BDBM156263 US9018217, [2-(5,7-Dimethyl-imidazo[1,2-a]pyrimidin-2-ylmethylsulfanyl)-4-phenyl-imidazol-1-yl]-acetonitrile::US9592230, [2-(5,7-Dimethyl-imidazo[1,2-a]pyrimidin-2-ylmethylsulfanyl)-4-phenyl-imidazol-1-yl]-acetonitrile

SMILES Cc1cc(C)n2cc(CSc3nc(cn3CC#N)-c3ccccc3)nc2n1

InChI Key InChIKey=ZZUNVRXZOYEJBS-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 156263   

LigandChemical structure of BindingDB Monomer ID 156263BDBM156263(US9018217, [2-(5,7-Dimethyl-imidazo[1,2-a]pyrimidi...)
Affinity DataIC50: 52nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 156263BDBM156263(US9018217, [2-(5,7-Dimethyl-imidazo[1,2-a]pyrimidi...)
Affinity DataIC50: 52nMAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2019
Entry Details
US Patent