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Found 44
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50518613(CHEMBL4448860)
Affinity DataIC50:  500nMAssay Description:Inhibition of Escherichia coli C-terminal His6-tagged ClpP expressed Escherichia coli SG1146a using Suc-LY-AMC as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50518615(CHEMBL4551942)
Affinity DataIC50:  500nMAssay Description:Inhibition of Escherichia coli C-terminal His6-tagged ClpP expressed Escherichia coli SG1146a using Suc-LY-AMC as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50518612(CHEMBL4444802)
Affinity DataIC50:  600nMAssay Description:Inhibition of Escherichia coli C-terminal His6-tagged ClpP expressed Escherichia coli SG1146a using Suc-LY-AMC as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50518616(CHEMBL4483092)
Affinity DataIC50:  600nMAssay Description:Inhibition of Escherichia coli C-terminal His6-tagged ClpP expressed Escherichia coli SG1146a using Suc-LY-AMC as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527098(CHEMBL4446834)
Affinity DataIC50:  900nMAssay Description:Inhibition of N-terminal His6-sumo-tagged full length Staphylococcus aureus ClpP expressed in Escherichia coli BL2 (DE3) pre-incubated for 10 mins be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527099(CHEMBL4438765)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of N-terminal His6-sumo-tagged full length Staphylococcus aureus ClpP expressed in Escherichia coli BL2 (DE3) pre-incubated for 10 mins be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527100(CHEMBL4457363)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of N-terminal His6-sumo-tagged full length Staphylococcus aureus ClpP expressed in Escherichia coli BL2 (DE3) pre-incubated for 10 mins be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527101(CHEMBL4540126)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of N-terminal His6-sumo-tagged full length Staphylococcus aureus ClpP expressed in Escherichia coli BL2 (DE3) pre-incubated for 10 mins be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527102(CHEMBL4536802)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of N-terminal His6-sumo-tagged full length Staphylococcus aureus ClpP expressed in Escherichia coli BL2 (DE3) pre-incubated for 10 mins be...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50398609(CHEMBL2141296 | IXAZOMIB CITRATE | Ixazomib | MLN2...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of N-terminal His6-sumo-tagged full length Staphylococcus aureus ClpP expressed in Escherichia coli BL2 (DE3) pre-incubated for 10 mins be...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of N-terminal His6-sumo-tagged full length Staphylococcus aureus ClpP expressed in Escherichia coli BL2 (DE3) pre-incubated for 10 mins be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50518619(CHEMBL4575669)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of Escherichia coli C-terminal His6-tagged ClpP expressed Escherichia coli SG1146a using Suc-LY-AMC as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50518624(CHEMBL4472140)
Affinity DataIC50:  1.31E+4nMAssay Description:Inhibition of Escherichia coli C-terminal His6-tagged ClpP expressed Escherichia coli SG1146a using Suc-LY-AMC as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50518623(CHEMBL4446383)
Affinity DataIC50:  1.42E+4nMAssay Description:Inhibition of Escherichia coli C-terminal His6-tagged ClpP expressed Escherichia coli SG1146a using Suc-LY-AMC as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50527103(CHEMBL4449233)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of Escherichia coli ClpPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50518611(CHEMBL4461379)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of Escherichia coli C-terminal His6-tagged ClpP expressed Escherichia coli SG1146a using Suc-LY-AMC as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50518621(CHEMBL4561263)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of Escherichia coli C-terminal His6-tagged ClpP expressed Escherichia coli SG1146a using Suc-LY-AMC as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50518617(CHEMBL3770879)
Affinity DataIC50:  3.98E+4nMAssay Description:Inhibition of Escherichia coli C-terminal His6-tagged ClpP expressed Escherichia coli SG1146a using Suc-LY-AMC as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50518622(CHEMBL4585066)
Affinity DataIC50:  4.81E+4nMAssay Description:Inhibition of Escherichia coli C-terminal His6-tagged ClpP expressed Escherichia coli SG1146a using Suc-LY-AMC as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50518618(CHEMBL4469279)
Affinity DataIC50:  4.95E+4nMAssay Description:Inhibition of Escherichia coli C-terminal His6-tagged ClpP expressed Escherichia coli SG1146a using Suc-LY-AMC as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50518620(CHEMBL4442349)
Affinity DataIC50:  7.13E+4nMAssay Description:Inhibition of Escherichia coli C-terminal His6-tagged ClpP expressed Escherichia coli SG1146a using Suc-LY-AMC as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50518614(CHEMBL4476496)
Affinity DataIC50:  7.97E+4nMAssay Description:Inhibition of Escherichia coli C-terminal His6-tagged ClpP expressed Escherichia coli SG1146a using Suc-LY-AMC as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50518625(CHEMBL4549411)
Affinity DataIC50:  1.01E+5nMAssay Description:Inhibition of Escherichia coli C-terminal His6-tagged ClpP expressed Escherichia coli SG1146a using Suc-LY-AMC as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)
Affinity DataEC50:  2.35E+4nMAssay Description:Inhibition of ClpP in methicillin-resistant Staphylococcus aureus ATCC 33591 assessed as reduction in bacteria-induced hemolysis of sheep erythrocyte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50462621(CHEMBL1813256 | MLN-9708 | US11542283, Compound ML...)
Affinity DataEC50:  1.99E+4nMAssay Description:Binding affinity to N-terminal His6-sumo-tagged full length Staphylococcus aureus ClpP expressed in Escherichia coli BL2 (DE3) assessed as shifting o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527102(CHEMBL4536802)
Affinity DataEC50:  3.30E+3nMAssay Description:Inhibition of ClpP in methicillin-resistant Staphylococcus aureus ATCC 33591 assessed as reduction in bacteria-induced hemolysis of sheep erythrocyte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527099(CHEMBL4438765)
Affinity DataEC50:  9.60E+3nMAssay Description:Inhibition of ClpP in methicillin-resistant Staphylococcus aureus ATCC 33591 assessed as reduction in bacteria-induced hemolysis of sheep erythrocyte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50462621(CHEMBL1813256 | MLN-9708 | US11542283, Compound ML...)
Affinity DataKd:  7.30E+3nMAssay Description:Binding affinity to N-terminal His6-sumo-tagged full length Staphylococcus aureus ClpP expressed in Escherichia coli BL2 (DE3) by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527100(CHEMBL4457363)
Affinity DataEC50:  1.48E+4nMAssay Description:Inhibition of ClpP in methicillin-resistant Staphylococcus aureus ATCC 33591 assessed as reduction in bacteria-induced hemolysis of sheep erythrocyte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527101(CHEMBL4540126)
Affinity DataEC50:  2.60E+3nMAssay Description:Inhibition of ClpP in methicillin-resistant Staphylococcus aureus ATCC 33591 assessed as reduction in bacteria-induced hemolysis of sheep erythrocyte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50398609(CHEMBL2141296 | IXAZOMIB CITRATE | Ixazomib | MLN2...)
Affinity DataEC50:  3.60E+3nMAssay Description:Inhibition of ClpP in methicillin-resistant Staphylococcus aureus ATCC 33591 assessed as reduction in bacteria-induced hemolysis of sheep erythrocyte...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527098(CHEMBL4446834)
Affinity DataEC50:  1.27E+3nMAssay Description:Binding affinity to N-terminal His6-sumo-tagged full length Staphylococcus aureus ClpP expressed in Escherichia coli BL2 (DE3) assessed as shifting o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527098(CHEMBL4446834)
Affinity DataEC50:  1.40E+3nMAssay Description:Inhibition of ClpP in methicillin-resistant Staphylococcus aureus ATCC 33591 assessed as reduction in bacteria-induced hemolysis of sheep erythrocyte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50535810(CHEMBL4593796)
Affinity DataEC50:  2.54E+4nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using Abz-DFAPKMALVPYNO2 as substrate assessed as degradation of substrate peptide preincubated for 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50535811(CHEMBL4549588)
Affinity DataEC50:  1.20E+3nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using FITC-beta casein as substrate assessed as degradation of substrate peptide preincubated for 15 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50535811(CHEMBL4549588)
Affinity DataEC50:  100nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using Abz-DFAPKMALVPYNO2 as substrate assessed as degradation of substrate peptide preincubated for 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50535809(Sclerotiamide)
Affinity DataEC50:  8.75E+4nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using FITC-beta casein as substrate assessed as degradation of substrate peptide preincubated for 15 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50535810(CHEMBL4593796)
Affinity DataEC50:  2.22E+4nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using FITC-beta casein as substrate assessed as degradation of substrate peptide preincubated for 15 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50535809(Sclerotiamide)
Affinity DataEC50:  3.96E+4nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using Abz-DFAPKMALVPYNO2 as substrate assessed as degradation of substrate peptide preincubated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50360281(CHEMBL1933116)
Affinity DataEC50:  5.40E+3nMAssay Description:Inhibition of recombinant Staphylococcus aureus NCTC 8325 peptidase activity of clpP expressed in Escherichia coli BL21 after 10 mins using SLY-AMC a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50360280(CHEMBL1933114)
Affinity DataEC50:  4.50E+3nMAssay Description:Inhibition of recombinant Staphylococcus aureus NCTC 8325 peptidase activity of clpP expressed in Escherichia coli BL21 after 10 mins using SLY-AMC a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Staphylococcus aureus (strain NCTC 8325))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50360279(CHEMBL1933113)
Affinity DataEC50:  3.40E+3nMAssay Description:Inhibition of recombinant Staphylococcus aureus NCTC 8325 peptidase activity of clpP expressed in Escherichia coli BL21 after 10 mins using SLY-AMC a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50028480(CHEMBL3342324)
Affinity DataKd:  300nMAssay Description:Activation of Escherichia coli ClpP by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50028481(CHEMBL3342325)
Affinity DataKd:  700nMAssay Description:Activation of Escherichia coli ClpP by ITC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed