Target Names are taken from UniProtKB. To view the associated UniProt page, click on the UniProt ID. When we have data for a given Target in multiple species or for mutants of a given Target, we provide a header row (upper case, bold font) with all of the data followed by a separate for each species or variant of the Target.
Target Name
Organism
Affinity Links
Articles
UniProts
Files
Human
Human
Human
Oryctolagus cuniculus (Rabbit)
IC50: 3
Human
Mus musculus (mouse)
IC50: 3
Mus musculus (mouse)
IC50: 18
Human
IC50: 229
Mus musculus (mouse)
Ki: 398
Human
Human
Human
Human
Marthasterias glacialis (starfish)
Human
IC50: 1
Cyclin-dependent kinase 1/G2/mitotic-specific cyclin-B1/G2/mitotic-specific cyclin-B2/G2/mitotic-specific cyclin-B3 O95067 P06493 P14635 Q8WWL7
Human
Cyclin-dependent kinase 1/G2/mitotic-specific cyclin-B1/G2/mitotic-specific cyclin-B2/G2/mitotic-specific cyclin-B3/cAMP-dependent protein kinase O95067 P06493 P14635 Q8WWL7 Q95J97
Human
IC50: 1
Human
Human
Human
Human immunodeficiency virus type 1 group M subtype B (isolate MN) (HIV-1)
IC50: 10
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 6
Human immunodeficiency virus type 1
Ki: 1
Dimer of Gag-Pol polyprotein [489-587,K509R,V521I,L522F,M525I,I543V,L552P,A560V,V571A,I573V,L579M] P04585
Human immunodeficiency virus type 1
Ki: 4
Human immunodeficiency virus type 1
Ki: 4
Human immunodeficiency virus type 1
Ki: 4
Human immunodeficiency virus type 1
Ki: 4
Dimer of Gag-Pol polyprotein [489-587,K509R,V521I,L522F,M525I,M535I,I543V,L552P,A560V,V571A,I573V,L579M] P04585
Human immunodeficiency virus type 1
Ki: 4
Dimer of Gag-Pol polyprotein [489-587,K509R,V521I,L522F,M525I,M535I,L552P,A560V,V571A,I573V,L579M] P04585
Human immunodeficiency virus type 1
Ki: 4
Human immunodeficiency virus type 1
Ki: 4
Dimer of Gag-Pol polyprotein [489-587,L499I,L508Q,K509R,E524D,M525I,S526N,M535I,I539V,I543V,I551V,L552P,A560V,V571A,L579M] P04585
Human immunodeficiency virus type 1
Ki: 6
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 6
Dimer of Gag-Pol polyprotein [489-587,Q496K,L499I,M525I,N526D,M535I,R546K,L552P,A560V,G562S,I573V,L579M,I582L] P12497
Human immunodeficiency virus type 1
IC50: 27
Dimer of Gag-Pol polyprotein [489-587,Q496K,L499I,M535I,I543V,Q547E,L552P,I553V,V566I,V571F,I573V,L579M,I582L] P12497
Human immunodeficiency virus type 1
IC50: 15
Dimer of Gag-Pol polyprotein [489-587,Q496K,L499I,N526S,R530K,M535I,I543V,I551V,L552P,A560V,V566I,V571A,L579M,I582L] P12497
Human immunodeficiency virus type 1
IC50: 11
Human immunodeficiency virus type 1
IC50: 73
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 62
Human immunodeficiency virus type 1
Ki: 19
Human immunodeficiency virus type 1
Ki: 19
Human immunodeficiency virus type 1
Ki: 19
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 2
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 2
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 2
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 2
Human immunodeficiency virus type 1
Ki: 2
Human immunodeficiency virus type 1
Ki: 2
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 8
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 2
Human immunodeficiency virus type 1
IC50: 3
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
Human immunodeficiency virus type 1 group M subtype B (isolate NY5) (HIV-1)
Human immunodeficiency virus type 1 (HIV-1)
Human immunodeficiency virus type 1 group M subtype B (isolate ARV2/SF2) (HIV-1)
Ki: 20
Human immunodeficiency virus
Ki: 10
Human immunodeficiency virus
Ki: 10
Human immunodeficiency virus
Ki: 9
Gag-Pol polyprotein [484-582,I497V,V499I,E519D,R541K,D544E,Q553K,A555V,G557S,I568V,L574M,L573M] Q9QBY3
Human immunodeficiency virus
Ki: 10
Gag-Pol polyprotein [484-582,Q491K,I494L,I497V,V499I,E519D,I534V,R541K,D544E,Q553K,A555V,L573M] Q9QBY3
Human immunodeficiency virus
Ki: 11
Human immunodeficiency virus
Ki: 11
Gag-Pol polyprotein [484-582,Q491K,I497V,V499I,E519D,G532V,I538V,R541K,D544E,L547P,Q553K,V566A,L573M] Q9QBY3
Human immunodeficiency virus
Ki: 11
Gag-Pol polyprotein [484-582,Q491K,I497V,V499I,E519D,R541K,D544E,L547P,Q553K,A555V,G557S,I568V,L573M,L574M] Q9QBY3
Human immunodeficiency virus
Ki: 11
Human immunodeficiency virus
Human immunodeficiency virus type 1
EC50: 83
Human immunodeficiency virus type 1
Gag-Pol polyprotein [489-892,N526H,R530K,V566I,I582L,V648I,Q690K,I723V,C750S,T788A,Q795E,T874A,V881I,P882Q] P12497
Human immunodeficiency virus
EC50: 6
Human immunodeficiency virus type 1
IC50: 84
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
IC50: 42
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
Human immunodeficiency virus type 1
IC50: 1143
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
IC50: 181
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
IC50: 2
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
IC50: 2
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
IC50: 2
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
IC50: 2
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
IC50: 2
Human immunodeficiency virus type 1
IC50: 9
Human immunodeficiency virus type 1
IC50: 11
Human immunodeficiency virus type 1
IC50: 10
Human immunodeficiency virus type 1
IC50: 10
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
IC50: 9
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
IC50: 18
Gag-Pol polyprotein [600-1028,D666N,K669R,T814F,K818Q,C879S]/[600-1151,D666N,K669R,T814F,K818Q,C879S] P03366
Human immunodeficiency virus type 1
IC50: 1
Human immunodeficiency virus type 1
IC50: 1
Human immunodeficiency virus type 1
IC50: 1
Human immunodeficiency virus type 1
IC50: 1
Human immunodeficiency virus type 1
IC50: 1
Human immunodeficiency virus type 1
IC50: 43
Gag-Pol polyprotein [600-1159,Y780C]/Imidazoleglycerol-phosphate dehydratase [600-1029,Y780C] P03366 P06633
Human immunodeficiency virus type 1
IC50: 3
Human immunodeficiency virus type 2
IC50: 5
Human immunodeficiency virus type 1 group M subtype B (isolate NY5) (HIV-1)
EC50: 79
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
IC50: 2
Rous sarcoma virus (strain Prague C) (RSV-PrC)
Rattus norvegicus (rat)
Human
Human
Rattus norvegicus (Rat)
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-200],P14867[176-456] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,A118C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,D95C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,F116C] P14867 P18507 P47870
Human
Other: 1
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,L179C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,M169C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R171C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R183C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R224C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R233C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T120C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T165C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T181C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-3 [26-473]/gamma-2 [40-467] P14867 P18507 P28472
Human
Ki: 8
Gamma-aminobutyric acid receptor subunit alpha-1 [A160C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [D97C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Other: 1
Gamma-aminobutyric acid receptor subunit alpha-1 [F99C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [G157C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [G200C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [S204C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [S205C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [T162C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [T206C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [V202C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [V211C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [Y209C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Other: 1
Human
Human
Rattus norvegicus (Rat)
Rattus norvegicus (Rat)
EC50: 1
Rattus norvegicus (Rat)
EC50: 2
Human
Rattus norvegicus (Rat)
Mus musculus
Human
Human
Rattus norvegicus (Rat)
Gamma-aminobutyric acid receptor subunit alpha-2 [29-451]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47869 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-2 [29-451]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P47869
Human
Ki: 8
Rattus norvegicus (Rat)
Ki: 25
Human
Rattus norvegicus (Rat)
Gamma-aminobutyric acid receptor subunit alpha-3 [29-492]/beta-2 [26-512]/gamma-2 [40-467] P18507 P34903 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-3 [29-492]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P34903
Human
Ki: 7
Rattus norvegicus (Rat)
Ki: 26
Human
Human
Human
Rattus norvegicus (Rat)
Gamma-aminobutyric acid receptor subunit alpha-4 [36-554]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47870 P48169
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-4 [36-554]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P48169
Human
Ki: 4
Human
Human
EC50: 1
Human
EC50: 18
Rattus norvegicus (Rat)
Human
EC50: 12
Rattus norvegicus (Rat)
Human
Human
Gamma-aminobutyric acid receptor subunit alpha-5 [32-462]/beta-2 [26-512]/gamma-2 [40-467] P18507 P31644 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-5 [32-462]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P31644
Human
Ki: 8
Human
Gamma-aminobutyric acid receptor subunit alpha-6 [20-453]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47870 Q16445
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-6 [20-453]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 Q16445
Human
Ki: 7
Rattus norvegicus (Rat)
IC50: 2
Rattus norvegicus (Rat)
Human
Ki: 20
Rattus norvegicus (Rat)
RAT
Rattus norvegicus (Rat)
IC50: 10
Human
Human
Human
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-200],P14867[176-456] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,A118C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,D95C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,F116C] P14867 P18507 P47870
Human
Other: 1
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,L179C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,M169C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R171C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R183C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R224C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R233C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T120C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T165C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T181C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [A160C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [D97C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Other: 1
Gamma-aminobutyric acid receptor subunit alpha-1 [F99C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [G157C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [G200C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [S204C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [S205C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [T162C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [T206C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [V202C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [V211C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [Y209C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Other: 1
Human
Human
Rattus norvegicus (Rat)
Gamma-aminobutyric acid receptor subunit alpha-2 [29-451]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47869 P47870
Human
Ki: 3
Rattus norvegicus (Rat)
Ki: 25
Human
Gamma-aminobutyric acid receptor subunit alpha-3 [29-492]/beta-2 [26-512]/gamma-2 [40-467] P18507 P34903 P47870
Human
Ki: 3
Rattus norvegicus (Rat)
Ki: 26
Human
Gamma-aminobutyric acid receptor subunit alpha-4 [36-554]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47870 P48169
Human
Ki: 3
Human
EC50: 1
Human
EC50: 18
Gamma-aminobutyric acid receptor subunit alpha-5 [32-462]/beta-2 [26-512]/gamma-2 [40-467] P18507 P31644 P47870
Human
Ki: 3
Human
Gamma-aminobutyric acid receptor subunit alpha-6 [20-453]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47870 Q16445
Human
Ki: 3
Rattus norvegicus (Rat)
IC50: 2
Rattus norvegicus (Rat)
Human
Ki: 20
Rattus norvegicus (Rat)
Human
Human
Human
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-3 [26-473]/gamma-2 [40-467] P14867 P18507 P28472
Human
Ki: 8
Rattus norvegicus (Rat)
EC50: 1
Rattus norvegicus (Rat)
EC50: 2
Human
Rattus norvegicus (Rat)
Mus musculus
Gamma-aminobutyric acid receptor subunit alpha-2 [29-451]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P47869
Human
Ki: 8
Rattus norvegicus (Rat)
Gamma-aminobutyric acid receptor subunit alpha-3 [29-492]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P34903
Human
Ki: 7
Human
Rattus norvegicus (Rat)
Gamma-aminobutyric acid receptor subunit alpha-4 [36-554]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P48169
Human
Ki: 4
Rattus norvegicus (Rat)
Human
EC50: 12
Rattus norvegicus (Rat)
Rattus norvegicus (Rat)
IC50: 1
Gamma-aminobutyric acid receptor subunit alpha-5 [32-462]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P31644
Human
Ki: 8
Rattus norvegicus (Rat)
Gamma-aminobutyric acid receptor subunit alpha-6 [20-453]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 Q16445
Human
Ki: 7
RAT
Rattus norvegicus (Rat)
IC50: 10
Human
Rattus norvegicus (Rat)
Human
Rattus norvegicus (Rat)
EC50: 2
Rattus norvegicus (Rat)
IC50: 17
Human
Human
EC50: 1
Human
EC50: 12
Rattus norvegicus (Rat)
Rattus norvegicus (Rat)
Human
Human
Human
Human
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-200],P14867[176-456] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,A118C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,D95C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,F116C] P14867 P18507 P47870
Human
Other: 1
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,L179C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,M169C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R171C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R183C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R224C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R233C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T120C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T165C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T181C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-3 [26-473]/gamma-2 [40-467] P14867 P18507 P28472
Human
Ki: 8
Gamma-aminobutyric acid receptor subunit alpha-1 [A160C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [D97C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Other: 1
Gamma-aminobutyric acid receptor subunit alpha-1 [F99C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [G157C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [G200C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [S204C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [S205C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [T162C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [T206C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [V202C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [V211C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [Y209C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Other: 1
Human
Rattus norvegicus (Rat)
Human
Rattus norvegicus (Rat)
Mus musculus
Gamma-aminobutyric acid receptor subunit alpha-2 [29-451]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47869 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-2 [29-451]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P47869
Human
Ki: 8
Rattus norvegicus (Rat)
Ki: 25
Human
Rattus norvegicus (Rat)
Gamma-aminobutyric acid receptor subunit alpha-3 [29-492]/beta-2 [26-512]/gamma-2 [40-467] P18507 P34903 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-3 [29-492]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P34903
Human
Ki: 7
Rattus norvegicus (Rat)
Ki: 26
Human
Human
Rattus norvegicus (Rat)
Gamma-aminobutyric acid receptor subunit alpha-4 [36-554]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47870 P48169
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-4 [36-554]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P48169
Human
Ki: 4
Human
EC50: 18
Rattus norvegicus (Rat)
IC50: 1
Gamma-aminobutyric acid receptor subunit alpha-5 [32-462]/beta-2 [26-512]/gamma-2 [40-467] P18507 P31644 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-5 [32-462]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P31644
Human
Ki: 8
Human
Rattus norvegicus (Rat)
Gamma-aminobutyric acid receptor subunit alpha-6 [20-453]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47870 Q16445
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-6 [20-453]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 Q16445
Human
Ki: 7
Human
Ki: 20
Rattus norvegicus (Rat)
Human
Rattus norvegicus (Rat)
Rattus norvegicus (Rat)
Human
Rattus norvegicus (rat)
Human
Rattus norvegicus (Rat)
Human
Human
Gamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2 P49768 P49810 Q8WW43 Q92542 Q96BI3 Q9NZ42
Human
IC50: 558
Human
RAT
IC50: 124
MOUSE
Ki: 22
Human
GENOME POLYPROTEIN A0A024B7W1 A0A0K1CY61 A0A143MHK7 A0A1D8D5K2 A3EZI9 A3EZJ3 B0B3F0 C1KIQ2 D2K2A8 G1FEK8 I1U3K2 K7XGM7 K7XJL6 O39927 O39929 O92972 P03300 P03303 P03313 P06935 P12823 P12916 P14340 P17763 P19711 P26660 P26661 P26662 P26663 P26664 P27914 P27915 P27958 P29846 P29990 P33478 P69035 Q04045 Q0ZMF1 Q32ZE1 Q3ZDS5 Q4U254 Q58HT7 Q66478 Q69422 Q6YMS4 Q7T664 Q80J95 Q81258 Q81495 Q82122 Q83883 Q91H74 Q91RS4 Q96662 Q99IB8 Q9WMX2 V5TFZ2
Bovine viral diarrhea virus (isolate NADL) (BVDV) (Mucosal disease virus)
EC50: 20
Hepatitis C virus genotype 3a (isolate k3a) (HCV)
Hepatitis C virus (HCV genotype 1a, isolate H)
Hepatitis C virus genotype 1b (isolate Taiwan)
Hepatitis C virus genotype 2b (isolate HC-J8) (HCV)
Hepatitis C virus genotype 1b (isolate BK) (HCV)
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Bovine viral diarrhea virus (strain CP7) (BVDV) (Mucosal diseasevirus)
IC50: 1
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
IC50: 4
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
IC50: 1
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
IC50: 4
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
IC50: 7
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
IC50: 4
Hepatitis C virus genotype 1a (isolate 1) (HCV)
IC50: 66
Hepatitis C virus genotype 1a (strain H77) (HCV)
Hepatitis C virus genotype 1b (isolate BK) (HCV)
IC50: 67
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 12
Hepatitis C virus genotype 1b (strain HC-J4) (HCV)
EC50: 27
Hepatitis C virus genotype 1a (isolate H) (HCV)
EC50: 17
Hepatitis C virus genotype 1b (strain J4L2S) (HCV)
EC50: 67
Dengue virus 2 (strain TSV01)
Dengue virus 1(Hawaii)
IC50: 10
Dengue virus 3 (strain S221/03)
IC50: 10
West Nile virus (WNV)
West Nile virus (WNV)
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 42
Hepatitis C virus genotype 1a (isolate H77) (HCV)
EC50: 17
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 30
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 22
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 22
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 18
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 22
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 22
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 22
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 42
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Hepatitis C virus genotype 1b (isolate BK) (HCV)
IC50: 2
Hepatitis C virus genotype 1b (isolate BK) (HCV)
IC50: 2
Hepatitis C virus genotype 1b (isolate BK) (HCV)
IC50: 2
Hepatitis C virus genotype 1b (isolate BK) (HCV)
IC50: 2
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Hepatitis C virus genotype 1b (strain HC-J4) (HCV)
Hepatitis C virus genotype 1b (strain HC-J4) (HCV)
Hepatitis C virus genotype 1b (strain HC-J4) (HCV)
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Hepatitis C virus genotype 1b (strain HC-J4) (HCV)
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
IC50: 3
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Hepatitis C virus genotype 1b (isolate BK) (HCV)
Hepatitis C virus genotype 1b (strain HC-J4) (HCV)
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 36
Hepatitis C virus genotype 1b (isolate Japanese) (HCV)
IC50: 5
Hepatitis C virus
Saccharomyces cerevisiae (Yeast)
Saccharomyces cerevisiae (Yeast)
Geranylgeranyl transferase type-1 subunit beta [A2V]/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha P49354 P53609
Human
Geranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha P29702 Q5EAD5
Bos taurus (bovine)
IC50: 183
Geranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha P49354 P53609
Human
Rattus norvegicus
IC50: 8
Human
Human
Mus musculus (Mouse)
EC50: 6
Rattus norvegicus (Rat)
Rattus norvegicus (Rat)
Human
Rattus norvegicus (Rat)
Rattus norvegicus (Rat)
Rattus norvegicus (Rat)
Human
IC50: 33
Rattus norvegicus (Rat)
Rattus norvegicus (Rat)
Human
Human
Human
Human
Rattus norvegicus (Rat)
Human
Rattus norvegicus (Rat)
Rattus norvegicus (Rat)
Rattus norvegicus (Rat)
Rattus norvegicus (Rat)
Human
Candida albicans
GLUTATHIONE S-TRANSFERASE P O60341 O60674 O75116 O75460 P09211 P10415 P11362 P22607 P23458 P24864 P24941 P33981 P42330 P43405 Q13464 Q9BUB5 Q9UDY8
Human
Human
IC50: 81
Human
IC50: 41
Human
IC50: 25
Human
IC50: 132
Human
IC50: 96
Glutathione S-transferase P/Isoform 2 of Lysine-specific histone demethylase 1A (2) [158-876] O60341 P09211
Human
Glutathione S-transferase P/Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) [T344D] P09211 Q9BUB5
Human
IC50: 110
Human
Human
IC50: 125
Glutathione S-transferase P/Mucosa-associated lymphoid tissue lymphoma translocation protein 1 P09211 Q9UDY8
Human
IC50: 48
Human
IC50: 11
Human
IC50: 10
Human
IC50: 182
Oryctolagus cuniculus (rabbit)
Human
Alpha-1,2-mannosidase/Alpha-1,2-mannosidase family protein/Alpha-1,2-mannosidase, putative/Glycoside hydrolase family 92/Putative alpha-1,2-mannosidase Q8A0C8 Q8A0C9 Q8A0E8 Q8A0M7 Q8A0N0 Q8A0N1 Q8A0Q6 Q8A0Q8 Q8A0Q9 Q8A113 Q8A182 Q8A193 Q8A1X8 Q8A1Y1 Q8A325 Q8A3K6 Q8A4H0 Q8A5N9 Q8A5X5 Q8A5Y1 Q8A6K3 Q8A6V7 Q8A8Y5
Bacteroides thetaiotaomicron
Ki: 1
Candida albicans (Yeast)
Macaca fascicularis (Crab-eating macaque) (Cynomolgus monkey)
IC50: 2
Human
Human
IC50: 150
Human
IC50: 7
Human
IC50: 1
Human
Human
IC50: 244
Guanine nucleotide-binding protein subunit alpha-15 [Y147C]/Metabotropic glutamate receptor 2 P30679 Q14416
Human
IC50: 315
Curated by BindingDB
Curated by ChEMBL