:
12
2
1
2D
3D
TSV
ACN81_06320
IC50:
661
7
1
2D
3D
TSV
ACN81_06325
IC50:
58
Kd:
1
1
1
2D
3D
TSV
ACP
IC50:
30
2
6
2D
3D
TSV
ACP 2
Ki:
1
IC50:
11
1
7
2D
3D
TSV
ACP1
Ki:
10
IC50:
864
27
10
2D
3D
TSV
ACP5
Ki:
6
1
1
2D
3D
TSV
ACR
Ki:
53
1
4
2D
3D
TSV
Acr96Ac
Ki:
8
IC50:
31
4
6
2D
3D
TSV
Acra3
Ki:
105
IC50:
3
EC50:
4
8
1
2D
3D
TSV
Acra4
IC50:
8
1
6
2D
3D
TSV
AcrAB-TolC
Kd:
4
2
1
2D
3D
TSV
AcrAB-TolC multidrug efflux transport system
Kd:
4
2
1
2D
3D
TSV
Acrb
1
1
2D
3D
TSV
Acrb2
1
3
2D
3D
TSV
Acrb4
Ki:
8
1
6
2D
3D
TSV
AcrC
Ki:
42
1
8
2D
3D
TSV
Acrd
EC50:
1
1
1
2D
3D
TSV
Acre
1
1
2D
3D
TSV
AcrF
Ki:
8
IC50:
31
4
6
2D
3D
TSV
Acrg
1
1
2D
3D
TSV
Acriflavine resistance protein B
Kd:
4
2
1
2D
3D
TSV
Acrosin
Ki:
53
IC50:
196
8
6
2D
3D
TSV
Acrosin heavy chain
Ki:
53
1
4
2D
3D
TSV
Acrosin light chain
Ki:
53
1
4
2D
3D
TSV
ACS
IC50:
13
2
16
2D
3D
TSV
ACS5
Ki:
2
IC50:
4
1
6
2D
3D
TSV
ACSS2
IC50:
12
1
9
2D
3D
TSV
ACSVL5
IC50:
75
2
4
2D
3D
TSV
ACT-2
IC50:
7
1
6
2D
3D
TSV
ACT1
IC50:
3
1
6
2D
3D
TSV
ACT1 (R183K)
IC50:
3
1
0
2D
3D
TSV
ACT1 (R335K)
IC50:
3
1
0
2D
3D
TSV
ACT3
IC50:
5
2
4
2D
3D
TSV
ACTA
IC50:
2
1
4
2D
3D
TSV
ACTA1
IC50:
2
1
4
2D
3D
TSV
ACTH receptor
IC50:
1
1
5
2D
3D
TSV
ACTH-R
IC50:
1
1
5
2D
3D
TSV
Actin
IC50:
6
1
6
2D
3D
TSV
Actin (R183K)
IC50:
3
1
0
2D
3D
TSV
Actin, alpha skeletal muscle
IC50:
2
1
4
2D
3D
TSV
Actin, alpha skeletal muscle, intermediate form
IC50:
2
1
4
2D
3D
TSV
Actin-like protein 2
IC50:
1
1
7
2D
3D
TSV
Actin-related protein 2
IC50:
1
1
7
2D
3D
TSV
Activated blood-coagulation factor II
Ki:
41
IC50:
2
3
1
2D
3D
TSV
Activated CDC42 kinase 1
IC50:
40
1
5
2D
3D
TSV
Activated CDC42 kinase 1 (ACK-1)
Ki:
106
IC50:
624
Kd:
126
44
5
2D
3D
TSV
Activated coagulation factor X (FXa)
Ki:
4528
IC50:
2951
Kd:
15
Koff:
6
Kon:
5
394
4
2D
3D
TSV
Activated factor Xa heavy chain
Ki:
4528
IC50:
2951
Kd:
15
Koff:
6
Kon:
5
394
4
2D
3D
TSV
Activated protein C cofactor
Ki:
237
IC50:
180
67
16
2D
3D
TSV
Activating signal cointegrator 1 complex subunit 3-like 1
IC50:
56
6
8
2D
3D
TSV
Activating transcription factor 1
IC50:
31
1
5
2D
3D
TSV
Activating transcription factor 2
1
0
2D
3D
TSV
Activating transcription factor 2-GST fusion
1
0
2D
3D
TSV
Activation inducer molecule
IC50:
26
Kd:
6
3
2
2D
3D
TSV
Activation molecule 3
IC50:
5
2
4
2D
3D
TSV
Activation peptide
Ki:
1101
IC50:
698
Kd:
13
EC50:
3
205
10
2D
3D
TSV
Activation peptide fragment 1
Ki:
5359
IC50:
4226
Kd:
85
EC50:
18
Kon:
7
Other:
1
ITC:
19
592
15
2D
3D
TSV
Activation peptide fragment 2
Ki:
5359
IC50:
4226
Kd:
85
EC50:
18
Kon:
7
Other:
1
ITC:
19
592
15
2D
3D
TSV
Activator of S phase kinase
1
8
2D
3D
TSV
Activator of S phase kinase DBF4/Cell division cycle 7-related protein kinase
Ki:
21
IC50:
273
Kd:
3
EC50:
11
16
3
2D
3D
TSV
Activator protein 1
IC50:
168
Kd:
1
EC50:
5
19
5
2D
3D
TSV
Activin A receptor type II-like protein kinase of 53kD
Ki:
63
IC50:
2575
Kd:
6
EC50:
250
82
6
2D
3D
TSV
Activin beta-A chain
IC50:
11
1
2
2D
3D
TSV
Activin receptor type I
IC50:
453
Kd:
127
27
2
2D
3D
TSV
Activin receptor type-1
IC50:
453
Kd:
127
27
2
2D
3D
TSV
Activin receptor type-1 (ACVR1)
IC50:
177
2
0
2D
3D
TSV
Activin receptor type-1 (ALK2 FOP) (R206H aa 172-499)
IC50:
88
1
0
2D
3D
TSV
Activin receptor type-1B
IC50:
201
Kd:
124
25
8
2D
3D
TSV
Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
IC50:
201
Kd:
124
25
8
2D
3D
TSV
Activin receptor type-2A
IC50:
2
Kd:
119
6
8
2D
3D
TSV
Activin receptor type-2B
IC50:
6
Kd:
124
10
3
2D
3D
TSV
Activin receptor-like kinase 1 (ALK-1)
IC50:
297
Kd:
121
23
4
2D
3D
TSV
Activin receptor-like kinase 1 (ALK1)(aa 166-493)
IC50:
88
1
0
2D
3D
TSV
Activin receptor-like kinase 2
IC50:
453
Kd:
127
27
2
2D
3D
TSV
Activin receptor-like kinase 2 (ALK-2)
IC50:
453
Kd:
127
27
2
2D
3D
TSV
Activin receptor-like kinase 2 (ALK-2)(aa 172-499)
IC50:
177
2
0
2D
3D
TSV
Activin receptor-like kinase 2 (ALK2/ACVR1)
IC50:
453
Kd:
127
27
2
2D
3D
TSV
Activin receptor-like kinase 3 (ALK-3)
IC50:
223
Kd:
121
20
4
2D
3D
TSV
Activin receptor-like kinase 3 (ALK3) (aa 198-525)
IC50:
88
1
0
2D
3D
TSV
Activin receptor-like kinase 5
Ki:
63
IC50:
2575
Kd:
6
EC50:
250
82
6
2D
3D
TSV
Activin receptor-like kinase 5 (ALK-5)(aa 162-503)
IC50:
88
1
0
2D
3D
TSV
Activin receptor-like kinase 6
IC50:
27
1
4
2D
3D
TSV
ACTR-I
IC50:
453
Kd:
127
27
2
2D
3D
TSV
ActR-IB
IC50:
5
1
2
2D
3D
TSV
ACTR2
IC50:
1
1
7
2D
3D
TSV
ActRIA
IC50:
38
EC50:
3
3
4
2D
3D
TSV
ActRIB
IC50:
5
1
2
2D
3D
TSV
ACU57_00610
IC50:
12
2
1
2D
3D
TSV
ACU57_19295
IC50:
58
Kd:
1
1
1
2D
3D
TSV
ACU57_19300
IC50:
661
7
1
2D
3D
TSV
ACU90_10770
IC50:
12
2
1
2D
3D
TSV
ACU90_27610
IC50:
58
Kd:
1
1
1
2D
3D
TSV
ACU90_27615
IC50:
661
7
1
2D
3D
TSV
Acute myeloid leukemia 1 protein
IC50:
243
Other:
6
6
24
2D
3D
TSV
Acute-phase response factor
Ki:
18
IC50:
220
Kd:
52
13
4
2D
3D
TSV
ACVI
1
1
2D
3D
TSV
Acvr
IC50:
38
EC50:
3
3
4
2D
3D
TSV
ACVR1
IC50:
453
Kd:
127
27
2
2D
3D
TSV
ACVR1B
IC50:
201
Kd:
124
25
8
2D
3D
TSV
ACVR2A
IC50:
2
Kd:
119
6
8
2D
3D
TSV
ACVR2B
IC50:
6
Kd:
124
10
3
2D
3D
TSV
ACVRL1
IC50:
297
Kd:
121
23
4
2D
3D
TSV
Acvrlk1
IC50:
5
1
4
2D
3D
TSV
ACVRLK2
IC50:
453
Kd:
127
27
2
2D
3D
TSV
Acvrlk4
IC50:
5
1
2
2D
3D
TSV
Acyl carrier protein, mitochondrial
IC50:
30
2
6
2D
3D
TSV
Acyl coA-diacylglycerol acyl transferase 1 (DGAT1)
Ki:
17
IC50:
1715
EC50:
45
59
5
2D
3D
TSV
Acyl coenzyme A:cholesterol acyltransferase
Ki:
421
IC50:
224
30
20
2D
3D
TSV
Acyl coenzyme A:cholesterol acyltransferase 1
IC50:
687
51
11
2D
3D
TSV
Acyl coenzyme A:cholesterol acyltransferase 2
IC50:
191
25
9
2D
3D
TSV
Acyl-activating enzyme
IC50:
12
1
9
2D
3D
TSV
Acyl-CoA desaturase
IC50:
1199
33
12
2D
3D
TSV
Acyl-CoA desaturase 1
IC50:
920
33
6
2D
3D
TSV
Acyl-CoA retinol O-fatty-acyltransferase
IC50:
822
Other:
2
31
12
2D
3D
TSV
Acyl-CoA synthetase short-chain family member 2
IC50:
12
1
9
2D
3D
TSV
Acyl-CoA wax alcohol acyltransferase 1
IC50:
11
1
4
2D
3D
TSV
Acyl-CoA wax alcohol acyltransferase 2
IC50:
11
1
4
2D
3D
TSV
Acyl-CoA-desaturase 4
IC50:
485
5
6
2D
3D
TSV
Acyl-CoA: cholesterol acyltransferase (ACAT)
Ki:
421
IC50:
749
77
27
2D
3D
TSV
Acyl-CoA:cholesterol acyltransferase
IC50:
1059
31
1
2D
3D
TSV
Acyl-CoA:dihydroxyacetonephos-hateacyltransferase
Ki:
3
IC50:
4
1
5
2D
3D
TSV
Acyl-CoA:monoacylglycerol acyltransferase 2
IC50:
194
5
8
2D
3D
TSV
Acyl-CoA:monoacylglycerol acyltransferase 2 (MOGAT2)
IC50:
192
5
7
2D
3D
TSV
Acyl-coenzyme A:cholesterol acyltransferase 1
IC50:
193
10
6
2D
3D
TSV
Acyl-coenzyme A:cholesterol acyltransferase 1 (ACAT1)
IC50:
525
47
8
2D
3D
TSV
Acyl-coenzyme A:cholesterol acyltransferase 2
IC50:
28
4
1
2D
3D
TSV
Acyl-peptide hydrolase
Ki:
1
IC50:
1
1
3
2D
3D
TSV
Acyl-protein thioesterase 1
Ki:
5
IC50:
26
4
5
2D
3D
TSV
Acyl-protein thioesterase 1 (APT1 I75L)
Ki:
2
1
0
2D
3D
TSV
Acyl-protein thioesterase 1 (APT1 I75L/S82A)
Ki:
2
1
0
2D
3D
TSV
Acyl-protein thioesterase 1 (APT1 I75L/S82A/Q83P)
Ki:
2
1
0
2D
3D
TSV
Acyl-protein thioesterase 1 (APT1 I75L/S82A/Q83P/R149H/A150R/S151A)
Ki:
2
1
0
2D
3D
TSV
Acyl-protein thioesterase 1 (APT1 L176M)
Ki:
2
1
0
2D
3D
TSV
Acyl-protein thioesterase 1 (APT1 Q83P)
Ki:
2
1
0
2D
3D
TSV
Acyl-protein thioesterase 1 (APT1 WT)
Ki:
5
IC50:
26
4
5
2D
3D
TSV
Acyl-protein thioesterase 1/2
Ki:
1
IC50:
111
7
1
2D
3D
TSV
Acyl-protein thioesterase 2
Ki:
10
IC50:
28
Kd:
4
4
4
2D
3D
TSV
Acyl-protein thioesterase 2 (APT2 H152R)
Ki:
2
1
0
2D
3D
TSV
Acyl-protein thioesterase 2 (APT2 L78I)
Ki:
2
1
0
2D
3D
TSV
Acyl-protein thioesterase 2 (APT2 L78I/A85S)
Ki:
2
1
0
2D
3D
TSV
Acyl-protein thioesterase 2 (APT2 L78I/A85S/P86Q)
Ki:
2
1
0
2D
3D
TSV
Acyl-protein thioesterase 2 (APT2 L78I/A85S/P86Q/H152R/R153A/A154S)
Ki:
2
1
0
2D
3D
TSV
Acyl-protein thioesterase 2 (APT2 M178L)
Ki:
2
1
0
2D
3D
TSV
Acyl-protein thioesterase 2 (APT2 P86Q)
Ki:
2
1
0
2D
3D
TSV
Acyl-protein thioesterase 2 (APT2 S122A)
IC50:
3
Kd:
4
1
0
2D
3D
TSV
Acyl-protein thioesterase 2 (APT2 WT)
Ki:
10
IC50:
28
Kd:
4
4
4
2D
3D
TSV
Acylamino-acid-releasing enzyme
Ki:
1
IC50:
1
1
3
2D
3D
TSV
Acylaminoacyl-peptidase
Ki:
1
IC50:
1
1
3
2D
3D
TSV
Acylcholine acylhydrolase
Ki:
504
IC50:
3536
Kd:
9
305
6
2D
3D
TSV
Acylsphingosine deacylase
IC50:
49
3
3
2D
3D
TSV
Acylsphingosine deacylase 2
IC50:
4
2
8
2D
3D
TSV
Acylsphingosine deacylase 3-like
IC50:
1
1
6
2D
3D
TSV
Acylsphingosine kinase
Ki:
4
IC50:
1
3
8
2D
3D
TSV
AD3
Ki:
26
IC50:
2232
EC50:
158
80
10
2D
3D
TSV
AD3LP
IC50:
8
1
5
2D
3D
TSV
AD5
IC50:
8
1
5
2D
3D
TSV
ADA
Ki:
464
IC50:
1
Other:
3
36
3
2D
3D
TSV
ADABP
Ki:
600
IC50:
4784
Kd:
26
EC50:
2
246
3
2D
3D
TSV
ADAM 17
Ki:
109
IC50:
506
31
8
2D
3D
TSV
ADAM-TS 11
IC50:
57
Other:
8
2
0
2D
3D
TSV
ADAM-TS 13
IC50:
3
2
8
2D
3D
TSV
ADAM-TS 6
IC50:
265
2
7
2D
3D
TSV
ADAM-TS13
IC50:
3
2
8
2D
3D
TSV
ADAM-TS6
IC50:
265
2
7
2D
3D
TSV
ADAM10
Ki:
20
IC50:
774
30
6
2D
3D
TSV
ADAM12
IC50:
5
1
7
2D
3D
TSV
ADAM17
Ki:
448
IC50:
3721
EC50:
10
142
11
2D
3D
TSV
ADAM9
Ki:
2
IC50:
67
12
5
2D
3D
TSV
ADAMTS-13
IC50:
3
2
8
2D
3D
TSV
ADAMTS-5 (Aggrecanase-2)
IC50:
57
Other:
8
2
0
2D
3D
TSV
ADAMTS-6
IC50:
265
2
7
2D
3D
TSV
ADAMTS1
Ki:
5
IC50:
7
3
7
2D
3D
TSV
ADAMTS13
IC50:
3
2
8
2D
3D
TSV
ADAMTS5
Ki:
14
IC50:
1563
35
6
2D
3D
TSV
Adapter protein GRB2
IC50:
16
1
4
2D
3D
TSV
Adaptor molecule disabled-2
Ki:
3
1
7
2D
3D
TSV
Adaptor protein complex AP-1 subunit beta-1
Kd:
1
1
7
2D
3D
TSV
Adaptor-associated kinase 1
Ki:
22
IC50:
1686
Kd:
149
24
5
2D
3D
TSV
Adaptor-related protein complex 1 subunit beta-1
Kd:
1
1
7
2D
3D
TSV
ADC-11
Ki:
3
IC50:
1
1
1
2D
3D
TSV
ADC-14 protein
IC50:
2
1
1
2D
3D
TSV
ADC-16 protein
IC50:
2
1
1
2D
3D
TSV
ADC-18 protein
IC50:
2
1
1
2D
3D
TSV
ADC-7 beta-lactamase (ADC-7)
Ki:
2
Kd:
2
ITC:
2
1
0
2D
3D
TSV
ADCK3
IC50:
1
Kd:
136
8
7
2D
3D
TSV
ADCK4
IC50:
1
Kd:
125
7
4
2D
3D
TSV
ADCP-I
IC50:
5
2
4
2D
3D
TSV
ADCP2
Ki:
600
IC50:
4784
Kd:
26
EC50:
2
246
3
2D
3D
TSV
Adcy1
Ki:
4
IC50:
6
EC50:
3
3
1
2D
3D
TSV
ADCY2
1
6
2D
3D
TSV
ADCY3
1
5
2D
3D
TSV
ADCY4
Ki:
9
1
7
2D
3D
TSV
ADCY6
1
4
2D
3D
TSV
ADCY7
1
3
2D
3D
TSV
ADCY8
IC50:
33
EC50:
2
2
2
2D
3D
TSV
ADCY9
Ki:
2
2
10
2D
3D
TSV
Adenomatous polyposis coli protein
IC50:
130
Kd:
50
3
7
2D
3D
TSV
ADENOSINE
Ki:
4
IC50:
160
9
4
2D
3D
TSV
Adenosine 5'-monophosphoramidase
Ki:
6
IC50:
2
Kd:
12
3
4
2D
3D
TSV
Adenosine 5-phosphotransferase
Ki:
4
IC50:
160
9
4
2D
3D
TSV
ADENOSINE A1
Ki:
10381
IC50:
996
Kd:
113
EC50:
626
Koff:
2
Kon:
2
Other:
10
617
19
2D
3D
TSV
ADENOSINE A1 high
Ki:
5231
IC50:
520
Kd:
20
EC50:
261
296
9
2D
3D
TSV
ADENOSINE A1 low
Ki:
5231
IC50:
520
Kd:
20
EC50:
261
296
9
2D
3D
TSV
Adenosine A1 receptor
Ki:
1244
IC50:
88
Kd:
14
EC50:
127
72
8
2D
3D
TSV
Adenosine A1 receptor (A1)
Ki:
3984
IC50:
435
Kd:
6
EC50:
136
255
1
2D
3D
TSV
Adenosine A1 receptor (A1AR)
Ki:
5130
IC50:
462
Kd:
93
EC50:
365
Koff:
2
Kon:
2
Other:
10
389
9
2D
3D
TSV
Adenosine A1-receptor
Ki:
5130
IC50:
462
Kd:
93
EC50:
365
Koff:
2
Kon:
2
Other:
10
389
9
2D
3D
TSV
ADENOSINE A2
Ki:
6720
IC50:
634
Kd:
44
EC50:
289
414
6
2D
3D
TSV
Adenosine A2 receptor
Ki:
3534
IC50:
208
Kd:
12
EC50:
190
222
5
2D
3D
TSV
ADENOSINE A2a
Ki:
8962
IC50:
685
Kd:
56
EC50:
354
502
5
2D
3D
TSV
Adenosine A2a receptor
Ki:
133
IC50:
109
EC50:
1
14
4
2D
3D
TSV
Adenosine A2a receptor (A2a)
Ki:
2346
IC50:
52
Kd:
12
EC50:
66
159
1
2D
3D
TSV
Adenosine A2A receptor (A2AAR)
Ki:
6616
IC50:
633
Kd:
44
EC50:
288
405
4
2D
3D
TSV
ADENOSINE A2B
Ki:
2940
IC50:
1051
Kd:
21
EC50:
463
198
1
2D
3D
TSV
Adenosine A2b receptor
Ki:
10
IC50:
4
Kd:
1
7
3
2D
3D
TSV
ADENOSINE A3
Ki:
101
8
5
2D
3D
TSV
Adenosine A3 receptor
Ki:
643
IC50:
2
EC50:
11
66
5
2D
3D
TSV
Adenosine A3 receptor (A3AR)
Ki:
5929
IC50:
554
Kd:
15
EC50:
184
353
6
2D
3D
TSV
Adenosine aminohydrolase
Ki:
537
IC50:
10
Other:
3
51
7
2D
3D
TSV
Adenosine deaminase
Ki:
547
IC50:
10
Other:
3
53
10
2D
3D
TSV
Adenosine deaminase 3 (SanADA3)
Ki:
2
1
1
2D
3D
TSV
Adenosine deaminase complexing protein
IC50:
5
2
4
2D
3D
TSV
Adenosine deaminase complexing protein 2
Ki:
600
IC50:
4784
Kd:
26
EC50:
2
246
3
2D
3D
TSV
Adenosine diphosphoribose pyrophosphatase
IC50:
1
1
5
2D
3D
TSV
Adenosine kinase
Ki:
121
IC50:
995
Kd:
3
42
18
2D
3D
TSV
Adenosine Kinase (AK)
Ki:
4
IC50:
160
9
4
2D
3D
TSV
Adenosine monophosphate-activated protein kinase (AMPK gamma 1, beta 1 and alpha 1)
IC50:
15
Kd:
29
EC50:
281
20
5
2D
3D
TSV
Adenosine Phosphosulfate Reductase (APSR)
Kd:
10
1
5
2D
3D
TSV
Adenosine receptor
Ki:
4076
IC50:
444
Kd:
8
EC50:
140
269
10
2D
3D
TSV
Adenosine receptor A1
Ki:
9177
IC50:
900
Kd:
99
EC50:
503
Koff:
2
Kon:
2
Other:
10
586
13
2D
3D
TSV
Adenosine receptor A1 (A1)
Ki:
5171
IC50:
462
Kd:
93
EC50:
365
Koff:
2
Kon:
2
Other:
10
391
10
2D
3D
TSV
Adenosine receptor A1 (hA1)
Ki:
5130
IC50:
462
Kd:
93
EC50:
365
Koff:
2
Kon:
2
Other:
10
389
9
2D
3D
TSV
Adenosine receptor A2
Ki:
8
2
2
2D
3D
TSV
Adenosine receptor A2a
Ki:
6730
IC50:
742
Kd:
44
EC50:
289
411
7
2D
3D
TSV
Adenosine receptor A2a and A3
Ki:
2858
IC50:
52
Kd:
12
EC50:
66
180
4
2D
3D
TSV
Adenosine receptor A2b
Ki:
2984
IC50:
1054
Kd:
23
EC50:
463
207
3
2D
3D
TSV
Adenosine receptor A2B (A2B)
Ki:
2940
IC50:
1051
Kd:
21
EC50:
463
198
1
2D
3D
TSV
Adenosine receptor A3
Ki:
6159
IC50:
564
Kd:
15
EC50:
195
361
11
2D
3D
TSV
Adenosine receptor A3 (A3)
Ki:
62
IC50:
7
3
0
2D
3D
TSV
Adenosine receptors A1
Ki:
3984
IC50:
435
Kd:
6
EC50:
136
255
1
2D
3D
TSV
Adenosine receptors A2a
Ki:
2346
IC50:
52
Kd:
12
EC50:
66
159
1
2D
3D
TSV
Adenosine Receptors A2a (A2a)
Ki:
2346
IC50:
52
Kd:
12
EC50:
66
159
1
2D
3D
TSV
Adenosine receptors A2b
Ki:
2940
IC50:
1051
Kd:
21
EC50:
463
198
1
2D
3D
TSV
Adenosine receptors; A2a & A2b
Ki:
2940
IC50:
1051
Kd:
21
EC50:
463
198
1
2D
3D
TSV
Adenosine transporter
Ki:
4
3
13
2D
3D
TSV
Adenosine transporter (AdT)
Ki:
5130
IC50:
462
Kd:
93
EC50:
365
Koff:
2
Kon:
2
Other:
10
389
9
2D
3D
TSV
Adenosine transporter 1
Ki:
36
2
1
2D
3D
TSV
Adenosine-5''-phosphosulfate 3''-phosphotransferase
EC50:
3
1
8
2D
3D
TSV
Adenosinetr-phosphatase
IC50:
4
1
1
2D
3D
TSV
Adenosylhom-cysteinase
Ki:
136
IC50:
245
55
16
2D
3D
TSV
Adenosylhom-cysteinase 2
IC50:
5
1
10
2D
3D
TSV
Adenylate cyclase
Ki:
33
IC50:
230
Kd:
8
EC50:
76
19
26
2D
3D
TSV
Adenylate cyclase Forskolin
Ki:
4
3
1
2D
3D
TSV
Adenylate cyclase homolog
IC50:
4
1
10
2D
3D
TSV
Adenylate cyclase type 10
IC50:
4
1
10
2D
3D
TSV
Adenylate cyclase type 2
Ki:
5
IC50:
2
2
7
2D
3D
TSV
Adenylate cyclase type 3
Ki:
4
3
6
2D
3D
TSV
Adenylate cyclase type 4
Ki:
9
1
8
2D
3D
TSV
Adenylate cyclase type 5
IC50:
5
EC50:
17
4
1
2D
3D
TSV
Adenylate cyclase type 6
1
5
2D
3D
TSV
Adenylate cyclase type 7
1
3
2D
3D
TSV
Adenylate cyclase type 8
IC50:
33
EC50:
2
2
4
2D
3D
TSV
Adenylate cyclase type 9
Ki:
2
2
10
2D
3D
TSV
Adenylate cyclase type I
Kd:
17
1
1
2D
3D
TSV
Adenylate cyclase type II
Ki:
5
IC50:
2
2
7
2D
3D
TSV
Adenylate cyclase type III
1
5
2D
3D
TSV
Adenylate cyclase type IV
Ki:
9
1
8
2D
3D
TSV
Adenylate cyclase type IX
Ki:
2
IC50:
5
EC50:
17
6
11
2D
3D
TSV
Adenylate cyclase type V
IC50:
85
Kd:
8
EC50:
20
10
7
2D
3D
TSV
Adenylate cyclase type VI
1
5
2D
3D
TSV
Adenylate cyclase type VII
1
3
2D
3D
TSV
Adenylate cyclase type VIII
IC50:
33
EC50:
2
2
4
2D
3D
TSV
Adenylate cyclase, olfactive type
1
5
2D
3D
TSV
Adenylate cyclase-stimulating G alpha protein
IC50:
8
1
9
2D
3D
TSV
Adenylate kinase 1
Ki:
34
2
4
2D
3D
TSV
Adenylate kinase 2
Ki:
60
6
13
2D
3D
TSV
Adenylate kinase 2, mitochondrial
Ki:
60
6
13
2D
3D
TSV
Adenylate kinase 3
Ki:
42
5
1
2D
3D
TSV
Adenylate kinase 3 alpha like 1
Ki:
42
5
1
2D
3D
TSV
Adenylate kinase 3 alpha-like 1
Ki:
42
5
1
2D
3D
TSV
Adenylate kinase 3-like
Ki:
1
1
7
2D
3D
TSV
Adenylate kinase 4
Ki:
1
1
7
2D
3D
TSV
Adenylate kinase isoenzyme 1
IC50:
2
1
1
2D
3D
TSV
Adenylate kinase isoenzyme 4, mitochondrial
Ki:
1
1
7
2D
3D
TSV
Adenylate monophosphate kinase
Ki:
56
6
3
2D
3D
TSV
Adenylosuccinate synthetase 2
IC50:
3
1
5
2D
3D
TSV
Adenylosuccinate synthetase isozyme 2
IC50:
3
1
5
2D
3D
TSV
Adenylosuccinate synthetase, acidic isozyme
IC50:
3
1
5
2D
3D
TSV
Adenylyl cyclase 2
Ki:
5
IC50:
2
2
7
2D
3D
TSV
Adenylyl cyclase 3
1
5
2D
3D
TSV
Adenylyl cyclase 4
Ki:
9
1
8
2D
3D
TSV
Adenylyl cyclase 5
IC50:
5
EC50:
17
4
1
2D
3D
TSV
Adenylyl cyclase 6
1
5
2D
3D
TSV
Adenylyl cyclase 7
1
4
2D
3D
TSV
Adenylyl cyclase 8
IC50:
33
EC50:
2
2
4
2D
3D
TSV
Adenylyl cyclase 9
Ki:
2
2
10
2D
3D
TSV
Adenylyl-sulfate kinase
EC50:
3
1
8
2D
3D
TSV
Adenylylsulfate 3''-phosphotransferase
EC50:
3
1
8
2D
3D
TSV
ADF
Ki:
1
IC50:
10
2
8
2D
3D
TSV
Adh-2
IC50:
2
1
7
2D
3D
TSV
ADH-B2
IC50:
2
1
7
2D
3D
TSV
Adh2
IC50:
2
1
7
2D
3D
TSV
ADH5
IC50:
87
3
4
2D
3D
TSV
Adhesin Ata autotransporter
IC50:
55
1
1
2D
3D
TSV
Adhesin protein fimH
IC50:
86
Kd:
4
5
3
2D
3D
TSV
Adhesion inhibitory receptor molecule 1
IC50:
10
Kd:
9
3
6
2D
3D
TSV
Adhesion molecule in glia
1
6
2D
3D
TSV
ADHX
IC50:
87
3
4
2D
3D
TSV
Adipocyte acid phosphatase
Ki:
10
IC50:
864
27
10
2D
3D
TSV
Adipocyte lipid-binding protein
Ki:
116
IC50:
538
Kd:
34
24
5
2D
3D
TSV
Adipocyte membrane protein
IC50:
103
3
3
2D
3D
TSV
Adipocyte-type fatty acid-binding protein
Ki:
2
1
1
2D
3D
TSV
Adiponectin receptor protein 1
Kd:
1
1
6
2D
3D
TSV
Adiponectin receptor protein 2
Kd:
1
1
4
2D
3D
TSV
ADIPOR1
Kd:
1
1
6
2D
3D
TSV
ADIPOR2
Kd:
1
1
4
2D
3D
TSV
Adipose triglyceride lipase
IC50:
52
2
16
2D
3D
TSV
Adipose-specific phospholipase A2
IC50:
56
1
7
2D
3D
TSV
Adipsin
Ki:
2
IC50:
4003
Kd:
26
34
8
2D
3D
TSV
ADK
Ki:
13
IC50:
5
1
5
2D
3D
TSV
ADM2
IC50:
8
1
3
2D
3D
TSV
ADMP-2
IC50:
57
Other:
8
2
0
2D
3D
TSV
Adn
IC50:
2
1
1
2D
3D
TSV
AdoHcyase
Ki:
11
IC50:
20
7
7
2D
3D
TSV
AdoHcyase 2
IC50:
5
1
10
2D
3D
TSV
adoK
Ki:
13
IC50:
5
1
5
2D
3D
TSV
AdoMet synthetase 1
Ki:
20
3
3
2D
3D
TSV
AdoMet synthetase 2
Ki:
28
IC50:
6
4
1
2D
3D
TSV
ADORA1
Ki:
5568
IC50:
482
Kd:
93
EC50:
490
Koff:
2
Kon:
2
Other:
10
412
14
2D
3D
TSV
ADORA2
Ki:
6616
IC50:
633
Kd:
44
EC50:
288
405
4
2D
3D
TSV
ADORA2A
Ki:
6618
IC50:
633
Kd:
44
EC50:
288
405
5
2D
3D
TSV
ADORA2B
Ki:
2940
IC50:
1051
Kd:
21
EC50:
463
198
1
2D
3D
TSV
ADORA3
Ki:
62
IC50:
1
6
4
2D
3D
TSV
Adora3 protein
Ki:
44
4
3
2D
3D
TSV
ADP-glucose receptor
Ki:
703
IC50:
973
Kd:
1
EC50:
123
39
4
2D
3D
TSV
ADP-ribose diphosphatase
IC50:
1
1
5
2D
3D
TSV
ADP-ribose glycohydrolase ARH3
IC50:
50
EC50:
3
3
0
2D
3D
TSV
ADP-ribose glycohydrolase MACROD1
Kd:
1
1
3
2D
3D
TSV
ADP-ribose glycohydrolase MACROD2
Kd:
1
1
9
2D
3D
TSV
ADP-ribose phosphohydrolase
IC50:
1
1
5
2D
3D
TSV
ADP-ribose pyrophosphatase, mitochondrial
IC50:
1
1
5
2D
3D
TSV
ADP-ribosyl cyclase 1
IC50:
86
2
4
2D
3D
TSV
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
IC50:
86
2
4
2D
3D
TSV
ADP-ribosylation factor 1
Kd:
1
1
5
2D
3D
TSV
ADP-ribosylation factor 6
IC50:
159
1
4
2D
3D
TSV
ADP-ribosylation factor GTPase-activating protein 1
IC50:
91
1
1
2D
3D
TSV
ADP-ribosylhydrolase 3
IC50:
50
EC50:
3
3
0
2D
3D
TSV
ADP-ribosyltransferase diphtheria toxin-like 1
Ki:
1174
IC50:
3474
Kd:
178
EC50:
309
171
5
2D
3D
TSV
ADP-ribosyltransferase diphtheria toxin-like 10
IC50:
257
EC50:
2
16
6
2D
3D
TSV
ADP-ribosyltransferase diphtheria toxin-like 11
IC50:
56
3
6
2D
3D
TSV
ADP-ribosyltransferase diphtheria toxin-like 12
IC50:
25
9
6
2D
3D
TSV
ADP-ribosyltransferase diphtheria toxin-like 14
IC50:
1713
4
6
2D
3D
TSV
ADP-ribosyltransferase diphtheria toxin-like 15
IC50:
20
7
5
2D
3D
TSV
ADP-ribosyltransferase diphtheria toxin-like 16
IC50:
2
2
5
2D
3D
TSV
ADP-ribosyltransferase diphtheria toxin-like 17
IC50:
7
4
8
2D
3D
TSV
ADP-ribosyltransferase diphtheria toxin-like 2
IC50:
72
Kd:
1
8
3
2D
3D
TSV
ADP-ribosyltransferase diphtheria toxin-like 3
IC50:
77
Kd:
22
23
6
2D
3D
TSV
ADP-ribosyltransferase diphtheria toxin-like 4
IC50:
40
11
6
2D
3D
TSV
ADP-ribosyltransferase diphtheria toxin-like 5
IC50:
1
1
3
2D
3D
TSV
ADP-ribosyltransferase diphtheria toxin-like 6
IC50:
1
1
4
2D
3D
TSV
ADP-ribosyltransferase diphtheria toxin-like 7
IC50:
59
12
4
2D
3D
TSV
ADP-ribosyltransferase diphtheria toxin-like 8
IC50:
197
Kd:
11
13
8
2D
3D
TSV
ADP-sugar pyrophosphatase
IC50:
1
1
5
2D
3D
TSV
ADPG
IC50:
7
1
11
2D
3D
TSV
ADPG-R
Ki:
703
IC50:
973
Kd:
1
EC50:
123
39
4
2D
3D
TSV
AdPLA
IC50:
56
1
7
2D
3D
TSV
ADPR-PPase
IC50:
1
1
5
2D
3D
TSV
ADPRC 1
IC50:
86
2
4
2D
3D
TSV
ADPRHL2
IC50:
50
EC50:
3
3
0
2D
3D
TSV
ADPRT
Ki:
1174
IC50:
3474
Kd:
178
EC50:
309
171
5
2D
3D
TSV
ADPRT 1
Ki:
1174
IC50:
3474
Kd:
178
EC50:
309
171
5
2D
3D
TSV
ADPRT-2
IC50:
72
Kd:
1
8
3
2D
3D
TSV
ADPRT-3
IC50:
43
Kd:
2
10
6
2D
3D
TSV
Adprt2
IC50:
72
Kd:
1
8
3
2D
3D
TSV
ADPRT3
IC50:
43
Kd:
2
10
6
2D
3D
TSV
ADPRTL1
IC50:
40
11
6
2D
3D
TSV
Adprtl2
IC50:
72
Kd:
1
8
3
2D
3D
TSV
ADPRTL3
IC50:
43
Kd:
2
10
6
2D
3D
TSV
ADRA1A
Ki:
3290
IC50:
456
Kd:
4
EC50:
571
254
26
2D
3D
TSV
ADRA1B
Ki:
242
12
5
2D
3D
TSV
Adra1b protein
Ki:
8
1
1
2D
3D
TSV
ADRA1C
Ki:
1947
IC50:
302
Kd:
4
EC50:
336
245
22
2D
3D
TSV
ADRA1D
Ki:
1301
IC50:
154
EC50:
235
129
4
2D
3D
TSV
ADRA2A
Ki:
90
IC50:
2
EC50:
1
17
2
2D
3D
TSV
ADRA2B
Ki:
809
IC50:
33
Kd:
8
EC50:
100
137
12
2D
3D
TSV
ADRA2C
Ki:
76
3
2
2D
3D
TSV
ADRA2L1
Ki:
665
IC50:
32
Kd:
8
EC50:
96
114
6
2D
3D
TSV
ADRA2R
Ki:
65
IC50:
2
EC50:
1
15
0
2D
3D
TSV
ADRA2RL1
Ki:
665
IC50:
32
Kd:
8
EC50:
96
114
6
2D
3D
TSV
ADRAR
Ki:
65
IC50:
2
EC50:
1
15
0
2D
3D
TSV
ADRB1
Ki:
539
IC50:
663
Kd:
444
EC50:
924
205
7
2D
3D
TSV
ADRB1R
Ki:
483
IC50:
626
Kd:
136
EC50:
877
174
6
2D
3D
TSV
ADRB1R, B1AR
Ki:
239
IC50:
21
Kd:
43
EC50:
12
47
1
2D
3D
TSV
ADRB2
Ki:
942
IC50:
687
Kd:
319
EC50:
1370
Other:
1
227
27
2D
3D
TSV
ADRB2R
Ki:
890
IC50:
681
Kd:
240
EC50:
1370
Other:
1
214
22
2D
3D
TSV
ADRB2RL1
Ki:
5792
IC50:
767
Kd:
11
EC50:
1146
528
4
2D
3D
TSV
ADRB3
Ki:
330
IC50:
57
Kd:
69
EC50:
1496
106
5
2D
3D
TSV
ADRBK1
Ki:
1
IC50:
310
Kd:
8
EC50:
59
22
7
2D
3D
TSV
ADRBK2
IC50:
6
1
1
2D
3D
TSV
ADRBRL1
Ki:
5792
IC50:
767
Kd:
11
EC50:
1146
528
4
2D
3D
TSV
Adrenal 4-binding protein
Ki:
6
IC50:
884
Kd:
2
EC50:
245
Other:
3
10
5
2D
3D
TSV
Adrenaline 2
Ki:
143
IC50:
3
36
3
2D
3D
TSV
Adrenaline alpha1
Ki:
50
IC50:
41
20
4
2D
3D
TSV
Adrenaline alpha2
Ki:
33
IC50:
44
13
4
2D
3D
TSV
Adrenergic Alpha
Ki:
1352
IC50:
144
78
9
2D
3D
TSV
adrenergic Alpha1
Ki:
2474
IC50:
410
Kd:
6
EC50:
354
295
31
2D
3D
TSV
Adrenergic alpha1A
Ki:
1947
IC50:
302
Kd:
4
EC50:
336
245
22
2D
3D
TSV
adrenergic Alpha1B
Ki:
365
IC50:
27
Kd:
52
EC50:
19
52
7
2D
3D
TSV
adrenergic Alpha1C
Ki:
1947
IC50:
302
Kd:
4
EC50:
336
245
22
2D
3D
TSV
adrenergic Alpha1D
Ki:
1301
IC50:
154
EC50:
235
129
4
2D
3D
TSV
adrenergic Alpha2
Ki:
552
IC50:
53
Kd:
2
71
8
2D
3D
TSV
Adrenergic alpha2 receptor
Ki:
4
4
1
2D
3D
TSV
adrenergic Alpha2A
Ki:
323
IC50:
56
Kd:
2
52
5
2D
3D
TSV
Adrenergic alpha2B
Ki:
665
IC50:
32
Kd:
8
EC50:
96
114
6
2D
3D
TSV
Adrenergic alpha2C
Ki:
880
IC50:
62
EC50:
183
144
5
2D
3D
TSV
adrenergic Alpha2D
Ki:
127
IC50:
53
Kd:
2
14
0
2D
3D
TSV
adrenergic Beta
Ki:
26
IC50:
6
Kd:
79
7
3
2D
3D
TSV
adrenergic Beta1
Ki:
778
IC50:
684
Kd:
487
EC50:
936
245
8
2D
3D
TSV
adrenergic Beta1,2
Ki:
239
IC50:
21
Kd:
43
EC50:
12
47
1
2D
3D
TSV
adrenergic Beta2
Ki:
67
IC50:
62
Kd:
248
EC50:
135
42
3
2D
3D
TSV
adrenergic Beta3
Ki:
330
IC50:
57
Kd:
69
EC50:
1486
105
4
2D
3D
TSV
Adrenergic receptor
Ki:
4454
IC50:
413
Kd:
329
EC50:
817
325
16
2D
3D
TSV
Adrenergic receptor alpha
Ki:
5933
IC50:
610
Kd:
27
EC50:
931
372
31
2D
3D
TSV
Adrenergic receptor alpha-1
Ki:
1428
IC50:
579
Kd:
1
EC50:
19
165
7
2D
3D
TSV
Adrenergic receptor alpha-2
Ki:
1253
IC50:
258
Kd:
16
EC50:
55
147
10
2D
3D
TSV
Adrenergic receptor beta
Ki:
414
IC50:
197
Kd:
112
EC50:
116
112
10
2D
3D
TSV
Adrenergic Receptors (alpha 2)
Ki:
190
IC50:
56
Kd:
16
EC50:
42
37
4
2D
3D
TSV
Adrenergic, alpha-2B-, receptor [Homo sapiens]
Ki:
665
IC50:
32
Kd:
8
EC50:
96
114
6
2D
3D
TSV
Adrenergic, alpha-2C-, receptor
Ki:
880
IC50:
62
EC50:
183
144
5
2D
3D
TSV
adrenergic, alpha-2C-, receptor [Homo sapiens]
Ki:
880
IC50:
62
EC50:
183
144
5
2D
3D
TSV
Adrenocorticotropic hormone receptor
IC50:
1
1
5
2D
3D
TSV
Adrenocorticotropin receptor
IC50:
1
1
5
2D
3D
TSV
Adrenomedullin receptor AM1, CALCRL/RAMP2
Ki:
1
1
3
2D
3D
TSV
Adrenomedullin receptor AM1; CALCRL/RAMP2
Ki:
520
IC50:
769
Kd:
6
EC50:
14
42
6
2D
3D
TSV
Adrenomedullin receptor, AM2; CALCRL/RAMP3
Ki:
1
1
3
2D
3D
TSV
AdSS 2
IC50:
3
1
5
2D
3D
TSV
ADT20_14595
Ki:
12
IC50:
17
1
3
2D
3D
TSV
ADT21_00085
Ki:
12
IC50:
17
1
3
2D
3D
TSV
ADTB1
Kd:
1
1
7
2D
3D
TSV
Adult folate-binding protein
IC50:
83
Kd:
10
8
7
2D
3D
TSV
Advanced glycosylation end product-specific receptor
Ki:
3
IC50:
35
Kd:
46
5
19
2D
3D
TSV
AF reductase
IC50:
70
1
6
2D
3D
TSV
AF1P
IC50:
1
Kd:
1
2
5
2D
3D
TSV
AF6q21 protein
Kd:
1
1
7
2D
3D
TSV
AF9
Ki:
28
IC50:
27
Kd:
1
1
8
2D
3D
TSV
AFABP
Ki:
116
IC50:
538
Kd:
34
24
5
2D
3D
TSV
AfChiB1
Ki:
2
IC50:
15
Kd:
3
5
4
2D
3D
TSV
AfChiB1(A217G)
Kd:
3
2
0
2D
3D
TSV
AfChiB1(D175A)
Kd:
3
2
0
2D
3D
TSV
AfChiB1(D246A)
Kd:
1
1
0
2D
3D
TSV
AfChiB1(E177A)
Kd:
1
1
0
2D
3D
TSV
AfChiB1(E322A)
Kd:
3
2
0
2D
3D
TSV
AfChiB1(M243A)
Kd:
3
2
0
2D
3D
TSV
AfChiB1(R301K)
Kd:
3
2
0
2D
3D
TSV
AfChiB1(T138A)
Kd:
3
2
0
2D
3D
TSV
AfChiB1(Y245F)
Kd:
2
2
0
2D
3D
TSV
aFGF
IC50:
2
Kd:
116
9
6
2D
3D
TSV
AFL synthase
Ki:
1
IC50:
2
1
1
2D
3D
TSV
Agammaglobulinaemia tyrosine kinase
Ki:
237
IC50:
13961
Kd:
150
EC50:
581
319
4
2D
3D
TSV
Agammaglobulinemia tyrosine kinase
Ki:
237
IC50:
14035
Kd:
150
EC50:
581
319
6
2D
3D
TSV
AGC1
Kd:
12
1
5
2D
3D
TSV
AGER
Ki:
3
IC50:
35
Kd:
45
5
18
2D
3D
TSV
Aggrecan core protein
Kd:
12
1
5
2D
3D
TSV
Aggrecanase-1
Ki:
11
IC50:
478
Other:
2
35
7
2D
3D
TSV
Aggrecanase-2
Ki:
14
IC50:
1321
35
4
2D
3D
TSV
Aging-associated gene 8 protein
Ki:
2470
IC50:
981
Kd:
12
198
12
2D
3D
TSV
Aglucosidase alfa
Ki:
17
IC50:
131
Kd:
2
24
6
2D
3D
TSV
Agmatine iminohydrolase
IC50:
2
1
3
2D
3D
TSV
agonist GABA site
Ki:
200
IC50:
44
Kd:
22
EC50:
57
32
13
2D
3D
TSV
Agp1p
EC50:
23
2
3
2D
3D
TSV
agr
IC50:
15
3
4
2D
3D
TSV
agrA
IC50:
15
3
4
2D
3D
TSV
AGS1
IC50:
63
1
13
2D
3D
TSV
AGTR1
Ki:
124
IC50:
39
Kd:
22
19
4
2D
3D
TSV
Agtr1.2 protein
Ki:
1
1
1
2D
3D
TSV
Agtr1a
IC50:
45
1
1
2D
3D
TSV
AGTR2
Ki:
1
1
1
2D
3D
TSV
AGTRL1
Ki:
103
IC50:
501
EC50:
4770
24
1
2D
3D
TSV
aguA
IC50:
2
1
3
2D
3D
TSV
Ah Receptor
IC50:
2
Kd:
10
EC50:
11
4
6
2D
3D
TSV
AH-related protein
IC50:
4
1
10
2D
3D
TSV
AHCYL1
IC50:
5
1
10
2D
3D
TSV
AHF
Ki:
2
IC50:
33
3
4
2D
3D
TSV
AhR
Ki:
36
IC50:
15
Kd:
11
EC50:
268
24
12
2D
3D
TSV
ahr2
IC50:
5
1
1
2D
3D
TSV
AI-2 kinase
IC50:
4
1
1
2D
3D
TSV
AI115505
IC50:
5
1
4
2D
3D
TSV
AI427544
IC50:
5
1
4
2D
3D
TSV
AIBP80
Ki:
20
IC50:
22
Kd:
22
1
6
2D
3D
TSV
AICAR Tfase
Ki:
45
IC50:
63
Kd:
1
EC50:
17
21
7
2D
3D
TSV
AICAR transformylase
Ki:
45
IC50:
72
Kd:
1
EC50:
17
22
14
2D
3D
TSV
AICD-50
Ki:
516
IC50:
1191
Kd:
31
EC50:
105
129
26
2D
3D
TSV
AICD-57
Ki:
516
IC50:
1191
Kd:
31
EC50:
105
129
26
2D
3D
TSV
AICD-59
Ki:
516
IC50:
1191
Kd:
31
EC50:
105
129
26
2D
3D
TSV
AID(50)
Ki:
516
IC50:
1191
Kd:
31
EC50:
105
129
26
2D
3D
TSV
AID(57)
Ki:
516
IC50:
1191
Kd:
31
EC50:
105
129
26
2D
3D
TSV
AID(59)
Ki:
516
IC50:
1191
Kd:
31
EC50:
105
129
26
2D
3D
TSV
AIG6
Ki:
105
IC50:
72
Kd:
7
8
5
2D
3D