Target Names are taken from UniProtKB. To view the associated UniProt page, click on the UniProt ID. When we have data for a given Target in multiple species or for mutants of a given Target, we provide a header row (upper case, bold font) with all of the data followed by a separate for each species or variant of the Target.

Target Name  
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Target Name
Organism
Affinity Links
Articles
UniProts
Files
Human cytomegalovirus
EC50: 12
Rattus norvegicus
EC50: 8
Rattus norvegicus
EC50: 29
Human
Ki: 59 IC50: 487 Kd: 4 EC50: 563
Human
IC50: 548 Kd: 3 EC50: 341
Human
Ki: 5 IC50: 428 EC50: 78
Mus musculus
IC50: 8 EC50: 7
Human
Ki: 72 IC50: 201 Kd: 1 EC50: 265
Human cytomegalovirus (strain AD169) (HHV-5) (Human herpesvirus 5)
IC50: 33 EC50: 32
Drosophila melanogaster
IC50: 2 Kd: 6
Marthasterias glacialis (starfish)
Ki: 2 IC50: 413 Other: 13
Asterina pectinifera
IC50: 11
Human immunodeficiency virus type 1 group M subtype B (isolate MN) (HIV-1)
IC50: 10
Avian erythroblastosis virus (strain ES4)
IC50: 15
Human immunodeficiency virus 1
Kd: 2
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 6
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
IC50: 73
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 613 IC50: 915 Other: 20
Human immunodeficiency virus type 1
Ki: 131 IC50: 30
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 62
Human immunodeficiency virus type 1
Ki: 10 Other: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 226 IC50: 43 EC50: 38
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 8
Human immunodeficiency virus type 1
Ki: 367 IC50: 98
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 2
Ki: 16 IC50: 7
Human immunodeficiency virus type 1
IC50: 3
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
IC50: 1332 Kd: 8 EC50: 250
Human immunodeficiency virus type 1 group M subtype B (isolate NY5) (HIV-1)
IC50: 28 Kd: 4 EC50: 79
Human immunodeficiency virus type 1 (HIV-1)
Ki: 5 IC50: 84 EC50: 12
Human immunodeficiency virus type 1 group M subtype B (isolate ARV2/SF2) (HIV-1)
Ki: 20
Human immunodeficiency virus type 1 (HIV-1)
IC50: 3
Woolly monkey sarcoma virus
Ki: 13 IC50: 22
Human immunodeficiency virus type 1
IC50: 132
Human immunodeficiency virus
Ki: 11 IC50: 52
Human immunodeficiency virus type 1
EC50: 83
Human immunodeficiency virus type 1
Ki: 1961 IC50: 2162 Kd: 84 EC50: 39 Koff: 39 Kon: 39
Human immunodeficiency virus
EC50: 6
Human immunodeficiency virus type 1
IC50: 84
Human immunodeficiency virus type 1
IC50: 32 EC50: 13
Human immunodeficiency virus type 1
Ki: 5 IC50: 5
Human immunodeficiency virus type 1
IC50: 42
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
Ki: 5 IC50: 42 EC50: 12
Human immunodeficiency virus type 1
IC50: 1143
Human immunodeficiency virus type 1
Ki: 4 IC50: 57
Human immunodeficiency virus type 1
IC50: 181
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
IC50: 2
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
IC50: 2
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
IC50: 2
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
IC50: 2
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
IC50: 2
Human immunodeficiency virus type 1
IC50: 9
Human immunodeficiency virus type 1
IC50: 10
Human immunodeficiency virus type 1
IC50: 10
Human immunodeficiency virus type 1
IC50: 296 Other: 5
Human immunodeficiency virus type 1
IC50: 9
Human immunodeficiency virus type 1
IC50: 155 Other: 1
Human immunodeficiency virus type 1
IC50: 56 Other: 3
Human immunodeficiency virus type 1
IC50: 18
Human immunodeficiency virus type 1
IC50: 1
Human immunodeficiency virus type 1
IC50: 1
Human immunodeficiency virus type 1
IC50: 43
Human immunodeficiency virus 1 (Virus)
IC50: 4
Human immunodeficiency virus type 1 group M subtype B (isolate NY5) (HIV-1)
EC50: 79
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
IC50: 2
Human immunodeficiency virus
EC50: 6
Human immunodeficiency virus
EC50: 6
Human immunodeficiency virus type 1
ITC: 13
Human immunodeficiency virus type 1
Ki: 4 ITC: 4
Human immunodeficiency virus type 1
ITC: 5
Human immunodeficiency virus type 1
Ki: 4 ITC: 4
Human immunodeficiency virus type 1
Ki: 4 ITC: 4
Human immunodeficiency virus type 1
Ki: 4 ITC: 4
Human immunodeficiency virus
EC50: 6
Human immunodeficiency virus
EC50: 6
Human immunodeficiency virus type 1
ITC: 4
Rous sarcoma virus (strain Prague C) (RSV-PrC)
IC50: 18 EC50: 8
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
IC50: 2 EC50: 223
Human T-cell leukemia virus 1 (strain Japan ATK-1 subtype A) (HTLV-1)
Ki: 4 IC50: 27
Mus musculus
Ki: 2
Mycobacterium tuberculosis
IC50: 1
Human
IC50: 242
Mus musculus
IC50: 8
Human
Ki: 67 IC50: 25 Kd: 7
Human
Ki: 54 IC50: 134 Kd: 7 EC50: 22
Gallus gallus
IC50: 18
Human
IC50: 52 Kd: 214
Rattus norvegicus
Kd: 4
Human
Kd: 22
Human
IC50: 460 Kd: 639 EC50: 5
Mus musculus
IC50: 57 Kd: 17
Human
Kd: 69
Human
Kd: 84
Mus musculus
Kd: 4
Human
Kd: 159
Human
IC50: 11 Kd: 132
Rattus norvegicus (Rat)
Ki: 282 IC50: 106 EC50: 4
Rattus norvegicus (Rat)
Ki: 19 IC50: 18 EC50: 1
Human
IC50: 2
Cryptosporidium parvum
IC50: 103
Emericella nidulans (strain FGSC A4 / ATCC 38163 / CBS 112.46 / NRRL194 / M139) (Aspergillus nidulans)
Ki: 1
Human
Ki: 21 IC50: 21
Rattus norvegicus
Ki: 3
Human
Kd: 13
Rattus norvegicus (Rat)
IC50: 19
Sus scrofa (Pig)
IC50: 20
Mus musculus
IC50: 3
Saccharomyces cerevisiae S288c
EC50: 23
Saccharomyces cerevisiae
Ki: 4
Murine norovirus 1
EC50: 143
Hepatitis C virus genotype 2a (isolate HC-J6) (HCV)
EC50: 76
Bovine viral diarrhea virus (isolate NADL) (BVDV) (Mucosal disease virus)
EC50: 20
Hepatitis C virus genotype 3a (isolate k3a) (HCV)
Ki: 89 IC50: 140 EC50: 24
Hu/NV/NV/1968/US
EC50: 2
Hepatitis C virus (HCV genotype 1a, isolate H)
Ki: 300 IC50: 930 EC50: 305
HRV-1B
EC50: 7
DENV-1
IC50: 4 EC50: 6
Hepatitis C virus genotype 1b (isolate Taiwan)
IC50: 6 Other: 6
Hepatitis C virus genotype 2b (isolate HC-J8) (HCV)
IC50: 19 EC50: 1
Hepatitis C virus genotype 2a
IC50: 1 EC50: 4
Hepatitis C virus genotype 4a (isolate ED43) (HCV)
IC50: 1
Hepatitis C virus genotype 6a (isolate EUHK2) (HCV)
IC50: 1
Hepatitis C virus
IC50: 146
Hepatitis C Virus
Ki: 22 IC50: 100 Koff: 1 Kon: 1
Coxsackievirus B3 (strain Nancy)
Ki: 9 IC50: 103
Hepatitis C virus
Ki: 241 IC50: 272 Kd: 41 EC50: 43
Hepatitis C virus
Ki: 11
Hepatitis C virus genotype 1b (isolate BK) (HCV)
IC50: 225 EC50: 114
Hepatitis C virus (HCV)
IC50: 189 EC50: 32
Hepatitis C virus genotype 1b (strain HC-J4) (HCV)
IC50: 55
Hepatitis C virus genotype 3a (isolate NZL1) (HCV)
IC50: 45
Hepatitis C virus
Ki: 15 IC50: 197
Hepatitis C virus
Ki: 10
Hepatitis C virus (HCV)
IC50: 82 EC50: 428
Dengue virus 2 (Virus)
IC50: 20
Hepatitis C Virus (Virus)
Ki: 89 IC50: 400 EC50: 370
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Ki: 19 IC50: 8
Hepacivirus C
Ki: 63
Zika virus
IC50: 20
Zika virus
IC50: 10 Kd: 2 EC50: 41
Human rhinovirus B
Ki: 167 IC50: 290 EC50: 144
Poliovirus type 1 (strain Mahoney)
IC50: 19 Kd: 1
Bovine viral diarrhea virus (strain CP7) (BVDV) (Mucosal diseasevirus)
IC50: 1
Hepatitis GB virus B
IC50: 121
Dengue virus 2
Ki: 112 IC50: 222 EC50: 137
West Nile virus
Ki: 14 IC50: 271 Kd: 2
Human rhinovirus 16
IC50: 9
Hepatitis C virus
Ki: 36 IC50: 11
Dengue virus 2
Ki: 9 IC50: 61 Kd: 3
Norovirus Hu/GII.4-2002/WeertE022/2002/NL
IC50: 13
Norovirus Hu/GI/10360/2010/VNM
IC50: 13
Dengue virus
Ki: 5 IC50: 71 Kd: 2 EC50: 2
Human rhinovirus 14
IC50: 16
Human enterovirus 71 (strain BrCr) (Ev 71)
EC50: 22
Human rhinovirus 1A
EC50: 56
Enterovirus A71
Ki: 26
Hepacivirus C
Ki: 7 IC50: 7
Dengue virus type 2
IC50: 78
Hepatitis C virus
Ki: 2 Koff: 2 Kon: 2
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
IC50: 4
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
IC50: 1
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
IC50: 4
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
IC50: 7
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
IC50: 4
Hepatitis C virus genotype 1a (isolate 1) (HCV)
IC50: 66
Hepatitis C virus (HCV)
Ki: 1 IC50: 1
Hepatitis C virus genotype 1a (strain H77) (HCV)
Ki: 12 IC50: 67 EC50: 62
Hepatitis C virus genotype 1b (isolate BK) (HCV)
IC50: 67
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 12
Hepatitis C virus genotype 1b (strain HC-J4) (HCV)
EC50: 27
Hepatitis C virus genotype 1a (isolate H) (HCV)
EC50: 17
Hepatitis C virus genotype 1b (strain J4L2S) (HCV)
EC50: 67
Dengue virus 2 (strain TSV01)
Ki: 5 IC50: 10 Kd: 7
Dengue virus 3 (strain S221/03)
IC50: 10
West Nile virus (WNV)
Ki: 26 IC50: 29 Kd: 5
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 42
Hepatitis C virus genotype 1a (isolate H77) (HCV)
EC50: 17
Hepatitis C virus
IC50: 4 Kd: 4
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 30
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 22
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 22
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 18
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 22
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 22
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 22
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 42
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
IC50: 28 EC50: 36
Hepatitis C virus genotype 1a (HCV)
EC50: 36
Hepatitis C virus genotype 1b (isolate BK) (HCV)
IC50: 2
Hepatitis C virus genotype 1b (isolate BK) (HCV)
IC50: 2
Hepatitis C virus genotype 1b (isolate BK) (HCV)
IC50: 2
Hepatitis C virus genotype 1b (isolate BK) (HCV)
IC50: 2
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Kd: 1 Koff: 1 Kon: 1
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Kd: 1 Koff: 1 Kon: 1
Hepatitis C virus genotype 1b (strain HC-J4) (HCV)
Kd: 1 Koff: 1 Kon: 1
Hepatitis C virus genotype 1b (strain HC-J4) (HCV)
Kd: 1 Koff: 1 Kon: 1
Hepatitis C virus genotype 1b (strain HC-J4) (HCV)
Kd: 1 Koff: 1 Kon: 1
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Kd: 1 Koff: 1 Kon: 1
Hepatitis C virus genotype 1b (strain HC-J4) (HCV)
Kd: 1 Koff: 1 Kon: 1
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
IC50: 3
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Kd: 1 Koff: 1 Kon: 1
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
IC50: 9 Kd: 10 EC50: 54 Koff: 10 Kon: 10
Hepatitis C virus genotype 1b (isolate BK) (HCV)
IC50: 7 EC50: 62
Hepatitis C virus genotype 1b (strain HC-J4) (HCV)
IC50: 7 Kd: 1 Koff: 1 Kon: 1
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
EC50: 36
Hepatitis C virus genotype 1b (isolate Japanese) (HCV)
IC50: 5
Hepatitis C virus
IC50: 8
Saccharomyces cerevisiae (Yeast)
Ki: 8 IC50: 9
Saccharomyces cerevisiae (Yeast)
IC50: 1
Pseudomonas aeruginosa
IC50: 41
Sus scrofa
Ki: 81
Vibrio cholerae (g-Proteobacteria)
IC50: 2
Human
Ki: 6
Human
Ki: 309 IC50: 1367 EC50: 174
Mus musculus
IC50: 101 EC50: 7
Rattus norvegicus
IC50: 95 Kd: 13 EC50: 9
Macaca mulatta
IC50: 1
Human
Ki: 116 IC50: 411 Kd: 10 EC50: 2359 Koff: 4
Rattus norvegicus
Ki: 2 IC50: 51 EC50: 52
Mus musculus
IC50: 2 EC50: 11
Macaca fascicularis
EC50: 4
Shiitake mushroom
IC50: 3
Aspergillus niger
Ki: 1 IC50: 1
Rhizopus oryzae
Ki: 1 IC50: 1
Saccharomyces cerevisiae S288c
Ki: 4 IC50: 3
Human
Ki: 1383 IC50: 3848 Kd: 13 EC50: 1508
MOUSE
Ki: 1 IC50: 3 Kd: 4 EC50: 24
RAT
Ki: 28 IC50: 192 EC50: 112
Canis lupus familiaris
Ki: 1 IC50: 4 EC50: 1
Sus scrofa
IC50: 4
Trypanosoma cruzi (strain CL Brener)
Ki: 2 IC50: 35
Rattus norvegicus
Kd: 9 EC50: 8
Human
IC50: 88 Kd: 14 EC50: 1
Mus musculus
Kd: 9 EC50: 62
Pseudomonas aeruginosa
IC50: 14
Plasmodium falciparum
IC50: 94
Oryctolagus cuniculus
Ki: 1
Human
Ki: 294 IC50: 321 Kd: 29 EC50: 5
Rattus norvegicus
Ki: 10 IC50: 52
Streptococcus pneumoniae
IC50: 4
Lactobacillus fermentum
Ki: 4
Helicobacter pylori J99
IC50: 74
Enterococcus faecalis
IC50: 33
Helicobacter pylori
Ki: 1 IC50: 21 Kd: 3
Xenopus laevis
EC50: 3
Rattus norvegicus (Rat)
IC50: 62
Rattus norvegicus (Rat)
Ki: 2 IC50: 2
Rattus norvegicus (Rat)
Ki: 433 IC50: 496 Kd: 10 EC50: 1
Rattus norvegicus (Rat)
Ki: 1 IC50: 2
Rattus norvegicus (Rat)
Ki: 73 IC50: 134 EC50: 3
Rattus norvegicus (Rat)
Ki: 1 IC50: 2
Rattus norvegicus (Rat)
IC50: 53
Rattus norvegicus (Rat)
Ki: 1 IC50: 2
Human
Ki: 142 IC50: 29 Kd: 4 EC50: 293
Rattus norvegicus
Ki: 101 IC50: 9 Kd: 1 EC50: 34
RAT
Ki: 169 IC50: 8 EC50: 31
Human
Ki: 57 IC50: 6 EC50: 28
Rattus norvegicus
Ki: 43 IC50: 7 EC50: 25
Human
Ki: 44 IC50: 4 EC50: 167
Rattus norvegicus (Rat)
IC50: 29
Pyrococcus horikoshii (strain ATCC 700860 / DSM 12428 / JCM 9974 /NBRC 100139 / OT-3)
Kd: 3
Onchocerca volvulus
Ki: 1
Escherichia coli
Ki: 4
Oryza sativa
IC50: 1
Escherichia coli (strain K12)
Ki: 7 IC50: 7
Salmonella typhimurium
Ki: 1
Glycine max
Ki: 1
Saccharomyces cerevisiae (Baker's yeast)
Ki: 4 IC50: 4
Staphylococcus aureus
Ki: 11
Streptococcus pyogenes serotype M1
IC50: 38
Human
Ki: 1
Escherichia coli
Ki: 2 IC50: 2
Human
Ki: 4 IC50: 5
Saccharomyces cerevisiae
Ki: 1 IC50: 11
Plasmodium falciparum (isolate 3D7)
Ki: 1 IC50: 4
Rattus norvegicus
IC50: 2
Plasmodium falciparum
IC50: 3
Anopheles gambiae (African malaria mosquito)
IC50: 5
Sus scrofa
IC50: 1
Crithidia fasciculata
Ki: 25 IC50: 22
Plasmodium falciparum
IC50: 42
Mus musculus
Ki: 2 IC50: 3
Bombyx mori
Ki: 6 IC50: 6 Kd: 1 ITC: 4
Oryctolagus cuniculus (rabbit)
Ki: 291 IC50: 502 EC50: 2 Other: 4
Rattus norvegicus
IC50: 6
Plasmodium falciparum (isolate 3D7)
IC50: 35
Dictyostelium discoideum
IC50: 6
Human
Ki: 33 IC50: 249 EC50: 10
Dictyostelium discoideum
IC50: 6
Human
Ki: 33 IC50: 249 EC50: 10
Rattus norvegicus (rat)
IC50: 193 EC50: 1
Human
Ki: 1040 IC50: 3942 Kd: 194 EC50: 5515 Koff: 2
Bos taurus (cattle)
IC50: 98
Mus musculus
IC50: 11 Kd: 1 EC50: 3
Human
Kd: 5
Human herpesvirus 4 type 2
IC50: 835
Nipah virus
EC50: 7
Oryctolagus cuniculus
IC50: 1
Staphylococcus aureus
IC50: 48
Saccharomyces cerevisiae
Ki: 12
Macaca fascicularis (Crab-eating macaque) (Cynomolgus monkey)
IC50: 2
Human
Ki: 23 IC50: 149
Human
Ki: 3
Human
Ki: 2 IC50: 328 Kd: 71 Koff: 2 Kon: 2 ITC: 10
Saccharomyces cerevisiae
Ki: 7
Saccharomyces cerevisiae
Ki: 5
Human
Ki: 1 IC50: 55 Kd: 4
Human
Ki: 1 IC50: 416
Human
Ki: 12 IC50: 1
Aspergillus oryzae
IC50: 19

BDB Curated by BindingDB
EBI Curated by ChEMBL