BDBM50318521 Ac-ARA-CONHMe::CHEMBL1084621

SMILES [#6]-[#7]-[#6](=O)-[#6@H](-[#6])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#7]-[#6](=O)-[#6@H](-[#6])-[#7]-[#6](-[#6])=O

InChI Key InChIKey=PYWIZEZTCCLSTR-QXEWZRGKSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50318521   

TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318521(Ac-ARA-CONHMe | CHEMBL1084621)
Affinity DataKi:  150nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50318521(Ac-ARA-CONHMe | CHEMBL1084621)
Affinity DataIC50:  700nMAssay Description:Binding affinity to WDR5 expressed in pLysS cells by optimized fluorescent polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed