BDBM50008071 5-methylfurmethide::CHEMBL92387::Trimethyl-(5-methyl-furan-2-ylmethyl)-ammonium

SMILES Cc1ccc(C[N+](C)(C)C)o1

InChI Key InChIKey=KOWVJDFMEZKDDT-UHFFFAOYSA-N

Data  7 KI  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50008071   

TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008071(5-methylfurmethide | CHEMBL92387 | Trimethyl-(5-me...)
Affinity DataKi:  955nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008071(5-methylfurmethide | CHEMBL92387 | Trimethyl-(5-me...)
Affinity DataKi:  6.17E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008071(5-methylfurmethide | CHEMBL92387 | Trimethyl-(5-me...)
Affinity DataKi:  6.31E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M4 receptor expressed in CHO cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008071(5-methylfurmethide | CHEMBL92387 | Trimethyl-(5-me...)
Affinity DataKi:  6.92E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008071(5-methylfurmethide | CHEMBL92387 | Trimethyl-(5-me...)
Affinity DataKi:  7.94E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor DM1(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50008071(5-methylfurmethide | CHEMBL92387 | Trimethyl-(5-me...)
Affinity DataKi:  1.23E+4nMAssay Description:Displacement of [3H]AF-DX 384 from Drosophila melanogaster mAChR by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor DM1(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50008071(5-methylfurmethide | CHEMBL92387 | Trimethyl-(5-me...)
Affinity DataKi:  1.49E+4nMAssay Description:Displacement of [3H]QNB from Drosophila melanogaster mAChR by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50008071(5-methylfurmethide | CHEMBL92387 | Trimethyl-(5-me...)
Affinity DataIC50:  1.41E+3nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50008071(5-methylfurmethide | CHEMBL92387 | Trimethyl-(5-me...)
Affinity DataIC50:  5.60nMAssay Description:Central presynaptic activity as effect on electrically evoked acetylcholine release from rat hippocampal slices (M2 model)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed